HRP20240525T1 - Pripravak na bazi lipida za oralnu primjenu antagonista bradikininskog b2-receptora - Google Patents

Pripravak na bazi lipida za oralnu primjenu antagonista bradikininskog b2-receptora Download PDF

Info

Publication number
HRP20240525T1
HRP20240525T1 HRP20240525TT HRP20240525T HRP20240525T1 HR P20240525 T1 HRP20240525 T1 HR P20240525T1 HR P20240525T T HRP20240525T T HR P20240525TT HR P20240525 T HRP20240525 T HR P20240525T HR P20240525 T1 HRP20240525 T1 HR P20240525T1
Authority
HR
Croatia
Prior art keywords
weight
propylene glycol
liquid pharmaceutical
pharmaceutical preparation
liquid
Prior art date
Application number
HRP20240525TT
Other languages
English (en)
Croatian (hr)
Inventor
Christoph Gibson
Original Assignee
Pharvaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharvaris Gmbh filed Critical Pharvaris Gmbh
Publication of HRP20240525T1 publication Critical patent/HRP20240525T1/hr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816Wall or shell material
    • A61K9/4825Proteins, e.g. gelatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HRP20240525TT 2021-08-05 2022-08-05 Pripravak na bazi lipida za oralnu primjenu antagonista bradikininskog b2-receptora HRP20240525T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP21189990 2021-08-05
EP22760986.4A EP4203919B1 (en) 2021-08-05 2022-08-05 Lipid-based composition for oral administration of bradykinin b2-receptor antagonists
PCT/EP2022/072049 WO2023012322A1 (en) 2021-08-05 2022-08-05 Lipid-based composition for oral administration of bradykinin b2-receptor antagonists

Publications (1)

Publication Number Publication Date
HRP20240525T1 true HRP20240525T1 (hr) 2024-07-05

Family

ID=77226756

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20240525TT HRP20240525T1 (hr) 2021-08-05 2022-08-05 Pripravak na bazi lipida za oralnu primjenu antagonista bradikininskog b2-receptora

Country Status (25)

Country Link
US (1) US20240350418A1 (https=)
EP (1) EP4203919B1 (https=)
JP (1) JP2024528195A (https=)
KR (1) KR20240039185A (https=)
CN (1) CN118076342B (https=)
AU (1) AU2022323749A1 (https=)
BR (1) BR112024002215A2 (https=)
CA (1) CA3227476A1 (https=)
CO (1) CO2024001171A2 (https=)
DK (1) DK4203919T3 (https=)
ES (1) ES2978563T3 (https=)
FI (1) FI4203919T3 (https=)
HR (1) HRP20240525T1 (https=)
HU (1) HUE066306T2 (https=)
IL (1) IL310321A (https=)
LT (1) LT4203919T (https=)
MA (1) MA61123B1 (https=)
MX (1) MX2024001711A (https=)
PL (1) PL4203919T3 (https=)
PT (1) PT4203919T (https=)
RS (1) RS65427B1 (https=)
SI (1) SI4203919T1 (https=)
SM (1) SMT202400157T1 (https=)
WO (1) WO2023012322A1 (https=)
ZA (1) ZA202401504B (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117224522B (zh) * 2023-11-15 2024-02-23 北京协和药厂有限公司 药物组合物及其制备方法、药物制剂

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2218554T3 (es) 1994-10-27 2004-11-16 Fujisawa Pharmaceutical Co., Ltd. Piridopirimidonas, quinolinas y n-heterociclos condensados que son antagonistas de bradiquinina.
FR2737892B1 (fr) 1995-08-17 1997-10-24 Fournier Ind & Sante Nouveaux composes de benzenesulfonamide, procede de preparation et utilisation en therapeutique
GB9602029D0 (en) 1996-02-01 1996-04-03 Fujisawa Pharmaceutical Co New heterocyclic compounds
DE19609827A1 (de) 1996-03-13 1997-09-18 Hoechst Ag Aminoalkyl- und Acylaminoalkylether, Verfahren zu deren Herstellung und ihre Verwendung als Bradykinin-Rezeptorantagonisten
DE19610784A1 (de) 1996-03-19 1997-09-25 Hoechst Ag Fluoralkyl- und Fluoralkoxysubstituierte heterocyclische Bradykinin-Antagonisten, Verfahren zu ihrer Herstellung und ihre Verwendung
AUPN952696A0 (en) 1996-04-29 1996-05-23 Fujisawa Pharmaceutical Co., Ltd. New heterocyclic compounds
DE19712960A1 (de) 1997-03-27 1998-10-01 Hoechst Ag Benzyloxy-substituierte, anellierte N-Heterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Bradykininrezeptorantagonisten
JP2002517461A (ja) 1998-06-08 2002-06-18 アドバンスド メディスン インコーポレーテッド ブラジキニンアンタゴニスト
CA2364178C (en) 2000-12-05 2006-01-10 Yasuhiro Katsu N-benzenesulfonyl l-proline compounds as bradykinin antagonists
WO2008055146A2 (en) * 2006-10-31 2008-05-08 Wyeth Formulations of phospholipase enzyme inhibitors
TWI407960B (zh) 2007-03-23 2013-09-11 Jerini Ag 小分子緩激肽b2受體調節劑
AR073304A1 (es) 2008-09-22 2010-10-28 Jerini Ag Moduladores del receptor de bradiquinina b2 de molecula pequena
WO2014159637A1 (en) 2013-03-14 2014-10-02 Shire Human Genetic Therapies, Inc. Methods of treating b2-bradykinin receptor mediated angioedema
AR113839A1 (es) 2017-11-24 2020-06-17 Pharvaris B V Antagonistas del receptor b2 de bradiquinina

Also Published As

Publication number Publication date
ES2978563T3 (es) 2024-09-16
PL4203919T3 (pl) 2024-06-10
FI4203919T3 (fi) 2024-05-03
KR20240039185A (ko) 2024-03-26
SI4203919T1 (sl) 2024-08-30
RS65427B1 (sr) 2024-05-31
US20240350418A1 (en) 2024-10-24
PT4203919T (pt) 2024-04-23
EP4203919A1 (en) 2023-07-05
EP4203919B1 (en) 2024-01-31
CN118076342B (zh) 2025-08-05
HUE066306T2 (hu) 2024-07-28
ZA202401504B (en) 2025-06-25
MA61123B1 (fr) 2024-06-28
CA3227476A1 (en) 2023-02-09
CO2024001171A2 (es) 2024-05-20
CN118076342A (zh) 2024-05-24
JP2024528195A (ja) 2024-07-26
AU2022323749A1 (en) 2024-02-08
DK4203919T3 (da) 2024-04-29
BR112024002215A2 (pt) 2024-04-30
SMT202400157T1 (it) 2024-05-14
IL310321A (en) 2024-03-01
WO2023012322A1 (en) 2023-02-09
MX2024001711A (es) 2024-03-05
TW202320774A (zh) 2023-06-01
LT4203919T (lt) 2024-05-10

Similar Documents

Publication Publication Date Title
ES2866933T3 (es) Regímenes de dosificación de amisulprida para tratar náuseas y vómitos
ES2496099T3 (es) El uso de amisulprida para el tratamiento de náuseas y vómitos inducidos por la quimioterapia
HRP20090341T1 (hr) Mekane kapsule koje sadrže palonosetron hidroksiklorid s poboljšanom stabilnosti i bioraspoloživosti
JP3743449B2 (ja) 4,5−エポキシモルヒナン誘導体を含有する安定なソフトカプセル剤
US20040092428A1 (en) Oral pharmaceuticals formulation comprising paclitaxel, derivatives and methods of administration thereof
ES2640572T3 (es) Formulaciones parenterales mejoradas de agentes farmacéuticos lipófilos y procedimientos de preparación y uso de las mismas
JP2005002123A5 (https=)
BR112014028602B1 (pt) Formulação líquida não aquosa oralmente biodisponível para administração oral
RU2001129362A (ru) Композиция, включающая ундеканоат тестостерона и касторовое масло
KR950031069A (ko) 골손실의 억제 및 혈청 콜레스테롤의 강하 방법
BRPI0008228B1 (pt) composição farmacêutica contendo n-benzoil estaurosporina e agentes solubilizantes
SA90100287B1 (ar) كبسولات صيدلية تحتوي على رانيتيدين
HRP20240525T1 (hr) Pripravak na bazi lipida za oralnu primjenu antagonista bradikininskog b2-receptora
PT1392318E (pt) 15-ceto-prostaglandinas para o tratamento de obstipação induzida por fármacos
JP3070930B2 (ja) 脳血管性疾患治療剤および抗炎症剤
ITMI962423A1 (it) Composizione farmaceutica orale ad attivita' antipiretica analgesica e infiammatoria
JP2024528195A5 (https=)
BR112020012157A2 (pt) composição farmacêutica oral de um antagonista de nk-1
US5063242A (en) 7-((substituted)amino)-8-((substituted)carbonyl)-methylamino-1-oxaspiro[4,5]decanes as diuretics antiinflammatory, and cerebrovascular agents
ES2472424T3 (es) Composición de mitotano automicroemulsionante
PT95422B (pt) Processo para a preparacao de composicoes farmaceuticas para o tratamento de psoriase incorporando compostos de acidos alquilfosforicos
Yedinak Use of Calcium Channel Antagonists for cardiovascular disease: This CE program reviews the role of calcium channel antagonists in managing certain diseases and compares agents
JP3748912B2 (ja) オーレオバシジン類の高濃度溶液製剤
JP2017513895A (ja) ブレクスピプラゾールとナルメフェンの組み合わせ剤及び物質関連障害を治療するためのその用途
JP2014208617A (ja) 医薬組成物