HUP0203596A3 - 3-methylene steroid derivative and pharmaceutical compositions containing them - Google Patents

3-methylene steroid derivative and pharmaceutical compositions containing them

Info

Publication number
HUP0203596A3
HUP0203596A3 HU0203596A HUP0203596A HUP0203596A3 HU P0203596 A3 HUP0203596 A3 HU P0203596A3 HU 0203596 A HU0203596 A HU 0203596A HU P0203596 A HUP0203596 A HU P0203596A HU P0203596 A3 HUP0203596 A3 HU P0203596A3
Authority
HU
Hungary
Prior art keywords
pharmaceutical compositions
compositions containing
steroid derivative
methylene steroid
methylene
Prior art date
Application number
HU0203596A
Other languages
English (en)
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of HUP0203596A2 publication Critical patent/HUP0203596A2/hu
Publication of HUP0203596A3 publication Critical patent/HUP0203596A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096—Alkynyl derivatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HU0203596A 1999-11-29 2000-11-23 3-methylene steroid derivative and pharmaceutical compositions containing them HUP0203596A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99204000 1999-11-29
PCT/EP2000/011787 WO2001040253A2 (en) 1999-11-29 2000-11-23 3-methylene steroid derivative for the treatment of autoimmune diseases

Publications (2)

Publication Number Publication Date
HUP0203596A2 HUP0203596A2 (hu) 2003-02-28
HUP0203596A3 true HUP0203596A3 (en) 2003-12-29

Family

ID=8240918

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0203596A HUP0203596A3 (en) 1999-11-29 2000-11-23 3-methylene steroid derivative and pharmaceutical compositions containing them

Country Status (30)

Country Link
US (2) US6579864B1 (hu)
EP (1) EP1240179B1 (hu)
JP (1) JP2003517472A (hu)
KR (1) KR100720326B1 (hu)
CN (1) CN1254479C (hu)
AR (1) AR033503A1 (hu)
AT (1) ATE319732T1 (hu)
AU (1) AU778773B2 (hu)
BR (1) BR0015950A (hu)
CA (1) CA2391096A1 (hu)
CO (1) CO5251432A1 (hu)
CY (1) CY1106088T1 (hu)
CZ (1) CZ20021837A3 (hu)
DE (1) DE60026608T2 (hu)
DK (1) DK1240179T3 (hu)
ES (1) ES2259624T3 (hu)
HK (1) HK1047595B (hu)
HU (1) HUP0203596A3 (hu)
IL (2) IL149412A0 (hu)
MX (1) MXPA02005334A (hu)
NO (1) NO323136B1 (hu)
NZ (1) NZ518756A (hu)
PE (1) PE20010980A1 (hu)
PL (1) PL355968A1 (hu)
PT (1) PT1240179E (hu)
RU (1) RU2248358C2 (hu)
SK (1) SK285398B6 (hu)
TW (1) TWI265167B (hu)
WO (1) WO2001040253A2 (hu)
ZA (1) ZA200203455B (hu)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI265167B (en) * 1999-11-29 2006-11-01 Akzo Nobel Nv 3-methylene steroid derivatives
WO2005117968A2 (en) 2004-04-14 2005-12-15 Genentech, Inc. Compositions and methods comprising an egfl7 antagonist for modulating vascular development

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1085035A (en) * 1913-05-01 1914-01-20 George H Greimann Ditch-digging machine.
US1171221A (en) * 1915-12-13 1916-02-08 Charles Ephriam Marion Combination-tool.
US3213117A (en) * 1963-07-03 1965-10-19 Syntex Corp Process for preparation of delta1(10)-5alpha-estren-17beta-ol-2-one and derivatives thereof
BE654772A (hu) * 1963-10-23
US4701450A (en) * 1984-03-21 1987-10-20 Akzo N.V. Steroids for use as immunomodulators
EP0157739B1 (de) 1984-03-29 1987-08-12 Ciba-Geigy Ag Substituierte 1-Propanole, Verfahren zu deren Herstellung, Chlorameisensäureester und deren Verwendung
GB8513723D0 (en) * 1985-05-31 1985-07-03 Erba Farmitalia 11-beta substituted steroids
IE63051B1 (en) * 1989-03-18 1995-03-22 Akzo Nv Pharmaceutical composition which contains a pharmaceutically suitable carrier and the compound having the structure (7alpha, 17alpha)-17-Hydroxy-7-methyl-19-nor-17-pregn-5(10)-en-20-yn- 3-one
TWI265167B (en) * 1999-11-29 2006-11-01 Akzo Nobel Nv 3-methylene steroid derivatives

Also Published As

Publication number Publication date
KR100720326B1 (ko) 2007-05-22
SK7272002A3 (en) 2002-09-10
ATE319732T1 (de) 2006-03-15
PT1240179E (pt) 2006-05-31
AU2508701A (en) 2001-06-12
DE60026608T2 (de) 2006-12-28
CO5251432A1 (es) 2003-02-28
JP2003517472A (ja) 2003-05-27
WO2001040253A3 (en) 2002-05-02
EP1240179B1 (en) 2006-03-08
CN1254479C (zh) 2006-05-03
DK1240179T3 (da) 2006-07-03
TWI265167B (en) 2006-11-01
US20040043972A1 (en) 2004-03-04
ES2259624T3 (es) 2006-10-16
PL355968A1 (en) 2004-05-31
RU2248358C2 (ru) 2005-03-20
ZA200203455B (en) 2004-04-28
KR20030024656A (ko) 2003-03-26
AU778773B2 (en) 2004-12-23
NO20022521D0 (no) 2002-05-28
SK285398B6 (sk) 2007-01-04
HUP0203596A2 (hu) 2003-02-28
IL149412A (en) 2007-07-24
US6579864B1 (en) 2003-06-17
NO323136B1 (no) 2007-01-08
WO2001040253A2 (en) 2001-06-07
NZ518756A (en) 2004-05-28
IL149412A0 (en) 2002-11-10
PE20010980A1 (es) 2001-10-02
CA2391096A1 (en) 2001-06-07
MXPA02005334A (es) 2003-04-10
CN1402734A (zh) 2003-03-12
BR0015950A (pt) 2002-11-12
NO20022521L (no) 2002-05-28
CZ20021837A3 (cs) 2002-08-14
CY1106088T1 (el) 2011-06-08
DE60026608D1 (de) 2006-05-04
HK1047595A1 (en) 2003-02-28
EP1240179A2 (en) 2002-09-18
HK1047595B (zh) 2006-05-04
AR033503A1 (es) 2003-12-26

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Legal Events

Date Code Title Description
GB9A Succession in title

Owner name: N.V. ORGANON, NL

Free format text: FORMER OWNER(S): AKZO NOBEL N.V., NL