MX391191B - Composiciones de liberación extendida de onapristona y métodos. - Google Patents

Composiciones de liberación extendida de onapristona y métodos.

Info

Publication number
MX391191B
MX391191B MX2017005163A MX2017005163A MX391191B MX 391191 B MX391191 B MX 391191B MX 2017005163 A MX2017005163 A MX 2017005163A MX 2017005163 A MX2017005163 A MX 2017005163A MX 391191 B MX391191 B MX 391191B
Authority
MX
Mexico
Prior art keywords
extended
onapristone
release
methods
formulations
Prior art date
Application number
MX2017005163A
Other languages
English (en)
Spanish (es)
Other versions
MX2017005163A (es
Inventor
Alexander Zukiwski
Stefan Proniuk
Original Assignee
Context Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Context Biopharma Inc filed Critical Context Biopharma Inc
Publication of MX2017005163A publication Critical patent/MX2017005163A/es
Publication of MX391191B publication Critical patent/MX391191B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MX2017005163A 2014-11-17 2015-11-16 Composiciones de liberación extendida de onapristona y métodos. MX391191B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462080868P 2014-11-17 2014-11-17
PCT/US2015/060940 WO2016081383A1 (en) 2014-11-17 2015-11-16 Onapristone extended-release compositions and methods

Publications (2)

Publication Number Publication Date
MX2017005163A MX2017005163A (es) 2018-01-18
MX391191B true MX391191B (es) 2025-03-21

Family

ID=56014429

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2017005163A MX391191B (es) 2014-11-17 2015-11-16 Composiciones de liberación extendida de onapristona y métodos.

Country Status (11)

Country Link
US (3) US10786461B2 (enExample)
EP (1) EP3247362A4 (enExample)
JP (1) JP6655075B2 (enExample)
KR (1) KR20170084086A (enExample)
CN (2) CN113559075A (enExample)
AU (2) AU2015350241B2 (enExample)
CA (1) CA2966753A1 (enExample)
HK (1) HK1246653A1 (enExample)
MX (1) MX391191B (enExample)
RU (1) RU2017112748A (enExample)
WO (1) WO2016081383A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113559075A (zh) 2014-11-17 2021-10-29 康泰科思特生物制药公司 奥那司酮延长释放组合物和方法
CA2998924A1 (en) 2015-09-25 2017-03-30 Context Biopharma Inc. Methods of making onapristone intermediates
JP2019503353A (ja) 2015-12-15 2019-02-07 コンテキスト・バイオファーマ・インコーポレイテッド 非晶質オナプリストン組成物およびそれを作製する方法
US20180148471A1 (en) 2016-11-30 2018-05-31 Arno Therapeutics, Inc. Methods for onapristone synthesis dehydration and deprotection

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Also Published As

Publication number Publication date
AU2015350241B2 (en) 2021-05-20
RU2017112748A3 (enExample) 2019-06-26
RU2017112748A (ru) 2018-12-19
CN113559075A (zh) 2021-10-29
EP3247362A1 (en) 2017-11-29
KR20170084086A (ko) 2017-07-19
MX2017005163A (es) 2018-01-18
AU2015350241A1 (en) 2017-05-04
WO2016081383A1 (en) 2016-05-26
EP3247362A4 (en) 2018-10-10
US10786461B2 (en) 2020-09-29
JP6655075B2 (ja) 2020-02-26
US20210220279A1 (en) 2021-07-22
JP2017537883A (ja) 2017-12-21
CN106999501B (zh) 2021-08-13
HK1246653A1 (zh) 2018-09-14
US20160166583A1 (en) 2016-06-16
US20230157960A1 (en) 2023-05-25
AU2021218093A1 (en) 2021-09-09
CN106999501A (zh) 2017-08-01
US11672762B2 (en) 2023-06-13
CA2966753A1 (en) 2016-05-26

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