IL107133A - Piperidine derivatives, their preparation and pharmaceutical preparations containing them - Google Patents
Piperidine derivatives, their preparation and pharmaceutical preparations containing themInfo
- Publication number
- IL107133A IL107133A IL107133A IL10713393A IL107133A IL 107133 A IL107133 A IL 107133A IL 107133 A IL107133 A IL 107133A IL 10713393 A IL10713393 A IL 10713393A IL 107133 A IL107133 A IL 107133A
- Authority
- IL
- Israel
- Prior art keywords
- alkyl
- disorder
- compound
- formula
- optionally substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9211551A FR2696177B1 (fr) | 1992-09-28 | 1992-09-28 | Dérivés de pipéridine, leur préparation et leur application en thérapeutique. |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL107133A0 IL107133A0 (en) | 1993-12-28 |
| IL107133A true IL107133A (en) | 1998-03-10 |
Family
ID=9433967
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL107133A IL107133A (en) | 1992-09-28 | 1993-09-27 | Piperidine derivatives, their preparation and pharmaceutical preparations containing them |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US5434169A (hu) |
| EP (1) | EP0591027A1 (hu) |
| JP (1) | JPH06211838A (hu) |
| KR (1) | KR940007020A (hu) |
| CN (1) | CN1087339A (hu) |
| AP (1) | AP424A (hu) |
| AU (1) | AU658533B2 (hu) |
| CA (1) | CA2107061A1 (hu) |
| CZ (1) | CZ282080B6 (hu) |
| DZ (1) | DZ1718A1 (hu) |
| FI (1) | FI934221A (hu) |
| FR (1) | FR2696177B1 (hu) |
| HU (2) | HUT65303A (hu) |
| IL (1) | IL107133A (hu) |
| MA (1) | MA22981A1 (hu) |
| MX (1) | MX9305932A (hu) |
| NO (1) | NO933435L (hu) |
| NZ (1) | NZ248776A (hu) |
| OA (1) | OA09840A (hu) |
| PL (1) | PL172860B1 (hu) |
| SK (1) | SK103193A3 (hu) |
| TN (1) | TNSN93107A1 (hu) |
| TW (1) | TW272190B (hu) |
| ZA (1) | ZA937156B (hu) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUP9900606A2 (hu) * | 1995-09-18 | 2000-03-28 | Glaxo Group Limited | 5-HT3 Receptor antagonisták mozgászavar kezelésére |
| WO1997039750A1 (en) * | 1996-04-19 | 1997-10-30 | The Regents Of The University Of California | Treatment of mood/affective disorders by glutamatergic upmodulators |
| FR2765221B1 (fr) * | 1997-06-25 | 1999-07-30 | Synthelabo | Derives de 4-[(1h-imidazol-4-yl)piperidin-1-yl]anilide, leur preparation et leur application en therapeutique |
| US6013654A (en) * | 1997-08-14 | 2000-01-11 | Pharmacia & Upjohn Company | Imidazo[1,2-A]pyridines for the treatment of CNS and cardiac diseases |
| GB9918425D0 (en) * | 1999-08-04 | 1999-10-06 | Novartis Ag | Organic compounds |
| US6887870B1 (en) * | 1999-10-12 | 2005-05-03 | Bristol-Myers Squibb Company | Heterocyclic sodium/proton exchange inhibitors and method |
| US7183305B2 (en) | 2003-11-11 | 2007-02-27 | Allergan, Inc. | Process for the synthesis of imidazoles |
| US7880017B2 (en) | 2003-11-11 | 2011-02-01 | Allergan, Inc. | Process for the synthesis of imidazoles |
| EP1917255A2 (en) * | 2005-07-29 | 2008-05-07 | F. Hoffmann-Roche AG | Indol-3-yl-carbonyl-piperidin and piperazin derivatives |
| FR2925902B1 (fr) * | 2008-01-02 | 2011-01-07 | Sanofi Aventis | DERIVES D'IMIDAZO°1,2-a!PYRIDINE-2-CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE |
| EP2379524A1 (en) * | 2008-12-18 | 2011-10-26 | Boehringer Ingelheim International GmbH | Serotonin 5-ht2b receptor inhibitors |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61210080A (ja) * | 1985-03-13 | 1986-09-18 | Chisso Corp | アルデヒドラクトンの製造法 |
| FR2579596B1 (fr) * | 1985-03-26 | 1987-11-20 | Inst Nat Sante Rech Med | (imidazolyl-4) piperidines, leur preparation et leur application en therapeutique |
| US5008390A (en) * | 1985-05-23 | 1991-04-16 | Smithkline Beckman Corporation | Compounds for preparing 6-phenyl-2,3-dihydroimidazo[2,1-b]-thiazoles and corresponding thiazines |
| IT1230703B (it) * | 1989-01-26 | 1991-10-29 | Luso Farmaco Inst | Derivati imidazolonici ad attivita' antiipertensiva, loro metodi di preparazione e composizioni farmaceutiche che li contengono. |
| US4925851A (en) * | 1989-05-23 | 1990-05-15 | Sandoz Pharmaceuticals Corp. | 2- or 4-substituted-[2-(1H-imidazol-1-yl)ethyl]piperidines |
| FR2671083B1 (fr) * | 1990-12-31 | 1994-12-23 | Inst Nat Sante Rech Med | Nouvelles 4-(4-imidazolyl) piperidines substituees en 1, leur preparation ainsi que leurs applications therapeutiques. |
-
1992
- 1992-09-28 FR FR9211551A patent/FR2696177B1/fr not_active Expired - Fee Related
-
1993
- 1993-09-17 TW TW082107634A patent/TW272190B/zh active
- 1993-09-20 EP EP93402281A patent/EP0591027A1/fr not_active Ceased
- 1993-09-27 IL IL107133A patent/IL107133A/en not_active IP Right Cessation
- 1993-09-27 HU HU9302727A patent/HUT65303A/hu unknown
- 1993-09-27 NO NO933435A patent/NO933435L/no unknown
- 1993-09-27 OA OA60417A patent/OA09840A/fr unknown
- 1993-09-27 TN TNTNSN93107A patent/TNSN93107A1/fr unknown
- 1993-09-27 CA CA002107061A patent/CA2107061A1/en not_active Abandoned
- 1993-09-27 KR KR1019930019850A patent/KR940007020A/ko not_active Application Discontinuation
- 1993-09-27 ZA ZA937156A patent/ZA937156B/xx unknown
- 1993-09-27 FI FI934221A patent/FI934221A/fi unknown
- 1993-09-27 JP JP5239571A patent/JPH06211838A/ja active Pending
- 1993-09-27 US US08/127,078 patent/US5434169A/en not_active Expired - Fee Related
- 1993-09-27 PL PL93300515A patent/PL172860B1/pl unknown
- 1993-09-27 MX MX9305932A patent/MX9305932A/es unknown
- 1993-09-27 NZ NZ248776A patent/NZ248776A/en unknown
- 1993-09-27 SK SK1031-93A patent/SK103193A3/sk unknown
- 1993-09-27 MA MA23294A patent/MA22981A1/fr unknown
- 1993-09-27 CN CN93118082A patent/CN1087339A/zh active Pending
- 1993-09-27 CZ CZ932015A patent/CZ282080B6/cs unknown
- 1993-09-27 AP APAP/P/1993/000575A patent/AP424A/en active
- 1993-09-27 AU AU48606/93A patent/AU658533B2/en not_active Ceased
- 1993-09-28 DZ DZ930106A patent/DZ1718A1/fr active
-
1995
- 1995-06-28 HU HU95P/P00490P patent/HU211249A9/hu unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR940007020A (ko) | 1994-04-26 |
| US5434169A (en) | 1995-07-18 |
| NZ248776A (en) | 1995-09-26 |
| FI934221A (fi) | 1994-03-29 |
| EP0591027A1 (fr) | 1994-04-06 |
| CA2107061A1 (en) | 1994-03-29 |
| AP9300575A0 (en) | 1993-10-31 |
| DZ1718A1 (fr) | 2002-02-17 |
| AU658533B2 (en) | 1995-04-13 |
| SK103193A3 (en) | 1994-08-10 |
| JPH06211838A (ja) | 1994-08-02 |
| TNSN93107A1 (fr) | 1994-03-17 |
| CN1087339A (zh) | 1994-06-01 |
| CZ282080B6 (cs) | 1997-05-14 |
| PL300515A1 (en) | 1994-04-05 |
| FR2696177A1 (fr) | 1994-04-01 |
| TW272190B (hu) | 1996-03-11 |
| MA22981A1 (fr) | 1994-04-01 |
| HUT65303A (en) | 1994-05-02 |
| OA09840A (fr) | 1994-08-15 |
| IL107133A0 (en) | 1993-12-28 |
| NO933435L (no) | 1994-03-29 |
| NO933435D0 (no) | 1993-09-27 |
| PL172860B1 (pl) | 1997-12-31 |
| MX9305932A (es) | 1994-04-29 |
| HU211249A9 (en) | 1995-11-28 |
| CZ9302015A3 (en) | 1994-04-13 |
| AP424A (en) | 1995-11-04 |
| AU4860693A (en) | 1994-04-14 |
| FR2696177B1 (fr) | 1995-05-12 |
| FI934221A0 (fi) | 1993-09-27 |
| HU9302727D0 (en) | 1993-12-28 |
| ZA937156B (en) | 1994-05-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| RH | Patent void |