HRP20131002A2 - Lijekovi koji sadržavaju vardenafil hidroklorid trihidrat - Google Patents

Lijekovi koji sadržavaju vardenafil hidroklorid trihidrat Download PDF

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Publication number
HRP20131002A2
HRP20131002A2 HRP20131002AA HRP20131002A HRP20131002A2 HR P20131002 A2 HRP20131002 A2 HR P20131002A2 HR P20131002A A HRP20131002A A HR P20131002AA HR P20131002 A HRP20131002 A HR P20131002A HR P20131002 A2 HRP20131002 A2 HR P20131002A2
Authority
HR
Croatia
Prior art keywords
trihydrate
production
vardenafil
tablets
hydrochloride
Prior art date
Application number
HRP20131002AA
Other languages
English (en)
Croatian (hr)
Inventor
Peter Serno
Alfons Grunenberg
Andreas Ohm
Rainer Bellinghausen
Eimer Vollers
Jan-Olav Henck
Original Assignee
Bayer Intellectual Property Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29796385&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20131002(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Intellectual Property Gmbh filed Critical Bayer Intellectual Property Gmbh
Publication of HRP20131002A2 publication Critical patent/HRP20131002A2/hr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893—Tablet coating processes
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Reproductive Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Gynecology & Obstetrics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HRP20131002AA 2002-07-16 2003-07-03 Lijekovi koji sadržavaju vardenafil hidroklorid trihidrat HRP20131002A2 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10232113A DE10232113A1 (de) 2002-07-16 2002-07-16 Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel
PCT/EP2003/007093 WO2004006894A1 (de) 2002-07-16 2003-07-03 Vardenafil hydrochlorid trihydrat enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
HRP20131002A2 true HRP20131002A2 (hr) 2014-03-28

Family

ID=29796385

Family Applications (3)

Application Number Title Priority Date Filing Date
HRP20120418AA HRP20120418B1 (hr) 2002-07-16 2003-07-03 Lijekovi koji sadržavaju vardenafil hidroklorid trihidrat
HRP20050143AA HRP20050143B1 (hr) 2002-07-16 2003-07-03 Lijekovi koji sadržavaju vardenafil hidroklorid trihidrat
HRP20131002AA HRP20131002A2 (hr) 2002-07-16 2003-07-03 Lijekovi koji sadržavaju vardenafil hidroklorid trihidrat

Family Applications Before (2)

Application Number Title Priority Date Filing Date
HRP20120418AA HRP20120418B1 (hr) 2002-07-16 2003-07-03 Lijekovi koji sadržavaju vardenafil hidroklorid trihidrat
HRP20050143AA HRP20050143B1 (hr) 2002-07-16 2003-07-03 Lijekovi koji sadržavaju vardenafil hidroklorid trihidrat

Country Status (31)

Country Link
US (2) US8273876B2 (enExample)
EP (2) EP2272505B1 (enExample)
JP (2) JP5173113B2 (enExample)
KR (2) KR101552418B1 (enExample)
CN (2) CN1681481B (enExample)
AT (1) ATE538777T1 (enExample)
AU (1) AU2003249942B2 (enExample)
BR (1) BRPI0305559B8 (enExample)
CA (2) CA2492747C (enExample)
CU (1) CU23473B7 (enExample)
CY (2) CY1112460T1 (enExample)
DE (1) DE10232113A1 (enExample)
DK (2) DK1523303T3 (enExample)
EC (1) ECSP055541A (enExample)
ES (2) ES2378358T3 (enExample)
HR (3) HRP20120418B1 (enExample)
HU (1) HUE032362T2 (enExample)
IL (2) IL166162A (enExample)
LT (1) LT2272505T (enExample)
MA (1) MA27320A1 (enExample)
MX (1) MXPA05000554A (enExample)
NO (2) NO335434B1 (enExample)
NZ (1) NZ537698A (enExample)
PH (1) PH12012501171A1 (enExample)
PL (1) PL223341B1 (enExample)
PT (2) PT2272505T (enExample)
RU (1) RU2349306C2 (enExample)
SI (2) SI2272505T1 (enExample)
UA (1) UA85542C2 (enExample)
WO (1) WO2004006894A1 (enExample)
ZA (1) ZA200500268B (enExample)

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CZ307091B6 (cs) 2012-09-14 2018-01-10 Zentiva, K.S. Stabilní farmaceutický přípravek obsahující Vardenafil hydrochlorid
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BR112020012239A2 (pt) 2017-12-20 2020-11-24 Klaria Pharma Holding Ab método para preparar um filme mucoadesivo, e, filme mucoadesivo
JP7336241B2 (ja) * 2019-04-02 2023-08-31 富士化学工業株式会社 バルデナフィル含有錠剤の製造方法
CN110507626B (zh) * 2019-09-19 2020-08-18 山东创新药物研发有限公司 一种稳定的盐酸伐地那非三水合物药物组合物的制备方法
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