HRP20041167A2 - Hidroxy tetrahydro-naphthalenylurea derivatives - Google Patents

Hidroxy tetrahydro-naphthalenylurea derivatives

Info

Publication number
HRP20041167A2
HRP20041167A2 HR20041167A HRP20041167A HRP20041167A2 HR P20041167 A2 HRP20041167 A2 HR P20041167A2 HR 20041167 A HR20041167 A HR 20041167A HR P20041167 A HRP20041167 A HR P20041167A HR P20041167 A2 HRP20041167 A2 HR P20041167A2
Authority
HR
Croatia
Prior art keywords
tetrahydro
pain
hidroxy
useful
treatment
Prior art date
Application number
HR20041167A
Other languages
English (en)
Inventor
Yura Takeshi
Mogi Muneto
Urbahns Klaus
Fujishima Hiroshi
Masuda Tsutomu
Moriwaki Toshiya
Yoshida Nagahiro
Kokubo Toshio
Shiroo Masahiro
Tajimi Masaomi
Tsukimi Yasuhiro
Yamamoto Noriyuki
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0210512.0A external-priority patent/GB0210512D0/en
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of HRP20041167A2 publication Critical patent/HRP20041167A2/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/28Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/42Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by carboxyl groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/28Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/32Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/28Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/40Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by nitrogen atoms not being part of nitro or nitroso groups
HR20041167A 2002-05-08 2004-12-07 Hidroxy tetrahydro-naphthalenylurea derivatives HRP20041167A2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0210512.0A GB0210512D0 (en) 2002-05-08 2002-05-08 Tetrahydro-napthalene derivatives
GBGB0227262.3A GB0227262D0 (en) 2002-05-08 2002-11-21 Tetrahydro-naphthalene derivatives
PCT/EP2003/004395 WO2003095420A1 (en) 2002-05-08 2003-04-28 Hydroxy tetrahydro-naphthalenylurea derivatives

Publications (1)

Publication Number Publication Date
HRP20041167A2 true HRP20041167A2 (en) 2005-08-31

Family

ID=29422108

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20041167A HRP20041167A2 (en) 2002-05-08 2004-12-07 Hidroxy tetrahydro-naphthalenylurea derivatives

Country Status (21)

Country Link
US (1) US7612113B2 (ja)
EP (1) EP1506167B1 (ja)
JP (1) JP4335131B2 (ja)
CN (1) CN1307150C (ja)
AT (1) ATE371641T1 (ja)
AU (1) AU2003229734B2 (ja)
BR (1) BR0309940A (ja)
CA (1) CA2487238C (ja)
DE (1) DE60315973T2 (ja)
DK (1) DK1506167T3 (ja)
ES (1) ES2292959T3 (ja)
HK (1) HK1082946A1 (ja)
HR (1) HRP20041167A2 (ja)
IL (1) IL165004A (ja)
MX (1) MXPA04010938A (ja)
NO (1) NO20045359L (ja)
NZ (1) NZ536418A (ja)
PL (1) PL210288B1 (ja)
RU (1) RU2331635C2 (ja)
TW (1) TWI271396B (ja)
WO (1) WO2003095420A1 (ja)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004028440A2 (en) * 2002-09-24 2004-04-08 Bayer Healthcare Ag Vr1 antagonists for the treatment of urological disorders
ATE370118T1 (de) 2002-12-06 2007-09-15 Bayer Healthcare Ag Tetrahydronaphtalen-derivate
ATE404531T1 (de) * 2002-12-09 2008-08-15 Xention Ltd Tetrahydronaphtalen-derivate als vanilloid- rezeptor-antagonisten
WO2005035471A1 (ja) 2003-10-14 2005-04-21 Ajinomoto Co., Inc. エーテル誘導体
CA2542494A1 (en) * 2003-10-15 2005-05-06 Bayer Healthcare Ag Tetrahydro-naphthalene and urea derivatives
WO2005044802A2 (en) * 2003-11-08 2005-05-19 Bayer Healthcare Ag Tetrahydro-quinolinylurea derivatives as vrl antagonists
WO2005095329A1 (en) * 2004-03-31 2005-10-13 Pfizer Japan Inc. Substituted benzamide compounds as vr1 receptor antagonists
CA2599778A1 (en) * 2005-03-05 2006-09-14 Bayer Healthcare Ag Use of hydroxy tetrahydro-naphtalene derivates for the treatment of respiratory diseases
EA200702020A1 (ru) * 2005-03-19 2008-02-28 Эморпасифик Корпорейшн Новые соединения, их изомеры или фармацевтически приемлемые соли в качестве антагонистов ваниллоидных рецепторов и содержащие их фармацевтические композиции
DE102005017286B3 (de) * 2005-04-14 2006-12-28 Schering Ag Tetrahydronaphthalinderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer
DE102005023943A1 (de) 2005-05-20 2006-11-23 Grünenthal GmbH Pentafluorsulfanyl-substituierte Verbindung und deren Verwendung zur Herstellung von Arzneimitteln
CA2672196A1 (en) * 2006-12-20 2008-07-03 Abbott Laboratories Antagonists of the trpv1 receptor and uses thereof
WO2008096755A1 (ja) * 2007-02-07 2008-08-14 Nippon Suisan Kaisha, Ltd. バニロイド受容体(vr1)阻害剤及びその用途
DE102009055915A1 (de) * 2009-11-27 2011-06-01 Beiersdorf Ag Verwendung von Zingeron zur Herstellung kosmetischer oder dermatologischer Zubereitungen, welche auf der Haut ein Prickeln hervorrufen
WO2021039023A1 (ja) 2019-08-23 2021-03-04 持田製薬株式会社 ヘテロシクリデンアセトアミド誘導体の製造方法
CA3150748A1 (en) 2019-08-23 2021-03-04 Mochida Pharmaceutical Co., Ltd. Method for producing heterocyclidene acetamide derivative
DE102022104759A1 (de) 2022-02-28 2023-08-31 SCi Kontor GmbH Co-Kristall-Screening Verfahren, insbesondere zur Herstellung von Co-Kristallen

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9713484D0 (en) 1997-06-27 1997-09-03 Smithkline Beecham Plc Neuroprotective vanilloid compounds
US6333337B1 (en) * 1998-01-27 2001-12-25 Icagen, Inc. Potassium channel inhibitors
US6476076B1 (en) * 1999-02-22 2002-11-05 Pacific Corporation Vanilloid analogues containing resinferatoxin pharmacophores as potent vanilloid receptor agonists and analgesics, compositions and uses thereof
MXPA01010108A (es) 1999-04-07 2002-06-04 Sankyo Co Compuestos de derivados de amina.
US6294694B1 (en) 1999-06-04 2001-09-25 Wisconsin Alumni Research Foundation Matrix metalloproteinase inhibitors and method of using same
ATE370118T1 (de) * 2002-12-06 2007-09-15 Bayer Healthcare Ag Tetrahydronaphtalen-derivate
EP1493438A1 (en) * 2003-07-03 2005-01-05 Bayer HealthCare AG Vanilloid receptor (VR) inhibitors for treatment of Human Immunodeficiency Virus (HIV)-mediated pain states
CA2542494A1 (en) * 2003-10-15 2005-05-06 Bayer Healthcare Ag Tetrahydro-naphthalene and urea derivatives
ES2315716T3 (es) * 2003-11-08 2009-04-01 Bayer Healthcare Ag Derivados de amida, carbamato o urea biciclica como moduladores del receptor vanilloide.

Also Published As

Publication number Publication date
DK1506167T3 (da) 2008-01-02
MXPA04010938A (es) 2005-02-14
TW200404052A (en) 2004-03-16
JP4335131B2 (ja) 2009-09-30
RU2004136281A (ru) 2005-07-10
TWI271396B (en) 2007-01-21
WO2003095420A1 (en) 2003-11-20
CN1307150C (zh) 2007-03-28
JP2005524717A (ja) 2005-08-18
CA2487238A1 (en) 2003-11-20
US7612113B2 (en) 2009-11-03
BR0309940A (pt) 2005-02-09
PL210288B1 (pl) 2011-12-30
AU2003229734A1 (en) 2003-11-11
CA2487238C (en) 2011-03-22
AU2003229734B2 (en) 2009-02-19
IL165004A0 (en) 2005-12-18
DE60315973T2 (de) 2008-05-21
NZ536418A (en) 2006-04-28
ATE371641T1 (de) 2007-09-15
ES2292959T3 (es) 2008-03-16
CN1665778A (zh) 2005-09-07
RU2331635C2 (ru) 2008-08-20
NO20045359L (no) 2004-12-07
PL373257A1 (en) 2005-08-22
US20060258742A1 (en) 2006-11-16
EP1506167A1 (en) 2005-02-16
EP1506167B1 (en) 2007-08-29
DE60315973D1 (de) 2007-10-11
IL165004A (en) 2010-12-30
HK1082946A1 (en) 2006-06-23

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