RU2017112748A - Композиции онапристона пролонгированного действия и способы - Google Patents

Композиции онапристона пролонгированного действия и способы Download PDF

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Publication number
RU2017112748A
RU2017112748A RU2017112748A RU2017112748A RU2017112748A RU 2017112748 A RU2017112748 A RU 2017112748A RU 2017112748 A RU2017112748 A RU 2017112748A RU 2017112748 A RU2017112748 A RU 2017112748A RU 2017112748 A RU2017112748 A RU 2017112748A
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RU
Russia
Prior art keywords
pharmaceutical composition
onapristone
sustained
release pharmaceutical
day
Prior art date
Application number
RU2017112748A
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English (en)
Russian (ru)
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RU2017112748A3 (enExample
Inventor
Александер ЖУКИВСКИ
Стефан ПРОНЮК
Original Assignee
Арно Терапьютикс, Инк.
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Application filed by Арно Терапьютикс, Инк. filed Critical Арно Терапьютикс, Инк.
Publication of RU2017112748A publication Critical patent/RU2017112748A/ru
Publication of RU2017112748A3 publication Critical patent/RU2017112748A3/ru

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
RU2017112748A 2014-11-17 2015-11-16 Композиции онапристона пролонгированного действия и способы RU2017112748A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462080868P 2014-11-17 2014-11-17
US62/080,868 2014-11-17
PCT/US2015/060940 WO2016081383A1 (en) 2014-11-17 2015-11-16 Onapristone extended-release compositions and methods

Publications (2)

Publication Number Publication Date
RU2017112748A true RU2017112748A (ru) 2018-12-19
RU2017112748A3 RU2017112748A3 (enExample) 2019-06-26

Family

ID=56014429

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2017112748A RU2017112748A (ru) 2014-11-17 2015-11-16 Композиции онапристона пролонгированного действия и способы

Country Status (11)

Country Link
US (3) US10786461B2 (enExample)
EP (1) EP3247362A4 (enExample)
JP (1) JP6655075B2 (enExample)
KR (1) KR20170084086A (enExample)
CN (2) CN106999501B (enExample)
AU (2) AU2015350241B2 (enExample)
CA (1) CA2966753A1 (enExample)
HK (1) HK1246653A1 (enExample)
MX (1) MX391191B (enExample)
RU (1) RU2017112748A (enExample)
WO (1) WO2016081383A1 (enExample)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20170084086A (ko) 2014-11-17 2017-07-19 아르노 테라퓨틱스 인코포레이티드 오나프리스톤 연장-방출 조성물 및 방법
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JP2019503353A (ja) 2015-12-15 2019-02-07 コンテキスト・バイオファーマ・インコーポレイテッド 非晶質オナプリストン組成物およびそれを作製する方法
WO2018102369A1 (en) 2016-11-30 2018-06-07 Arno Therapeutics, Inc. Methods for onapristone synthesis dehydration and deprotection

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Also Published As

Publication number Publication date
MX2017005163A (es) 2018-01-18
EP3247362A4 (en) 2018-10-10
EP3247362A1 (en) 2017-11-29
AU2015350241B2 (en) 2021-05-20
AU2021218093A1 (en) 2021-09-09
US20160166583A1 (en) 2016-06-16
HK1246653A1 (zh) 2018-09-14
CN106999501A (zh) 2017-08-01
MX391191B (es) 2025-03-21
US20230157960A1 (en) 2023-05-25
JP6655075B2 (ja) 2020-02-26
RU2017112748A3 (enExample) 2019-06-26
JP2017537883A (ja) 2017-12-21
CN113559075A (zh) 2021-10-29
US20210220279A1 (en) 2021-07-22
US10786461B2 (en) 2020-09-29
US11672762B2 (en) 2023-06-13
CN106999501B (zh) 2021-08-13
KR20170084086A (ko) 2017-07-19
WO2016081383A1 (en) 2016-05-26
AU2015350241A1 (en) 2017-05-04
CA2966753A1 (en) 2016-05-26

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Effective date: 20191022