IE910575A1 - Novel¹2,4,8-trisubstituted-3h-6h-1,4,5a,8a-tetraazaacenaphthylene-¹3,5-(4h)-diones - Google Patents

Novel¹2,4,8-trisubstituted-3h-6h-1,4,5a,8a-tetraazaacenaphthylene-¹3,5-(4h)-diones

Info

Publication number
IE910575A1
IE910575A1 IE057591A IE57591A IE910575A1 IE 910575 A1 IE910575 A1 IE 910575A1 IE 057591 A IE057591 A IE 057591A IE 57591 A IE57591 A IE 57591A IE 910575 A1 IE910575 A1 IE 910575A1
Authority
IE
Ireland
Prior art keywords
alkyl
compound
carbon atoms
hydrogen
formula
Prior art date
Application number
IE057591A
Other languages
English (en)
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of IE910575A1 publication Critical patent/IE910575A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16—Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IE057591A 1990-02-21 1991-02-20 Novel¹2,4,8-trisubstituted-3h-6h-1,4,5a,8a-tetraazaacenaphthylene-¹3,5-(4h)-diones IE910575A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/482,568 US5013737A (en) 1988-02-22 1990-02-21 2,4,8-Trisubstituted-3H,6H-1,4,5A,8A-tetraazaacenaphtylene-3,5-(4H)-diones and 2,4-8-trisubstituted-4,5-dihydro-5-thioxo-3H,6H-1,4,5A,8A-tetrazaacenaphthylen-3-ones

Publications (1)

Publication Number Publication Date
IE910575A1 true IE910575A1 (en) 1991-08-28

Family

ID=23916572

Family Applications (1)

Application Number Title Priority Date Filing Date
IE057591A IE910575A1 (en) 1990-02-21 1991-02-20 Novel¹2,4,8-trisubstituted-3h-6h-1,4,5a,8a-tetraazaacenaphthylene-¹3,5-(4h)-diones

Country Status (24)

Country Link
US (1) US5013737A (ja)
EP (1) EP0443312B1 (ja)
JP (1) JP3046851B2 (ja)
KR (1) KR0183395B1 (ja)
AT (1) ATE152723T1 (ja)
AU (1) AU640202B2 (ja)
CA (1) CA2036589A1 (ja)
CZ (1) CZ285584B6 (ja)
DE (1) DE69125962T2 (ja)
DK (1) DK0443312T3 (ja)
ES (1) ES2102371T3 (ja)
FI (1) FI93963C (ja)
GR (1) GR3024063T3 (ja)
HU (1) HUT60500A (ja)
IE (1) IE910575A1 (ja)
IL (1) IL97289A (ja)
NO (1) NO177749C (ja)
NZ (1) NZ237123A (ja)
PH (1) PH27464A (ja)
PL (1) PL166100B1 (ja)
PT (1) PT96805B (ja)
SG (1) SG47638A1 (ja)
SK (1) SK279997B6 (ja)
ZA (1) ZA911260B (ja)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2350642A1 (en) * 1998-11-12 2000-05-18 Neurocrine Biosciences, Inc. Crf receptor antagonists and methods relating thereto
CN1178941C (zh) * 1998-11-12 2004-12-08 纽罗克里恩生物科学有限公司 Crf受体拮抗剂以及与其有关的方法
WO2007109093A2 (en) * 2006-03-17 2007-09-27 Wyeth Pyrazolo[1,5-a]pyrimidine derivatives and methods of use thereof
US20070219183A1 (en) * 2006-03-17 2007-09-20 Wyeth Dihydropyrazolo[1,5-A]pyrimidine and dihydroimidazo[1,5-A]pyrimidine derivatives and methods of use thereof
KR200480580Y1 (ko) * 2015-09-30 2016-06-13 김영직 어린이용 우산

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4178449A (en) * 1978-04-17 1979-12-11 American Cyanamid Company Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines
US4236005A (en) * 1979-07-02 1980-11-25 American Cyanamid Company Imidazo[1,5-a]pyrimidines
US4281000A (en) * 1979-07-09 1981-07-28 American Cyanamid Company Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents
US4713383A (en) * 1984-10-01 1987-12-15 Ciba-Geigy Corporation Triazoloquinazoline compounds, and their methods of preparation, pharmaceutical compositions, and uses
US4614732A (en) * 1984-10-26 1986-09-30 Warner-Lambert Company N6 -acenaphthyl adenosines and analogs thereof
ATE99686T1 (de) * 1988-02-22 1994-01-15 American Cyanamid Co 5-(substituierte amino)-8-(phenyl oder substituierte phenyl)-3h,6h-1,4,5a,8atetraazaacenaphthylen-3-one.

Also Published As

Publication number Publication date
KR0183395B1 (ko) 1999-05-01
EP0443312B1 (en) 1997-05-07
AU640202B2 (en) 1993-08-19
FI93963C (fi) 1995-06-26
NO910686D0 (no) 1991-02-20
NO177749B (no) 1995-08-07
HU910584D0 (en) 1991-09-30
CS41991A3 (en) 1991-09-15
NZ237123A (en) 1994-07-26
EP0443312A3 (en) 1992-02-19
JP3046851B2 (ja) 2000-05-29
GR3024063T3 (en) 1997-10-31
FI93963B (fi) 1995-03-15
PT96805B (pt) 1998-07-31
NO910686L (no) 1991-08-22
EP0443312A2 (en) 1991-08-28
PL289157A1 (en) 1992-06-26
JPH04211086A (ja) 1992-08-03
ES2102371T3 (es) 1997-08-01
PH27464A (en) 1993-07-09
IL97289A (en) 1995-06-29
FI910816A0 (fi) 1991-02-20
PT96805A (pt) 1991-10-31
AU7122591A (en) 1991-08-22
ATE152723T1 (de) 1997-05-15
FI910816A (fi) 1991-08-22
NO177749C (no) 1995-11-15
CA2036589A1 (en) 1991-08-22
DK0443312T3 (da) 1997-11-17
SG47638A1 (en) 1998-04-17
HUT60500A (en) 1992-09-28
IL97289A0 (en) 1992-05-25
ZA911260B (en) 1992-10-28
US5013737A (en) 1991-05-07
PL166100B1 (pl) 1995-03-31
SK279997B6 (sk) 1999-06-11
DE69125962T2 (de) 1997-10-16
CZ285584B6 (cs) 1999-09-15
DE69125962D1 (de) 1997-06-12

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Legal Events

Date Code Title Description
FC9A Application refused sect. 31(1)