HRP20020904A2 - Substituted 1-aminoalkyil-lactams and their use as muscarinic receptor antagonists - Google Patents

Substituted 1-aminoalkyil-lactams and their use as muscarinic receptor antagonists

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Publication number
HRP20020904A2
HRP20020904A2 HRP20020904A HRP20020904A2 HR P20020904 A2 HRP20020904 A2 HR P20020904A2 HR P20020904 A HRP20020904 A HR P20020904A HR P20020904 A2 HRP20020904 A2 HR P20020904A2
Authority
HR
Croatia
Prior art keywords
butyl
compound
methylethyl
ethyl
alkyl
Prior art date
Application number
Other languages
English (en)
Croatian (hr)
Inventor
Charles Alois Dvorak
Lawrence Emerson Fisher
Keena Lynn Green
Ralph New Harris Iii
Hans Maag
Anthony Prince
David Bruce Repke
Russell Stephen Stabler
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of HRP20020904A2 publication Critical patent/HRP20020904A2/hr

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    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/27—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
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HRP20020904 2000-05-25 2002-11-14 Substituted 1-aminoalkyil-lactams and their use as muscarinic receptor antagonists HRP20020904A2 (en)

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PL2300461T3 (pl) * 2008-05-01 2013-09-30 Vitae Pharmaceuticals Inc Cykliczne inhibitory dehydrogenazy 11beta-hydroksysteroidów 1
EP2687525B1 (en) * 2008-07-25 2015-09-23 Boehringer Ingelheim International GmbH Cyclic inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
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US20020004501A1 (en) 2002-01-10
CZ20024200A3 (cs) 2004-01-14
MA26906A1 (fr) 2004-12-20
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AU782191B2 (en) 2005-07-07
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CN1178922C (zh) 2004-12-08
ATE307806T1 (de) 2005-11-15
CA2409841A1 (en) 2001-11-29
US20060287293A1 (en) 2006-12-21
MY140835A (en) 2010-01-29
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US6667301B2 (en) 2003-12-23
NZ522411A (en) 2004-05-28
KR100544000B1 (ko) 2006-01-20
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JP4071000B2 (ja) 2008-04-02
UY26729A1 (es) 2001-12-28
HUP0302010A2 (hu) 2003-09-29
JP2003534330A (ja) 2003-11-18
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AR028624A1 (es) 2003-05-14
NO20025640D0 (no) 2002-11-22
US7094778B2 (en) 2006-08-22
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