HK1125287A1 - Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels - Google Patents

Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels

Info

Publication number
HK1125287A1
HK1125287A1 HK09102821.2A HK09102821A HK1125287A1 HK 1125287 A1 HK1125287 A1 HK 1125287A1 HK 09102821 A HK09102821 A HK 09102821A HK 1125287 A1 HK1125287 A1 HK 1125287A1
Authority
HK
Hong Kong
Prior art keywords
lowering
benzo
fused heterocycle
blood glucose
glucose levels
Prior art date
Application number
HK09102821.2A
Other languages
English (en)
Inventor
Virginia L Smith-Swintosky
Allen B Reitz
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HK1125287A1 publication Critical patent/HK1125287A1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
HK09102821.2A 2005-12-19 2009-03-24 Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels HK1125287A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US75167705P 2005-12-19 2005-12-19
US11/611,961 US8497298B2 (en) 2005-12-19 2006-12-18 Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
PCT/US2006/048477 WO2007092086A2 (en) 2005-12-19 2006-12-19 Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels

Publications (1)

Publication Number Publication Date
HK1125287A1 true HK1125287A1 (en) 2009-08-07

Family

ID=38225368

Family Applications (1)

Application Number Title Priority Date Filing Date
HK09102821.2A HK1125287A1 (en) 2005-12-19 2009-03-24 Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels

Country Status (25)

Country Link
US (1) US8497298B2 (xx)
EP (1) EP1973541B1 (xx)
JP (1) JP5190374B2 (xx)
KR (1) KR101363332B1 (xx)
CN (1) CN101365441B (xx)
AT (1) ATE486595T1 (xx)
AU (1) AU2006337617B8 (xx)
BR (1) BRPI0620011A2 (xx)
CA (1) CA2634419C (xx)
CR (1) CR10169A (xx)
CY (1) CY1111161T1 (xx)
DE (1) DE602006018066D1 (xx)
DK (1) DK1973541T3 (xx)
EA (2) EA016892B1 (xx)
HK (1) HK1125287A1 (xx)
HR (1) HRP20110008T1 (xx)
IL (1) IL192101A (xx)
MY (1) MY148866A (xx)
NO (1) NO20083003L (xx)
NZ (1) NZ569043A (xx)
PL (1) PL1973541T3 (xx)
PT (1) PT1973541E (xx)
RS (1) RS51521B (xx)
SI (1) SI1973541T1 (xx)
WO (1) WO2007092086A2 (xx)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
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MY147767A (en) 2004-06-16 2013-01-31 Janssen Pharmaceutica Nv Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders
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US8937096B2 (en) 2005-12-19 2015-01-20 Janssen Pharmaceutica Nv Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder
US8691867B2 (en) 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
US8497298B2 (en) 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
US20070155827A1 (en) * 2005-12-19 2007-07-05 Smith-Swintosky Virginia L Use of benzo-fused heterocycle sulfamide derivatives for the treatment of depression
EP2026790A2 (en) 2006-05-19 2009-02-25 Janssen Pharmaceutica, N.V. Co-therapy for the treatment of epilepsy and related disorders
US20090247616A1 (en) * 2008-03-26 2009-10-01 Smith-Swintosky Virginia L Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety
US20090247617A1 (en) * 2008-03-26 2009-10-01 Abdel-Magid Ahmed F Process for the preparation of benzo-fused heteroaryl sulfamates
MX2011000090A (es) * 2008-06-23 2011-03-02 Janssen Pharmaceutica Nv Forma cristalina de (2s)-(-)-n-(6-cloro-2,3-dihidro-benzo[1,4]diox in-2-ilmetil)sulfamida.
US8815939B2 (en) * 2008-07-22 2014-08-26 Janssen Pharmaceutica Nv Substituted sulfamide derivatives
CA2850015A1 (en) 2011-09-29 2013-04-04 Janssen Pharmaceutica Nv Improved process for the preparation of sulfamide derivatives
JP2014528953A (ja) 2011-09-29 2014-10-30 ヤンセン ファーマシューティカ エヌ．ベー． スルファミド誘導体の調製プロセス
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CN105232544A (zh) * 2015-11-11 2016-01-13 朱忠良 一种抗糖尿病的口服药物组合物
CN105232543A (zh) * 2015-11-11 2016-01-13 朱忠良 一种抗糖尿病的口服药物组合物

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EA201000630A1 (ru) 2010-10-29
US8497298B2 (en) 2013-07-30
CA2634419C (en) 2014-10-14
RS51521B (en) 2011-06-30
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CN101365441B (zh) 2011-11-16
ATE486595T1 (de) 2010-11-15
KR20080089408A (ko) 2008-10-06
EA015606B1 (ru) 2011-10-31
MY148866A (en) 2013-06-14
CR10169A (es) 2009-01-14
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EP1973541B1 (en) 2010-11-03
KR101363332B1 (ko) 2014-02-19
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EA016892B1 (ru) 2012-08-30
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US20070155821A1 (en) 2007-07-05
PT1973541E (pt) 2010-12-14
DE602006018066D1 (de) 2010-12-16
CN101365441A (zh) 2009-02-11
EP1973541A2 (en) 2008-10-01
IL192101A (en) 2013-03-24
IL192101A0 (en) 2009-08-03
SI1973541T1 (sl) 2011-02-28
AU2006337617A1 (en) 2007-08-16
EA200870088A1 (ru) 2009-02-27
WO2007092086A2 (en) 2007-08-16
AU2006337617B2 (en) 2013-02-07
CA2634419A1 (en) 2007-08-16
NZ569043A (en) 2011-03-31
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AU2006337617B8 (en) 2013-05-30
CY1111161T1 (el) 2015-06-11

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