ID30235A - Senyawa bifenil dan analognya sebagai antagonis-antagonis integrin - Google Patents

Senyawa bifenil dan analognya sebagai antagonis-antagonis integrin

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Publication number
ID30235A
ID30235A IDW00200101362A ID20011362A ID30235A ID 30235 A ID30235 A ID 30235A ID W00200101362 A IDW00200101362 A ID W00200101362A ID 20011362 A ID20011362 A ID 20011362A ID 30235 A ID30235 A ID 30235A
Authority
ID
Indonesia
Prior art keywords
compounds
integrin antagonists
bifenyl
analogue
biphenyl
Prior art date
Application number
IDW00200101362A
Other languages
English (en)
Indonesian (id)
Inventor
Markus Albers
Klaus Urbahns
Andrea Vaupel
Michael Harter
Delf Schmidt
Beatrix Stelte Ludwig
Christoph Gerdes
Elke Stahl
Jorg Keldenich
Ulf Bruggeier
Klemens Lustig
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of ID30235A publication Critical patent/ID30235A/id

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/40—Acylated substituent nitrogen atom
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    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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IDW00200101362A 1998-12-16 1999-12-13 Senyawa bifenil dan analognya sebagai antagonis-antagonis integrin ID30235A (id)

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PA8557501A1 (es) 2001-11-12 2003-06-30 Pfizer Prod Inc Benzamida, heteroarilamida y amidas inversas
WO2003042190A1 (fr) 2001-11-12 2003-05-22 Pfizer Products Inc. Derives de n-adamantylalkyle benzamide en tant qu'antagonistes du recepteur p2x7
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DE69927050D1 (de) 2005-10-06
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