HRP20210814T1 - Derivati piridokinazolina korisni kao inhibitori proteinskih kinaza - Google Patents

Derivati piridokinazolina korisni kao inhibitori proteinskih kinaza Download PDF

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Publication number
HRP20210814T1
HRP20210814T1 HRP20210814TT HRP20210814T HRP20210814T1 HR P20210814 T1 HRP20210814 T1 HR P20210814T1 HR P20210814T T HRP20210814T T HR P20210814TT HR P20210814 T HRP20210814 T HR P20210814T HR P20210814 T1 HRP20210814 T1 HR P20210814T1
Authority
HR
Croatia
Prior art keywords
pyrido
quinazoline
carboxamide
oxo
unbranched
Prior art date
Application number
HRP20210814TT
Other languages
English (en)
Croatian (hr)
Inventor
Guido Kurz
Juan CAMACHO GÓMEZ
Original Assignee
Oncostellae, S.L.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oncostellae, S.L. filed Critical Oncostellae, S.L.
Publication of HRP20210814T1 publication Critical patent/HRP20210814T1/hr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • F—MECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F24—HEATING; RANGES; VENTILATING
    • F24C—DOMESTIC STOVES OR RANGES ; DETAILS OF DOMESTIC STOVES OR RANGES, OF GENERAL APPLICATION
    • F24C7/00—Stoves or ranges heated by electric energy
    • F24C7/08—Arrangement or mounting of control or safety devices
    • F24C7/082—Arrangement or mounting of control or safety devices on ranges, e.g. control panels, illumination
    • F—MECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F24—HEATING; RANGES; VENTILATING
    • F24C—DOMESTIC STOVES OR RANGES ; DETAILS OF DOMESTIC STOVES OR RANGES, OF GENERAL APPLICATION
    • F24C7/00—Stoves or ranges heated by electric energy
    • F24C7/08—Arrangement or mounting of control or safety devices
    • F24C7/087—Arrangement or mounting of control or safety devices of electric circuits regulating heat
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Combustion & Propulsion (AREA)
  • Mechanical Engineering (AREA)
  • General Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HRP20210814TT 2017-06-01 2018-05-31 Derivati piridokinazolina korisni kao inhibitori proteinskih kinaza HRP20210814T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ES201730759 2017-06-01
EP18759146.6A EP3632912B1 (en) 2017-06-01 2018-05-31 Pyridoquinazoline derivatives useful as protein kinase inhibitors
PCT/ES2018/070396 WO2018220252A1 (es) 2017-06-01 2018-05-31 Derivados de piridoquinazolina eficaces como inhibidores de proteína quinasa

Publications (1)

Publication Number Publication Date
HRP20210814T1 true HRP20210814T1 (hr) 2021-06-25

Family

ID=61569288

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20210814TT HRP20210814T1 (hr) 2017-06-01 2018-05-31 Derivati piridokinazolina korisni kao inhibitori proteinskih kinaza

Country Status (21)

Country Link
US (1) US11021479B2 (enExample)
EP (1) EP3632912B1 (enExample)
JP (1) JP7110335B2 (enExample)
KR (1) KR102629854B1 (enExample)
CN (1) CN111247143B (enExample)
AU (1) AU2018278283B2 (enExample)
CY (1) CY1124087T1 (enExample)
DK (1) DK3632912T3 (enExample)
EA (1) EA037384B1 (enExample)
ES (1) ES2881960T3 (enExample)
HR (1) HRP20210814T1 (enExample)
HU (1) HUE054792T2 (enExample)
LT (1) LT3632912T (enExample)
MX (1) MX385475B (enExample)
PL (1) PL3632912T3 (enExample)
PT (1) PT3632912T (enExample)
RS (1) RS61833B1 (enExample)
SI (1) SI3632912T1 (enExample)
SM (1) SMT202100312T1 (enExample)
WO (1) WO2018220252A1 (enExample)
ZA (1) ZA201908372B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11978921B2 (en) 2020-01-31 2024-05-07 Lg Energy Solution, Ltd. Method of manufacturing separator-composite electrode comprising multilayer-structured inorganic layer and separator-composite electrode manufactured thereby

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4551460A (en) 1982-05-10 1985-11-05 Hoffmann-La Roche Inc. Pyrido[2,1-b]quinazoline derivatives useful as agents for treatment of allergic conditions and vascular disorders involving thrombosis
WO1998023617A1 (en) 1996-11-26 1998-06-04 American Cyanamid Company Hetero-biaryl-pyridoquinazolinone derivatives as anti-cancer agents
WO2005048953A2 (en) 2003-11-13 2005-06-02 Ambit Biosciences Corporation Amide derivatives as kinase modulators
AU2008345225A1 (en) * 2007-12-21 2009-07-09 University Of Rochester Method for altering the lifespan of eukaryotic organisms
KR101361027B1 (ko) 2008-11-28 2014-02-11 코와 가부시키가이샤 피리딘-3-카르복시아미드 유도체
EP3778600A1 (en) 2014-03-20 2021-02-17 The Johns Hopkins University Compounds which inhibit rna polymerase, compositions including such compounds, and their use

Also Published As

Publication number Publication date
SMT202100312T1 (it) 2021-07-12
EA201992793A1 (ru) 2020-03-26
US11021479B2 (en) 2021-06-01
EP3632912B1 (en) 2021-03-17
PT3632912T (pt) 2021-06-02
HUE054792T2 (hu) 2021-09-28
RS61833B1 (sr) 2021-06-30
CN111247143B (zh) 2022-07-05
MX385475B (es) 2025-03-18
EA037384B1 (ru) 2021-03-23
PL3632912T3 (pl) 2021-09-06
ZA201908372B (en) 2021-04-28
BR112019024892A2 (pt) 2020-06-16
US20200148676A1 (en) 2020-05-14
CA3066009A1 (en) 2018-12-06
KR102629854B1 (ko) 2024-01-25
JP2020521817A (ja) 2020-07-27
WO2018220252A1 (es) 2018-12-06
AU2018278283A1 (en) 2019-12-19
KR20200011990A (ko) 2020-02-04
SI3632912T1 (sl) 2021-08-31
JP7110335B2 (ja) 2022-08-01
MX2019014436A (es) 2020-02-10
CN111247143A (zh) 2020-06-05
EP3632912A1 (en) 2020-04-08
LT3632912T (lt) 2021-06-10
CY1124087T1 (el) 2022-05-27
AU2018278283B2 (en) 2021-06-17
DK3632912T3 (da) 2021-05-10
ES2881960T3 (es) 2021-11-30

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