HRP20170607T1 - Proizvodni postupak vortioksetina - Google Patents

Proizvodni postupak vortioksetina Download PDF

Info

Publication number
HRP20170607T1
HRP20170607T1 HRP20170607TT HRP20170607T HRP20170607T1 HR P20170607 T1 HRP20170607 T1 HR P20170607T1 HR P20170607T T HRP20170607T T HR P20170607TT HR P20170607 T HRP20170607 T HR P20170607T HR P20170607 T1 HRP20170607 T1 HR P20170607T1
Authority
HR
Croatia
Prior art keywords
process according
formula
compound
equivalents
piperazine
Prior art date
Application number
HRP20170607TT
Other languages
English (en)
Croatian (hr)
Inventor
Thomas Ruhland
Kim Lasse Christensen
Original Assignee
H. Lundbeck A/S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by H. Lundbeck A/S filed Critical H. Lundbeck A/S
Publication of HRP20170607T1 publication Critical patent/HRP20170607T1/hr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/02Iron compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Compounds Of Unknown Constitution (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
HRP20170607TT 2013-02-22 2014-02-20 Proizvodni postupak vortioksetina HRP20170607T1 (hr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201361767883P 2013-02-22 2013-02-22
DKPA201300104 2013-02-22
PCT/EP2014/053313 WO2014128207A1 (en) 2013-02-22 2014-02-20 Vortioxetine manufacturing process
EP14705524.8A EP2958903B1 (en) 2013-02-22 2014-02-20 Vortioxetine manufacturing process

Publications (1)

Publication Number Publication Date
HRP20170607T1 true HRP20170607T1 (hr) 2017-06-30

Family

ID=59215387

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20170607TT HRP20170607T1 (hr) 2013-02-22 2014-02-20 Proizvodni postupak vortioksetina

Country Status (37)

Country Link
US (1) US9353073B2 (enExample)
EP (1) EP2958903B1 (enExample)
JP (1) JP6464098B2 (enExample)
KR (1) KR102230628B1 (enExample)
CN (1) CN104995181B (enExample)
AP (1) AP2015008640A0 (enExample)
AU (1) AU2014220735B2 (enExample)
BR (1) BR112015019268B1 (enExample)
CA (1) CA2901821A1 (enExample)
CL (1) CL2015002309A1 (enExample)
CR (1) CR20150423A (enExample)
CY (1) CY1118883T1 (enExample)
DK (1) DK2958903T3 (enExample)
DO (1) DOP2015000187A (enExample)
EA (1) EA027756B1 (enExample)
ES (1) ES2625380T3 (enExample)
GE (1) GEP201706749B (enExample)
HR (1) HRP20170607T1 (enExample)
IL (1) IL240501B (enExample)
LT (1) LT2958903T (enExample)
MA (1) MA38338B1 (enExample)
ME (1) ME02671B (enExample)
MX (1) MX362355B (enExample)
MY (1) MY172337A (enExample)
PE (1) PE20151589A1 (enExample)
PH (1) PH12015501807B1 (enExample)
PL (1) PL2958903T3 (enExample)
PT (1) PT2958903T (enExample)
RS (1) RS55932B1 (enExample)
RU (1) RU2652265C2 (enExample)
SG (1) SG11201506651SA (enExample)
SI (1) SI2958903T1 (enExample)
SM (1) SMT201700238T1 (enExample)
TN (1) TN2015000335A1 (enExample)
UA (1) UA116236C2 (enExample)
WO (1) WO2014128207A1 (enExample)
ZA (1) ZA201506050B (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX340997B (es) 2010-08-18 2016-08-03 Samumed Llc Dicetonas e hidroxicetonas como activadores de la trayectoria de señalizacion de catenina.
SG11201506592SA (en) 2013-02-22 2015-09-29 Samumed Llc Gamma-diketones as wnt/beta -catenin signaling pathway activators
WO2016029021A1 (en) 2014-08-20 2016-02-25 Samumed, Llc Gamma-diketones for treatment and prevention of aging skin and wrinkles
WO2016125191A2 (en) 2015-02-04 2016-08-11 Mylan Laboratories Limited Processes for the preparation of vortioxetine hydrobromide
EP3274330A1 (en) 2015-03-26 2018-01-31 Cipla Limited Method for making serotonin reuptake inhibitors
CN106279065A (zh) * 2015-05-12 2017-01-04 北京深蓝海生物医药科技有限公司 一种氢溴酸沃替西汀的精制转晶方法
JO3456B1 (ar) 2015-05-13 2020-07-05 H Lundbeck As فيروتيوكسيتين بيروجلوتامات
CN109071374A (zh) * 2016-02-08 2018-12-21 Aaa化学公司 脂肪胺的芳基化
MA45532A (fr) 2016-07-01 2019-05-08 H Lundbeck As Schémas posologiques de la vortioxétine destinés à une apparition rapide de l'effet antidépresseur
US10519121B2 (en) 2016-12-30 2019-12-31 Apicore Us Llc Process and novel polymorphic form of vortioxetine and its pharmaceutically acceptable salts
EP3870292A4 (en) 2018-10-26 2022-11-09 The Research Foundation for The State University of New York COMBINATION OF SEROTONIN-SPECIFIC RESUPPUT INHIBITOR AND SEROTONIN 1A RECEPTOR PARTIAL AGONIST TO REDUCE L-DOPA-INDUCED DYSKINESIA
CN109912538B (zh) * 2019-01-22 2021-03-12 安徽赛乐普制药有限公司 一种抗抑郁药沃替西汀的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA81749C2 (uk) * 2001-10-04 2008-02-11 Х. Луннбек А/С Фенілпіперазинові похідні як інгібітори зворотного захоплення серотоніну
IL161966A0 (en) * 2001-12-20 2005-11-20 Lundbeck & Co As H Aryloxyphenyl and arylsulfanylphenyl
EA015287B1 (ru) * 2006-06-16 2011-06-30 Х. Лундбекк А/С 1-[2-(2,4-диметилфенилсульфанил)фенил]пиперазин в качестве соединения с сочетанием активности в отношении повторного захвата серотонина, 5-нти 5-нтдля лечения когнитивного нарушения
TW201033181A (en) * 2009-02-17 2010-09-16 Lundbeck & Co As H Purification of 1-[2-(2,4-dimethylphenylsulfanyl)phenyl]piperazine

Also Published As

Publication number Publication date
KR20150118146A (ko) 2015-10-21
RU2652265C2 (ru) 2018-04-27
GEP201706749B (en) 2017-10-10
RS55932B1 (sr) 2017-09-29
CN104995181A (zh) 2015-10-21
PT2958903T (pt) 2017-05-26
WO2014128207A1 (en) 2014-08-28
MA38338A1 (fr) 2016-09-30
HK1216098A1 (en) 2016-10-14
DK2958903T3 (en) 2017-05-15
US9353073B2 (en) 2016-05-31
EA027756B1 (ru) 2017-08-31
RU2015134407A (ru) 2017-03-28
EP2958903A1 (en) 2015-12-30
TN2015000335A1 (en) 2017-01-03
AU2014220735B2 (en) 2017-06-22
CL2015002309A1 (es) 2016-03-04
SMT201700238T1 (it) 2017-07-18
PH12015501807B1 (en) 2019-05-31
US20160009670A1 (en) 2016-01-14
MA38338B1 (fr) 2018-10-31
CN104995181B (zh) 2017-03-08
MY172337A (en) 2019-11-21
MX2015010656A (es) 2015-12-17
AU2014220735A1 (en) 2015-08-20
BR112015019268A2 (pt) 2020-01-28
MX362355B (es) 2019-01-14
DOP2015000187A (es) 2015-11-30
SI2958903T1 (sl) 2017-09-29
IL240501A0 (en) 2015-09-24
CY1118883T1 (el) 2018-01-10
JP2016509042A (ja) 2016-03-24
ZA201506050B (en) 2017-08-30
SG11201506651SA (en) 2015-09-29
BR112015019268B1 (pt) 2023-01-10
PH12015501807A1 (en) 2015-11-09
KR102230628B1 (ko) 2021-03-22
PE20151589A1 (es) 2015-12-03
CA2901821A1 (en) 2014-08-28
LT2958903T (lt) 2017-08-25
EA201591349A1 (ru) 2015-12-30
IL240501B (en) 2018-08-30
CR20150423A (es) 2015-10-20
UA116236C2 (uk) 2018-02-26
EP2958903B1 (en) 2017-04-12
ME02671B (me) 2017-06-20
AP2015008640A0 (en) 2015-08-31
JP6464098B2 (ja) 2019-02-06
PL2958903T3 (pl) 2017-08-31
ES2625380T3 (es) 2017-07-19

Similar Documents

Publication Publication Date Title
HRP20170607T1 (hr) Proizvodni postupak vortioksetina
Wang et al. Electrochemical intramolecular dehydrogenative C–S bond formation for the synthesis of benzothiazoles
US8536371B2 (en) Carbon dioxide scrubbing using ionic materials
HRP20201480T1 (hr) Derivati indolinona i postupak za njihovu proizvodnju
Li et al. Synthesis of dioctyl phthalate using acid functionalized ionic liquid as catalyst
Sharma et al. Effects of anions on absorption capacity of carbon dioxide in acid functionalized ionic liquids
HRP20150885T1 (hr) Postupak za pripremu 4-{4-[({[4-kloro-3-(trifluorometil)-fenil]amino}karbonil)amino]-3-fluorofenoksi}-n-metilpiridin-2-karboksamida, njegovih soli i monohidrata
JP2016509042A5 (enExample)
CN105461654B (zh) 一种苯并噻唑离子液体及其制备方法和应用
HRP20211965T1 (hr) Novi selektivni inhibitori jak1 i njihova upotreba
CN105732717B (zh) 含笼状磷酸酯结构的咪唑离子液体型阻燃剂及其制备方法
HRP20200830T1 (hr) Postupak za pripremu n-boc-bifenil-alaninola
CN103709023B (zh) 3,5-二氯-2-戊酮的合成方法
Karimi-Jaberi et al. A mild, efficient, and environmentally friendly synthesis of N, N′-arylidene bisamides using B (HSO4) 3 under solvent-free conditions
HRP20100260T1 (hr) Postupak za proizvodnju stroncij ranelata i njegovih hidrata
HRP20200488T1 (hr) Proizvodnja 4,5,6,7-tetrahidroizozaksolo[5,4-c]piridin-3-ola
CN102584521A (zh) 一种氯代炔烃的合成方法
HRP20170023T1 (hr) Kristalni oblik pemirolasta
KR102127055B1 (ko) 레독스흐름전지용 전해액을 위한 알킬기 치환된 이온성 액체 제조방법
CN202748025U (zh) 遥控测距生成工程蓝图的装置
CN103304411B (zh) 一种丙二酸酯的制备方法
CN106831549B (zh) 一种抗过敏药物卡比沙明的不对称合成方法
JP2016184162A5 (enExample)
CN105315284A (zh) 阿拉格列汀中间体的制备方法
Chen et al. Studying of the basicity of ionic liquids by potentiometric titration