ES2978563T3 - Composición lipídica para la administración oral de antagonistas del receptor de bradicinina B2 - Google Patents

Composición lipídica para la administración oral de antagonistas del receptor de bradicinina B2 Download PDF

Info

Publication number
ES2978563T3
ES2978563T3 ES22760986T ES22760986T ES2978563T3 ES 2978563 T3 ES2978563 T3 ES 2978563T3 ES 22760986 T ES22760986 T ES 22760986T ES 22760986 T ES22760986 T ES 22760986T ES 2978563 T3 ES2978563 T3 ES 2978563T3
Authority
ES
Spain
Prior art keywords
weight
propylene glycol
liquid
pharmaceutical composition
liquid pharmaceutical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
ES22760986T
Other languages
English (en)
Spanish (es)
Inventor
Christoph Gibson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharvaris GmbH
Original Assignee
Pharvaris GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharvaris GmbH filed Critical Pharvaris GmbH
Application granted granted Critical
Publication of ES2978563T3 publication Critical patent/ES2978563T3/es
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816Wall or shell material
    • A61K9/4825Proteins, e.g. gelatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES22760986T 2021-08-05 2022-08-05 Composición lipídica para la administración oral de antagonistas del receptor de bradicinina B2 Active ES2978563T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP21189990 2021-08-05
PCT/EP2022/072049 WO2023012322A1 (en) 2021-08-05 2022-08-05 Lipid-based composition for oral administration of bradykinin b2-receptor antagonists

Publications (1)

Publication Number Publication Date
ES2978563T3 true ES2978563T3 (es) 2024-09-16

Family

ID=77226756

Family Applications (1)

Application Number Title Priority Date Filing Date
ES22760986T Active ES2978563T3 (es) 2021-08-05 2022-08-05 Composición lipídica para la administración oral de antagonistas del receptor de bradicinina B2

Country Status (25)

Country Link
US (1) US20240350418A1 (https=)
EP (1) EP4203919B1 (https=)
JP (1) JP2024528195A (https=)
KR (1) KR20240039185A (https=)
CN (1) CN118076342B (https=)
AU (1) AU2022323749A1 (https=)
BR (1) BR112024002215A2 (https=)
CA (1) CA3227476A1 (https=)
CO (1) CO2024001171A2 (https=)
DK (1) DK4203919T3 (https=)
ES (1) ES2978563T3 (https=)
FI (1) FI4203919T3 (https=)
HR (1) HRP20240525T1 (https=)
HU (1) HUE066306T2 (https=)
IL (1) IL310321A (https=)
LT (1) LT4203919T (https=)
MA (1) MA61123B1 (https=)
MX (1) MX2024001711A (https=)
PL (1) PL4203919T3 (https=)
PT (1) PT4203919T (https=)
RS (1) RS65427B1 (https=)
SI (1) SI4203919T1 (https=)
SM (1) SMT202400157T1 (https=)
WO (1) WO2023012322A1 (https=)
ZA (1) ZA202401504B (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117224522B (zh) * 2023-11-15 2024-02-23 北京协和药厂有限公司 药物组合物及其制备方法、药物制剂

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2218554T3 (es) 1994-10-27 2004-11-16 Fujisawa Pharmaceutical Co., Ltd. Piridopirimidonas, quinolinas y n-heterociclos condensados que son antagonistas de bradiquinina.
FR2737892B1 (fr) 1995-08-17 1997-10-24 Fournier Ind & Sante Nouveaux composes de benzenesulfonamide, procede de preparation et utilisation en therapeutique
GB9602029D0 (en) 1996-02-01 1996-04-03 Fujisawa Pharmaceutical Co New heterocyclic compounds
DE19609827A1 (de) 1996-03-13 1997-09-18 Hoechst Ag Aminoalkyl- und Acylaminoalkylether, Verfahren zu deren Herstellung und ihre Verwendung als Bradykinin-Rezeptorantagonisten
DE19610784A1 (de) 1996-03-19 1997-09-25 Hoechst Ag Fluoralkyl- und Fluoralkoxysubstituierte heterocyclische Bradykinin-Antagonisten, Verfahren zu ihrer Herstellung und ihre Verwendung
AUPN952696A0 (en) 1996-04-29 1996-05-23 Fujisawa Pharmaceutical Co., Ltd. New heterocyclic compounds
DE19712960A1 (de) 1997-03-27 1998-10-01 Hoechst Ag Benzyloxy-substituierte, anellierte N-Heterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Bradykininrezeptorantagonisten
JP2002517461A (ja) 1998-06-08 2002-06-18 アドバンスド メディスン インコーポレーテッド ブラジキニンアンタゴニスト
CA2364178C (en) 2000-12-05 2006-01-10 Yasuhiro Katsu N-benzenesulfonyl l-proline compounds as bradykinin antagonists
WO2008055146A2 (en) * 2006-10-31 2008-05-08 Wyeth Formulations of phospholipase enzyme inhibitors
TWI407960B (zh) 2007-03-23 2013-09-11 Jerini Ag 小分子緩激肽b2受體調節劑
AR073304A1 (es) 2008-09-22 2010-10-28 Jerini Ag Moduladores del receptor de bradiquinina b2 de molecula pequena
WO2014159637A1 (en) 2013-03-14 2014-10-02 Shire Human Genetic Therapies, Inc. Methods of treating b2-bradykinin receptor mediated angioedema
AR113839A1 (es) 2017-11-24 2020-06-17 Pharvaris B V Antagonistas del receptor b2 de bradiquinina

Also Published As

Publication number Publication date
PL4203919T3 (pl) 2024-06-10
FI4203919T3 (fi) 2024-05-03
KR20240039185A (ko) 2024-03-26
SI4203919T1 (sl) 2024-08-30
RS65427B1 (sr) 2024-05-31
US20240350418A1 (en) 2024-10-24
PT4203919T (pt) 2024-04-23
EP4203919A1 (en) 2023-07-05
EP4203919B1 (en) 2024-01-31
CN118076342B (zh) 2025-08-05
HUE066306T2 (hu) 2024-07-28
ZA202401504B (en) 2025-06-25
MA61123B1 (fr) 2024-06-28
CA3227476A1 (en) 2023-02-09
CO2024001171A2 (es) 2024-05-20
CN118076342A (zh) 2024-05-24
JP2024528195A (ja) 2024-07-26
AU2022323749A1 (en) 2024-02-08
DK4203919T3 (da) 2024-04-29
BR112024002215A2 (pt) 2024-04-30
SMT202400157T1 (it) 2024-05-14
IL310321A (en) 2024-03-01
WO2023012322A1 (en) 2023-02-09
MX2024001711A (es) 2024-03-05
TW202320774A (zh) 2023-06-01
LT4203919T (lt) 2024-05-10
HRP20240525T1 (hr) 2024-07-05

Similar Documents

Publication Publication Date Title
ES2225600T3 (es) Composicion semi-solida de isotretinoina.
ES2892029T3 (es) Formulaciones de enzalutamida
ES2464367T3 (es) Composición Farmacéutica para un Inhibidor de Proteasa del Virus de la Hepatitis C
KR102593075B1 (ko) 셀렉시파그를 포함하는 약학 조성물
ES2451540T3 (es) Formas de dosificación oral de bendamustina
JP6276756B2 (ja) 1,1−ジメチルエチル[(1s)−1−{[(2s,4r)−4−(7−クロロ−4メトキシイソキノリン−1−イルオキシ)−2−({(1r,2s)−1−[(シクロプロピルスルホニル)カルバモイル]−2−エテニルシクロプロピル}カルバモイル)ピロリジン−1−イル]カルボニル}−2,2−ジメチルプロピル]カルバメートの可溶化カプセル製剤
ES2591352T3 (es) Composición de tacrolimus estabilizada
ES3018260T3 (en) Method for producing an apixaban granulate
KR20170008252A (ko) 사이클로포스파미드 액상 농축 제제
ES2978563T3 (es) Composición lipídica para la administración oral de antagonistas del receptor de bradicinina B2
WO2021108343A1 (en) Formulations comprising lipid-lowering and blood pressure-lowering drugs
ES2535106T3 (es) Composiciones farmacéuticas de rosuvastatina cálcica
US20120213855A1 (en) Dosage forms for weakly ionizable compounds
WO2008087076A1 (en) Pharmaceutical composition of improved stability containing taxane derivatives
ES2276110T3 (es) Formulacion farmaceutica que incluye un inhibidor de renina no peptidico y un tensioactivo.
JP2019502751A5 (https=)
WO2025229501A1 (es) Composición farmacéutica que comprende enalapril maleato, uso y proceso de preparación
ES3062067T3 (en) Solid composition comprising solubilised bradykinin b2-receptor antagonists
ES2946260T3 (es) Sistemas de dos componentes que comprenden ácido acetilsalicílico y una sal de fosfato
JP6014252B2 (ja) ネパデュタントを含有する小児用経口液体組成物
HK40088043A (en) Lipid-based composition for oral administration of bradykinin b2-receptor antagonists
HK40088043B (en) Lipid-based composition for oral administration of bradykinin b2-receptor antagonists
EA051972B1 (ru) Композиция на основе липидов для перорального применения антагонистов брадикининовых b2-рецепторов
ES2824818T3 (es) Cápsulas de gelatina blanda que comprenden una suspensión de tadalafilo
JP2022136160A (ja) 炭酸ランタンを含有する医薬組成物