AU2022323749A1 - Lipid-based composition for oral administration of bradykinin b2-receptor antagonists - Google Patents

Lipid-based composition for oral administration of bradykinin b2-receptor antagonists Download PDF

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Publication number
AU2022323749A1
AU2022323749A1 AU2022323749A AU2022323749A AU2022323749A1 AU 2022323749 A1 AU2022323749 A1 AU 2022323749A1 AU 2022323749 A AU2022323749 A AU 2022323749A AU 2022323749 A AU2022323749 A AU 2022323749A AU 2022323749 A1 AU2022323749 A1 AU 2022323749A1
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AU
Australia
Prior art keywords
propylene glycol
pharmaceutical composition
liquid
liquid pharmaceutical
capsule
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
AU2022323749A
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English (en)
Inventor
Christoph Gibson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharvaris GmbH
Original Assignee
Pharvaris GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharvaris GmbH filed Critical Pharvaris GmbH
Publication of AU2022323749A1 publication Critical patent/AU2022323749A1/en
Pending legal-status Critical Current

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816Wall or shell material
    • A61K9/4825Proteins, e.g. gelatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2022323749A 2021-08-05 2022-08-05 Lipid-based composition for oral administration of bradykinin b2-receptor antagonists Pending AU2022323749A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP21189990 2021-08-05
EP21189990.1 2021-08-05
PCT/EP2022/072049 WO2023012322A1 (en) 2021-08-05 2022-08-05 Lipid-based composition for oral administration of bradykinin b2-receptor antagonists

Publications (1)

Publication Number Publication Date
AU2022323749A1 true AU2022323749A1 (en) 2024-02-08

Family

ID=77226756

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2022323749A Pending AU2022323749A1 (en) 2021-08-05 2022-08-05 Lipid-based composition for oral administration of bradykinin b2-receptor antagonists

Country Status (25)

Country Link
US (1) US20240350418A1 (https=)
EP (1) EP4203919B1 (https=)
JP (1) JP2024528195A (https=)
KR (1) KR20240039185A (https=)
CN (1) CN118076342B (https=)
AU (1) AU2022323749A1 (https=)
BR (1) BR112024002215A2 (https=)
CA (1) CA3227476A1 (https=)
CO (1) CO2024001171A2 (https=)
DK (1) DK4203919T3 (https=)
ES (1) ES2978563T3 (https=)
FI (1) FI4203919T3 (https=)
HR (1) HRP20240525T1 (https=)
HU (1) HUE066306T2 (https=)
IL (1) IL310321A (https=)
LT (1) LT4203919T (https=)
MA (1) MA61123B1 (https=)
MX (1) MX2024001711A (https=)
PL (1) PL4203919T3 (https=)
PT (1) PT4203919T (https=)
RS (1) RS65427B1 (https=)
SI (1) SI4203919T1 (https=)
SM (1) SMT202400157T1 (https=)
WO (1) WO2023012322A1 (https=)
ZA (1) ZA202401504B (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117224522B (zh) * 2023-11-15 2024-02-23 北京协和药厂有限公司 药物组合物及其制备方法、药物制剂

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2218554T3 (es) 1994-10-27 2004-11-16 Fujisawa Pharmaceutical Co., Ltd. Piridopirimidonas, quinolinas y n-heterociclos condensados que son antagonistas de bradiquinina.
FR2737892B1 (fr) 1995-08-17 1997-10-24 Fournier Ind & Sante Nouveaux composes de benzenesulfonamide, procede de preparation et utilisation en therapeutique
GB9602029D0 (en) 1996-02-01 1996-04-03 Fujisawa Pharmaceutical Co New heterocyclic compounds
DE19609827A1 (de) 1996-03-13 1997-09-18 Hoechst Ag Aminoalkyl- und Acylaminoalkylether, Verfahren zu deren Herstellung und ihre Verwendung als Bradykinin-Rezeptorantagonisten
DE19610784A1 (de) 1996-03-19 1997-09-25 Hoechst Ag Fluoralkyl- und Fluoralkoxysubstituierte heterocyclische Bradykinin-Antagonisten, Verfahren zu ihrer Herstellung und ihre Verwendung
AUPN952696A0 (en) 1996-04-29 1996-05-23 Fujisawa Pharmaceutical Co., Ltd. New heterocyclic compounds
DE19712960A1 (de) 1997-03-27 1998-10-01 Hoechst Ag Benzyloxy-substituierte, anellierte N-Heterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Bradykininrezeptorantagonisten
JP2002517461A (ja) 1998-06-08 2002-06-18 アドバンスド メディスン インコーポレーテッド ブラジキニンアンタゴニスト
CA2364178C (en) 2000-12-05 2006-01-10 Yasuhiro Katsu N-benzenesulfonyl l-proline compounds as bradykinin antagonists
WO2008055146A2 (en) * 2006-10-31 2008-05-08 Wyeth Formulations of phospholipase enzyme inhibitors
TWI407960B (zh) 2007-03-23 2013-09-11 Jerini Ag 小分子緩激肽b2受體調節劑
AR073304A1 (es) 2008-09-22 2010-10-28 Jerini Ag Moduladores del receptor de bradiquinina b2 de molecula pequena
WO2014159637A1 (en) 2013-03-14 2014-10-02 Shire Human Genetic Therapies, Inc. Methods of treating b2-bradykinin receptor mediated angioedema
AR113839A1 (es) 2017-11-24 2020-06-17 Pharvaris B V Antagonistas del receptor b2 de bradiquinina

Also Published As

Publication number Publication date
ES2978563T3 (es) 2024-09-16
PL4203919T3 (pl) 2024-06-10
FI4203919T3 (fi) 2024-05-03
KR20240039185A (ko) 2024-03-26
SI4203919T1 (sl) 2024-08-30
RS65427B1 (sr) 2024-05-31
US20240350418A1 (en) 2024-10-24
PT4203919T (pt) 2024-04-23
EP4203919A1 (en) 2023-07-05
EP4203919B1 (en) 2024-01-31
CN118076342B (zh) 2025-08-05
HUE066306T2 (hu) 2024-07-28
ZA202401504B (en) 2025-06-25
MA61123B1 (fr) 2024-06-28
CA3227476A1 (en) 2023-02-09
CO2024001171A2 (es) 2024-05-20
CN118076342A (zh) 2024-05-24
JP2024528195A (ja) 2024-07-26
DK4203919T3 (da) 2024-04-29
BR112024002215A2 (pt) 2024-04-30
SMT202400157T1 (it) 2024-05-14
IL310321A (en) 2024-03-01
WO2023012322A1 (en) 2023-02-09
MX2024001711A (es) 2024-03-05
TW202320774A (zh) 2023-06-01
LT4203919T (lt) 2024-05-10
HRP20240525T1 (hr) 2024-07-05

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