HUP0304054A2 - A kortikotropin-realising faktor (CRF) antagonistáiként alkalmazható kondenzált pirimidinek, eljárás az előállításukra és ezeket tartalmazó gyógyszerkészítmények - Google Patents

A kortikotropin-realising faktor (CRF) antagonistáiként alkalmazható kondenzált pirimidinek, eljárás az előállításukra és ezeket tartalmazó gyógyszerkészítmények Download PDF

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Publication number
HUP0304054A2
HUP0304054A2 HU0304054A HUP0304054A HUP0304054A2 HU P0304054 A2 HUP0304054 A2 HU P0304054A2 HU 0304054 A HU0304054 A HU 0304054A HU P0304054 A HUP0304054 A HU P0304054A HU P0304054 A2 HUP0304054 A2 HU P0304054A2
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HU
Hungary
Prior art keywords
methyl
phenyl
dihydro
group
pyrrolo
Prior art date
Application number
HU0304054A
Other languages
English (en)
Hungarian (hu)
Inventor
Anna Maria Capelli
Romano Di Fabio
Chiara Marchionni
Fabrizio Micheli
Alessandra Pasquarello
Benedetta Perini
Yves St-Denis
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0110570A external-priority patent/GB0110570D0/en
Priority claimed from GB0110569A external-priority patent/GB0110569D0/en
Priority claimed from GB0110567A external-priority patent/GB0110567D0/en
Priority claimed from GB0117401A external-priority patent/GB0117401D0/en
Priority claimed from GB0117420A external-priority patent/GB0117420D0/en
Priority claimed from GB0117399A external-priority patent/GB0117399D0/en
Priority claimed from GB0203201A external-priority patent/GB0203201D0/en
Priority claimed from GB0206834A external-priority patent/GB0206834D0/en
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of HUP0304054A2 publication Critical patent/HUP0304054A2/hu

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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • A61K51/041—Heterocyclic compounds
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    • A61K51/0459—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
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    • A61K51/0463—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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HU0304054A 2001-04-30 2002-04-30 A kortikotropin-realising faktor (CRF) antagonistáiként alkalmazható kondenzált pirimidinek, eljárás az előállításukra és ezeket tartalmazó gyógyszerkészítmények HUP0304054A2 (hu)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
GB0110570A GB0110570D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110569A GB0110569D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110567A GB0110567D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0117401A GB0117401D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117420A GB0117420D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117399A GB0117399D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0203201A GB0203201D0 (en) 2002-02-11 2002-02-11 Chemical compounds
GB0206834A GB0206834D0 (en) 2002-03-22 2002-03-22 Chemical compounds
PCT/GB2002/002029 WO2002088095A1 (en) 2001-04-30 2002-04-30 Fused pyrimidines as antagonists of the corticotropin releasing factor (crf)

Publications (1)

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HUP0304054A2 true HUP0304054A2 (hu) 2004-04-28

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HU0304054A HUP0304054A2 (hu) 2001-04-30 2002-04-30 A kortikotropin-realising faktor (CRF) antagonistáiként alkalmazható kondenzált pirimidinek, eljárás az előállításukra és ezeket tartalmazó gyógyszerkészítmények

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US (1) US7279474B2 (https=)
EP (1) EP1383747B1 (https=)
JP (1) JP2004528349A (https=)
KR (1) KR20040015206A (https=)
CN (1) CN1649848A (https=)
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DE (1) DE60225127T2 (https=)
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HU (1) HUP0304054A2 (https=)
IL (1) IL158062A0 (https=)
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US20040176400A1 (en) 2004-09-09
JP2004528349A (ja) 2004-09-16
ATE386727T1 (de) 2008-03-15
MXPA03009938A (es) 2005-09-07
PL366934A1 (en) 2005-02-07
IL158062A0 (en) 2004-03-28
CZ20032946A3 (en) 2004-05-12
ES2301633T3 (es) 2008-07-01
NO20034836D0 (no) 2003-10-29
DE60225127T2 (de) 2009-02-19
US7279474B2 (en) 2007-10-09
CA2446514A1 (en) 2002-11-07
DE60225127D1 (en) 2008-04-03
EP1383747A1 (en) 2004-01-28
AU2002253357B2 (en) 2006-08-24
CN1649848A (zh) 2005-08-03
AR033295A1 (es) 2003-12-10
EP1383747B1 (en) 2008-02-20
WO2002088095A1 (en) 2002-11-07
BR0209267A (pt) 2004-06-15
NO20034836L (no) 2003-10-29
KR20040015206A (ko) 2004-02-18

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