HUP0500870A2 - Nitrogéntartalmú heterociklusos melanokortin receptor ligandumok, az ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk - Google Patents

Nitrogéntartalmú heterociklusos melanokortin receptor ligandumok, az ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk

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Publication number
HUP0500870A2
HUP0500870A2 HU0500870A HUP0500870A HUP0500870A2 HU P0500870 A2 HUP0500870 A2 HU P0500870A2 HU 0500870 A HU0500870 A HU 0500870A HU P0500870 A HUP0500870 A HU P0500870A HU P0500870 A2 HUP0500870 A2 HU P0500870A2
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Hungary
Prior art keywords
receptor ligands
malanocortin
pharmaceutical compositions
rings
compositions containing
Prior art date
Application number
HU0500870A
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English (en)
Inventor
Adam Wieslaw Mazur
Xinrong Tian
Xiufeng Eric Hu
Frank Hallock Ebetino
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The Procter & Gamble Company
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Publication date
Application filed by The Procter & Gamble Company filed Critical The Procter & Gamble Company
Publication of HUP0500870A2 publication Critical patent/HUP0500870A2/hu
Publication of HUP0500870A3 publication Critical patent/HUP0500870A3/hu

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    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
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Abstract

A találmány tárgyát az általános képletű MC-3/MC-4 melanokortinreceptor ligandumok - ahol A korlátozott konformációjú gyűrűrendszer akövetkező csoportból: a) nemaromás karbociklikus gyűrűk, b) aromáskarbociklikus gyűrűk, c) nemaromás heterociklikus gyűrűk, d) aromásheterociklikus gyűrűk, ahol az illető gyűrűk 5-8 atomosak, W egy (II)általános képletű csoport, előnyösen (D)-4-fluor-fenilalanin, Yheteroatomot tartalmazó egység, és Z egy aromás gyűrűt tartalmazóegység - és gyógyszerészetileg elfogadható sóik, ezeket tartalmazó, azMC-3/MC-4 receptorok által közvetített betegségek és állapotokkezelésére szolgáló gyógyszerkészítmények képezik.
HU0500870A 2001-04-25 2002-04-24 Nitrogen containing heterocyclic malanocortin receptor ligands, pharmaceutical compositions containing them and their use HUP0500870A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28661001P 2001-04-25 2001-04-25
PCT/US2002/013340 WO2002085925A2 (en) 2001-04-25 2002-04-24 Melanocortin receptor ligands

Publications (2)

Publication Number Publication Date
HUP0500870A2 true HUP0500870A2 (hu) 2005-12-28
HUP0500870A3 HUP0500870A3 (en) 2008-03-28

Family

ID=23099366

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HU0500870A HUP0500870A3 (en) 2001-04-25 2002-04-24 Nitrogen containing heterocyclic malanocortin receptor ligands, pharmaceutical compositions containing them and their use

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US (3) US6911447B2 (hu)
EP (1) EP1390361A4 (hu)
JP (1) JP2005503342A (hu)
KR (2) KR100662309B1 (hu)
CN (1) CN1543461A (hu)
AR (1) AR035863A1 (hu)
AU (1) AU2002254744B2 (hu)
BR (1) BR0209193A (hu)
CA (1) CA2444599A1 (hu)
CZ (1) CZ20032806A3 (hu)
HU (1) HUP0500870A3 (hu)
IL (1) IL157969A0 (hu)
MA (1) MA27016A1 (hu)
MX (1) MXPA03009791A (hu)
NO (1) NO20034774L (hu)
NZ (1) NZ528262A (hu)
PE (1) PE20021087A1 (hu)
PL (1) PL373503A1 (hu)
RU (1) RU2277535C2 (hu)
SK (1) SK13222003A3 (hu)
WO (1) WO2002085925A2 (hu)
ZA (1) ZA200307439B (hu)

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