HK1210153A1 - Compound for preparing an intermediate compound of optically-active diazabicyclooctane derivative - Google Patents

Compound for preparing an intermediate compound of optically-active diazabicyclooctane derivative

Info

Publication number
HK1210153A1
HK1210153A1 HK15110896.7A HK15110896A HK1210153A1 HK 1210153 A1 HK1210153 A1 HK 1210153A1 HK 15110896 A HK15110896 A HK 15110896A HK 1210153 A1 HK1210153 A1 HK 1210153A1
Authority
HK
Hong Kong
Prior art keywords
compound
optically
preparing
diazabicyclooctane derivative
active diazabicyclooctane
Prior art date
Application number
HK15110896.7A
Other languages
English (en)
Chinese (zh)
Inventor
阿部隆夫
奧江雅之
坂卷儀晃
Original Assignee
Meiji Seika Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Meiji Seika Pharma Co Ltd filed Critical Meiji Seika Pharma Co Ltd
Publication of HK1210153A1 publication Critical patent/HK1210153A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • A61K31/431Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems containing further heterocyclic rings, e.g. ticarcillin, azlocillin, oxacillin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
HK15110896.7A 2010-12-22 2015-11-04 Compound for preparing an intermediate compound of optically-active diazabicyclooctane derivative HK1210153A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2010073093 2010-12-22

Publications (1)

Publication Number Publication Date
HK1210153A1 true HK1210153A1 (en) 2016-04-15

Family

ID=46313528

Family Applications (1)

Application Number Title Priority Date Filing Date
HK15110896.7A HK1210153A1 (en) 2010-12-22 2015-11-04 Compound for preparing an intermediate compound of optically-active diazabicyclooctane derivative

Country Status (18)

Country Link
EP (1) EP2657234B1 (xx)
JP (3) JP5903386B2 (xx)
KR (1) KR101836554B1 (xx)
CN (2) CN104892490B (xx)
AR (1) AR116907A2 (xx)
AU (2) AU2011346224B2 (xx)
CA (1) CA2822758C (xx)
DK (1) DK2657234T3 (xx)
ES (1) ES2622004T3 (xx)
HK (1) HK1210153A1 (xx)
HU (1) HUE032491T2 (xx)
IL (5) IL227087A0 (xx)
PL (1) PL2657234T3 (xx)
RU (1) RU2591701C2 (xx)
SG (2) SG191320A1 (xx)
SI (1) SI2657234T1 (xx)
TW (1) TWI599355B (xx)
WO (1) WO2012086241A1 (xx)

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CN106565712A (zh) * 2016-09-30 2017-04-19 天津津泰生物医药技术有限公司 一种阿维巴坦钠中间体的制备方法
CN106699756B (zh) * 2016-12-30 2019-10-29 淄博鑫泉医药技术服务有限公司 β内酰胺酶抑制剂阿维巴坦的合成方法
CN106866668B (zh) * 2017-01-23 2019-01-11 齐鲁天和惠世制药有限公司 一锅法制备阿维巴坦钠的方法
CN106831772B (zh) * 2017-03-04 2019-12-17 丽珠医药集团股份有限公司 一种阿维巴坦中间体的合成方法
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CN109400521B (zh) * 2017-08-18 2020-05-08 新发药业有限公司 一种改进的5r-苄氧氨基哌啶-2s-甲酸酯、其草酸盐的制备方法
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CN109678856B (zh) * 2017-10-18 2020-09-25 新发药业有限公司 一种阿维巴坦中间体的制备方法
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Also Published As

Publication number Publication date
AU2011346224B2 (en) 2017-04-06
RU2591701C2 (ru) 2016-07-20
IL248246A0 (en) 2016-11-30
IL238032A (en) 2017-05-29
AR116907A2 (es) 2021-06-23
SG191320A1 (en) 2013-07-31
DK2657234T3 (da) 2017-02-20
TW201225958A (en) 2012-07-01
SI2657234T1 (sl) 2017-06-30
PL2657234T3 (pl) 2017-06-30
JP6364431B2 (ja) 2018-07-25
AU2017203187B2 (en) 2018-07-26
KR101836554B1 (ko) 2018-04-19
CA2822758A1 (en) 2012-06-28
HUE032491T2 (en) 2017-09-28
KR20140040688A (ko) 2014-04-03
JP2016117742A (ja) 2016-06-30
IL244239A0 (en) 2016-04-21
EP2657234B1 (en) 2017-01-11
CN103328476B (zh) 2016-12-28
WO2012086241A1 (ja) 2012-06-28
IL243939A0 (en) 2016-04-21
CN103328476A (zh) 2013-09-25
IL244239B (en) 2019-01-31
TWI599355B (zh) 2017-09-21
CN104892490A (zh) 2015-09-09
JP5903386B2 (ja) 2016-04-13
AU2011346224A1 (en) 2013-07-04
ES2622004T3 (es) 2017-07-05
RU2013133870A (ru) 2015-01-27
IL227087A0 (en) 2016-10-31
CN104892490B (zh) 2017-07-21
EP2657234A1 (en) 2013-10-30
CA2822758C (en) 2018-03-20
SG10201510576WA (en) 2016-01-28
EP2657234A4 (en) 2014-10-08
JP2018009008A (ja) 2018-01-18
JPWO2012086241A1 (ja) 2014-05-22
IL248246B (en) 2021-02-28
AU2017203187A1 (en) 2017-06-01

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