HK1076445A1 - Substituted phenylalkanoic acid derivatives and use thereof - Google Patents

Substituted phenylalkanoic acid derivatives and use thereof

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Publication number
HK1076445A1
HK1076445A1 HK05108316.5A HK05108316A HK1076445A1 HK 1076445 A1 HK1076445 A1 HK 1076445A1 HK 05108316 A HK05108316 A HK 05108316A HK 1076445 A1 HK1076445 A1 HK 1076445A1
Authority
HK
Hong Kong
Prior art keywords
group
carbon atoms
alkyl group
acid derivatives
integer
Prior art date
Application number
HK05108316.5A
Other languages
English (en)
Inventor
Motoshi Shoda
Hiroshi Kuriyama
Original Assignee
Asahi Kasei Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asahi Kasei Pharma Corp filed Critical Asahi Kasei Pharma Corp
Publication of HK1076445A1 publication Critical patent/HK1076445A1/xx

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    • C07C59/68—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings the oxygen atom of the ether group being bound to a non-condensed six-membered aromatic ring
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HK05108316.5A 2002-02-21 2005-09-22 Substituted phenylalkanoic acid derivatives and use thereof HK1076445A1 (en)

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PCT/JP2003/001849 WO2003070686A1 (fr) 2002-02-21 2003-02-20 Derive de l'acide phenylalcanoyle substitue et son utilisation

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ATE420847T1 (de) * 2002-02-21 2009-01-15 Asahi Kasei Pharma Corp Substituiertes phenylalkansäurederivat und dessen verwendung
JP4594611B2 (ja) * 2002-11-08 2010-12-08 武田薬品工業株式会社 受容体機能調節剤
EP2385032A1 (de) * 2002-11-08 2011-11-09 Takeda Pharmaceutical Company Limited GPR40 Rezeptorfunktionsregler
JP4697962B2 (ja) * 2003-02-13 2011-06-08 ウェルスタット セラピューティクス コーポレイション 代謝性障害の処置のための化合物
CA2535665A1 (en) * 2003-08-14 2005-02-24 Asahi Kasei Pharma Corporation Substituted arylalkanoic acid derivative and use thereof
CA2547430A1 (en) * 2003-11-26 2005-06-09 Takeda Pharmaceutical Company Limited Receptor function regulating agent
EP1720855A4 (de) * 2004-03-02 2008-12-17 Smithkline Beecham Corp Hemmer der akt aktivität
GB0409921D0 (en) * 2004-05-04 2004-06-09 Novartis Ag Organic compounds
TW200716588A (en) * 2005-06-02 2007-05-01 Kyowa Hakko Kogyo Kk A process for preparing dibenzoxepin derivative
US7405302B2 (en) * 2005-10-11 2008-07-29 Amira Pharmaceuticals, Inc. 5-lipoxygenase-activating protein (FLAP) inhibitors
KR20120084790A (ko) * 2006-07-20 2012-07-30 아사히 가세이 파마 가부시키가이샤 치환 페닐알칸산의 신규 결정 및 제조 방법
CL2008000973A1 (es) * 2007-04-05 2009-01-02 Astrazeneca Ab Compuestos derivados de 1-oxo-isoquinolina; procedimiento de preparación; composición farmacéutica; y su uso en el tratamiento de enfermedades pulmonares obstructvas crónicas (epoc) y asma.
EP2154131A4 (de) * 2007-04-26 2011-09-21 Pharmafrontier Co Ltd Inhibitor des g-protein-gekoppelten rezeptors und pharmazeutisches produkt
TW200911798A (en) * 2007-08-02 2009-03-16 Amgen Inc PI3 kinase modulators and methods of use
JP5301468B2 (ja) * 2008-01-18 2013-09-25 旭化成ファーマ株式会社 安定な医薬組成物
CA2722102C (en) * 2008-04-28 2013-06-11 Asahi Kasei Pharma Corporation Phenylpropionic acid derivative and use thereof
DK2292592T3 (da) 2008-06-05 2012-10-08 Asahi Kasei Pharma Corp Sulfonamidforbindelse og anvendelse deraf
CN102391264A (zh) * 2011-09-21 2012-03-28 河北九派制药有限公司 6-溴咪唑并[1,2-a]吡啶的制备方法
JP5802518B2 (ja) 2011-10-31 2015-10-28 公益財団法人微生物化学研究会 新規化合物、その製造方法、及びその用途
US8889730B2 (en) 2012-04-10 2014-11-18 Pfizer Inc. Indole and indazole compounds that activate AMPK
CA2905242C (en) 2013-03-15 2016-11-29 Pfizer Inc. Indole compounds that activate ampk
CN105315167A (zh) * 2014-08-01 2016-02-10 华东师范大学 一种2,2,3-三芳基-3-芳基氨基丙酸甲酯衍生物及其合成方法和应用
CA3121986C (en) * 2014-12-24 2024-04-09 Lg Chem, Ltd. Biaryl derivative as gpr120 agonist
JP6635999B2 (ja) * 2017-10-13 2020-01-29 株式会社ダイセル カリウム塩の製造方法、及びカリウム塩
CN110092774B (zh) * 2018-01-29 2022-04-08 中国科学院上海药物研究所 芳香丙酸类衍生物、及其制备方法和用途
CN117120090A (zh) * 2021-02-12 2023-11-24 林伯士萨顿公司 Hpk1拮抗剂和其用途
CN117295737A (zh) 2021-03-05 2023-12-26 林伯士萨顿公司 Hpk1拮抗剂和其用途

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ATE420847T1 (de) * 2002-02-21 2009-01-15 Asahi Kasei Pharma Corp Substituiertes phenylalkansäurederivat und dessen verwendung

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DK1477472T3 (da) 2009-04-06
JPWO2003070686A1 (ja) 2005-06-09
CN1653032A (zh) 2005-08-10
CA2477208A1 (en) 2003-08-28
EP1477472A1 (de) 2004-11-17
PT1477472E (pt) 2009-03-17
WO2003070686A1 (fr) 2003-08-28
DE60325830D1 (de) 2009-03-05
AU2003211384B2 (en) 2008-12-11
KR20040094712A (ko) 2004-11-10
EP1477472B1 (de) 2009-01-14
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CA2477208C (en) 2010-11-30
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MXPA04008176A (es) 2004-11-26
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AU2003211384A1 (en) 2003-09-09
JP5048017B2 (ja) 2012-10-17

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