HK1246653A1 - 奥那司酮延长释放组合物和方法 - Google Patents

奥那司酮延长释放组合物和方法 Download PDF

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Publication number
HK1246653A1
HK1246653A1 HK18106169.2A HK18106169A HK1246653A1 HK 1246653 A1 HK1246653 A1 HK 1246653A1 HK 18106169 A HK18106169 A HK 18106169A HK 1246653 A1 HK1246653 A1 HK 1246653A1
Authority
HK
Hong Kong
Prior art keywords
methods
onapristone
extended
release formulations
release compositions
Prior art date
Application number
HK18106169.2A
Other languages
English (en)
Chinese (zh)
Inventor
ZUKIWSKI Alexander
Proniuk Stefan
Original Assignee
Context Biopharma Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Context Biopharma Inc. filed Critical Context Biopharma Inc.
Publication of HK1246653A1 publication Critical patent/HK1246653A1/zh

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HK18106169.2A 2014-11-17 2015-11-16 奥那司酮延长释放组合物和方法 HK1246653A1 (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462080868P 2014-11-17 2014-11-17
US62/080,868 2014-11-17
PCT/US2015/060940 WO2016081383A1 (en) 2014-11-17 2015-11-16 Onapristone extended-release compositions and methods

Publications (1)

Publication Number Publication Date
HK1246653A1 true HK1246653A1 (zh) 2018-09-14

Family

ID=56014429

Family Applications (1)

Application Number Title Priority Date Filing Date
HK18106169.2A HK1246653A1 (zh) 2014-11-17 2015-11-16 奥那司酮延长释放组合物和方法

Country Status (11)

Country Link
US (3) US10786461B2 (enExample)
EP (1) EP3247362A4 (enExample)
JP (1) JP6655075B2 (enExample)
KR (1) KR20170084086A (enExample)
CN (2) CN106999501B (enExample)
AU (2) AU2015350241B2 (enExample)
CA (1) CA2966753A1 (enExample)
HK (1) HK1246653A1 (enExample)
MX (1) MX391191B (enExample)
RU (1) RU2017112748A (enExample)
WO (1) WO2016081383A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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CA3008422A1 (en) 2015-12-15 2017-06-22 Context Biopharma Inc. Amorphous onapristone compositions and methods of making the same
US20180148471A1 (en) 2016-11-30 2018-05-31 Arno Therapeutics, Inc. Methods for onapristone synthesis dehydration and deprotection

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Also Published As

Publication number Publication date
AU2015350241A1 (en) 2017-05-04
CN113559075A (zh) 2021-10-29
AU2015350241B2 (en) 2021-05-20
EP3247362A4 (en) 2018-10-10
MX391191B (es) 2025-03-21
CN106999501B (zh) 2021-08-13
CN106999501A (zh) 2017-08-01
US20230157960A1 (en) 2023-05-25
JP2017537883A (ja) 2017-12-21
JP6655075B2 (ja) 2020-02-26
KR20170084086A (ko) 2017-07-19
US11672762B2 (en) 2023-06-13
US20160166583A1 (en) 2016-06-16
CA2966753A1 (en) 2016-05-26
WO2016081383A1 (en) 2016-05-26
US20210220279A1 (en) 2021-07-22
AU2021218093A1 (en) 2021-09-09
RU2017112748A (ru) 2018-12-19
EP3247362A1 (en) 2017-11-29
MX2017005163A (es) 2018-01-18
RU2017112748A3 (enExample) 2019-06-26
US10786461B2 (en) 2020-09-29

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