HK1160139A1 - Biocidal boronophthalide compounds 2-[c] - Google Patents

Biocidal boronophthalide compounds 2-[c]

Info

Publication number
HK1160139A1
HK1160139A1 HK12100416.2A HK12100416A HK1160139A1 HK 1160139 A1 HK1160139 A1 HK 1160139A1 HK 12100416 A HK12100416 A HK 12100416A HK 1160139 A1 HK1160139 A1 HK 1160139A1
Authority
HK
Hong Kong
Prior art keywords
boronophthalide
biocidal
compounds
boronophthalide compounds
biocidal boronophthalide
Prior art date
Application number
HK12100416.2A
Other languages
English (en)
Chinese (zh)
Inventor
Stephen Baker
Tsutomu Akama
Carolyn Bellinger-Kawahara
Vincent Hernandez
Hold Karin G
James Leyden
Kirk Maples
Jacob Plattner
Virginia Sanders
Yong-Kang Zhang
Original Assignee
Anacor Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36917059&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1160139(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Anacor Pharmaceuticals Inc filed Critical Anacor Pharmaceuticals Inc
Publication of HK1160139A1 publication Critical patent/HK1160139A1/xx

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    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/05Cyclic compounds having at least one ring containing boron but no carbon in the ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
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    • A61P17/14Drugs for dermatological disorders for baldness or alopecia
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    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
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    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
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    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
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    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • AHUMAN NECESSITIES
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    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/04Amoebicides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/08Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis for Pneumocystis carinii
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/027Organoboranes and organoborohydrides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Biotechnology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Ophthalmology & Optometry (AREA)
  • AIDS & HIV (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HK12100416.2A 2005-02-16 2008-03-11 Biocidal boronophthalide compounds 2-[c] HK1160139A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US65406005P 2005-02-16 2005-02-16

Publications (1)

Publication Number Publication Date
HK1160139A1 true HK1160139A1 (en) 2012-08-10

Family

ID=36917059

Family Applications (3)

Application Number Title Priority Date Filing Date
HK12100416.2A HK1160139A1 (en) 2005-02-16 2008-03-11 Biocidal boronophthalide compounds 2-[c]
HK08102801.7A HK1109735A1 (en) 2005-02-16 2008-03-11 Halogen-substituted boronophthalides for the treatment of infections
HK16110032.1A HK1221956A1 (zh) 2005-02-16 2016-08-23 用於治療感染的鹵代類苯酞化硼

Family Applications After (2)

Application Number Title Priority Date Filing Date
HK08102801.7A HK1109735A1 (en) 2005-02-16 2008-03-11 Halogen-substituted boronophthalides for the treatment of infections
HK16110032.1A HK1221956A1 (zh) 2005-02-16 2016-08-23 用於治療感染的鹵代類苯酞化硼

Country Status (26)

Country Link
US (11) US7582621B2 (he)
EP (4) EP1853251B1 (he)
JP (6) JP5038912B2 (he)
KR (4) KR101456815B1 (he)
CN (2) CN101160124A (he)
AU (3) AU2006214247C1 (he)
BR (1) BRPI0608431B8 (he)
CA (1) CA2597982C (he)
CY (3) CY1120695T1 (he)
DK (3) DK2987796T3 (he)
ES (4) ES2872962T3 (he)
FR (1) FR20C1024I2 (he)
HK (3) HK1160139A1 (he)
HU (4) HUE040060T2 (he)
IL (2) IL185080A (he)
LT (1) LTC2343304I2 (he)
LU (1) LUC00157I2 (he)
MX (1) MX369262B (he)
NL (1) NL301049I2 (he)
NZ (3) NZ560448A (he)
PL (4) PL2343304T3 (he)
PT (4) PT3424932T (he)
RU (3) RU2414906C2 (he)
SI (3) SI2343304T1 (he)
WO (1) WO2006089067A2 (he)
ZA (4) ZA200707408B (he)

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RU2016145916A3 (he) 2020-07-21
JP2017105826A (ja) 2017-06-15
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US20210070780A1 (en) 2021-03-11
US8440642B2 (en) 2013-05-14
PL1853251T3 (pl) 2013-09-30
PT2987796T (pt) 2018-10-18
CA2597982A1 (en) 2006-08-24
US20190048026A1 (en) 2019-02-14
JP2010248265A (ja) 2010-11-04
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ES2872962T3 (es) 2021-11-03
BRPI0608431B8 (pt) 2021-05-25
CY1120695T1 (el) 2019-12-11
KR20100105869A (ko) 2010-09-30
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SI3424932T1 (sl) 2021-08-31
ZA201506944B (en) 2018-08-29
DK3424932T3 (da) 2021-05-25
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US20130244980A1 (en) 2013-09-19
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PL2343304T3 (pl) 2015-09-30
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BRPI0608431B1 (pt) 2020-09-15
BRPI0608431A2 (pt) 2009-12-29
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FR20C1024I1 (he) 2020-07-31
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US20160108063A1 (en) 2016-04-21
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FR20C1024I2 (fr) 2021-07-09
PL2987796T3 (pl) 2018-12-31
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SI2987796T1 (sl) 2018-11-30
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EP3424932A1 (en) 2019-01-09
IL185080A (he) 2012-07-31
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NZ560448A (en) 2009-08-28
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ES2686981T3 (es) 2018-10-23
IL207156A (he) 2014-04-30

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