GB1598294A - Process for the preparation of kanamycin derivatives - Google Patents

Process for the preparation of kanamycin derivatives Download PDF

Info

Publication number
GB1598294A
GB1598294A GB16571/78A GB1657178A GB1598294A GB 1598294 A GB1598294 A GB 1598294A GB 16571/78 A GB16571/78 A GB 16571/78A GB 1657178 A GB1657178 A GB 1657178A GB 1598294 A GB1598294 A GB 1598294A
Authority
GB
United Kingdom
Prior art keywords
kanamycin
acid
amino
polysilylated
silyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB16571/78A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Co
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of GB1598294A publication Critical patent/GB1598294A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
GB16571/78A 1977-04-28 1978-04-26 Process for the preparation of kanamycin derivatives Expired GB1598294A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79180677A 1977-04-28 1977-04-28
US88858578A 1978-03-20 1978-03-20

Publications (1)

Publication Number Publication Date
GB1598294A true GB1598294A (en) 1981-09-16

Family

ID=27121201

Family Applications (1)

Application Number Title Priority Date Filing Date
GB16571/78A Expired GB1598294A (en) 1977-04-28 1978-04-26 Process for the preparation of kanamycin derivatives

Country Status (27)

Country Link
JP (1) JPS53149951A (fi)
AR (1) AR218910A1 (fi)
AT (1) AT357675B (fi)
CA (2) CA1100953A (fi)
CH (1) CH639104A5 (fi)
CS (1) CS207607B2 (fi)
CY (1) CY1241A (fi)
DE (2) DE2818822A1 (fi)
DK (2) DK165450C (fi)
EG (1) EG13710A (fi)
ES (1) ES469303A1 (fi)
FI (1) FI781288A (fi)
FR (2) FR2388827A1 (fi)
GB (1) GB1598294A (fi)
HK (1) HK51484A (fi)
IE (2) IE47271B1 (fi)
IT (2) IT1105500B (fi)
KE (1) KE3398A (fi)
LU (1) LU79541A1 (fi)
MY (1) MY8500528A (fi)
NL (1) NL178790C (fi)
NO (2) NO149635C (fi)
PL (1) PL117307B1 (fi)
PT (1) PT67959B (fi)
SE (2) SE447259B (fi)
SG (1) SG22884G (fi)
YU (2) YU41590B (fi)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003070693A1 (fr) * 2002-02-19 2003-08-28 Amato Pharmaceutical Products, Ltd. Derive de l'acide lactique
US8383596B2 (en) 2007-11-21 2013-02-26 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8492354B2 (en) 2009-05-15 2013-07-23 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8524675B2 (en) 2009-05-15 2013-09-03 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8524689B2 (en) 2009-05-15 2013-09-03 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8653042B2 (en) 2009-05-15 2014-02-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8658606B2 (en) 2009-05-15 2014-02-25 Achaogen, Inc. Antibacterial aminoglycoside analogs

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55306A (en) * 1978-04-28 1980-01-05 Bristol Myers Co Manufacture of 11nn*omegaaaminooalphaahydroxy alkanoyl**aminoglycoside antibiotic

Cited By (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003070693A1 (fr) * 2002-02-19 2003-08-28 Amato Pharmaceutical Products, Ltd. Derive de l'acide lactique
US8383596B2 (en) 2007-11-21 2013-02-26 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8822424B2 (en) 2007-11-21 2014-09-02 Achaogen, Inc. Antibacterial aminoglycoside analogs
US9266919B2 (en) 2007-11-21 2016-02-23 Achaogen, Inc. Antibacterial aminoglycoside analogs
US9688711B2 (en) 2007-11-21 2017-06-27 Achaogen, Inc. Antibacterial aminoglycoside analogs
US11117915B2 (en) 2007-11-21 2021-09-14 Cipla USA, Inc. Antibacterial aminoglycoside analogs
US8492354B2 (en) 2009-05-15 2013-07-23 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8524675B2 (en) 2009-05-15 2013-09-03 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8524689B2 (en) 2009-05-15 2013-09-03 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8653042B2 (en) 2009-05-15 2014-02-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
US8658606B2 (en) 2009-05-15 2014-02-25 Achaogen, Inc. Antibacterial aminoglycoside analogs
USRE47741E1 (en) 2009-05-15 2019-11-26 Achaogen, Inc. Antibacterial aminoglycoside analogs

Also Published As

Publication number Publication date
FI781288A (fi) 1978-10-29
DK183078A (da) 1978-10-29
FR2388827A1 (fr) 1978-11-24
YU41590B (en) 1987-12-31
IT1105500B (it) 1985-11-04
PL206457A1 (fi) 1980-03-24
FR2388827B1 (fi) 1982-07-09
IE46945B1 (en) 1983-11-16
NO149635B (no) 1984-02-13
FR2388826A1 (fr) 1978-11-24
YU102578A (en) 1983-01-21
CA1105454A (en) 1981-07-21
NO149635C (no) 1984-05-23
DK165450B (da) 1992-11-30
IT1156718B (it) 1987-02-04
IE780841L (en) 1978-10-28
YU102478A (en) 1982-10-31
CH639104A5 (en) 1983-10-31
DE2818992A1 (de) 1978-11-23
JPS53149951A (en) 1978-12-27
FR2388826B1 (fi) 1982-12-10
LU79541A1 (fr) 1978-11-28
JPS5721277B2 (fi) 1982-05-06
DE2818822A1 (de) 1978-11-09
AR218910A1 (es) 1980-07-15
HK51484A (en) 1984-06-22
CA1100953A (en) 1981-05-12
NL178790C (nl) 1986-05-16
NO154697B (no) 1986-08-25
EG13710A (en) 1982-09-30
NL178790B (nl) 1985-12-16
CS207607B2 (en) 1981-08-31
NO781437L (no) 1978-10-31
PT67959B (en) 1980-03-05
ATA312778A (de) 1979-12-15
PT67959A (en) 1978-05-01
NL7804503A (nl) 1978-10-31
SE447259B (sv) 1986-11-03
ES469303A1 (es) 1979-09-16
PL117307B1 (en) 1981-07-31
DK172543B1 (da) 1998-12-07
IT7849136A0 (it) 1978-04-28
CY1241A (en) 1984-06-29
NO831197L (no) 1978-10-31
IE47271B1 (en) 1984-02-08
IE780842L (en) 1978-10-28
DK165450C (da) 1993-04-13
IT7849137A0 (it) 1978-04-28
DE2818992C2 (fi) 1988-03-17
DK182978A (da) 1978-10-29
MY8500528A (en) 1985-12-31
SE8305538L (sv) 1983-10-07
DE2818822C2 (fi) 1989-01-26
SE8305538D0 (sv) 1983-10-07
NO154697C (no) 1986-12-03
SE7804973L (sv) 1978-10-29
SE461148B (sv) 1990-01-15
KE3398A (en) 1984-06-08
AT357675B (de) 1980-07-25
SG22884G (en) 1985-01-04

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Legal Events

Date Code Title Description
PS Patent sealed [section 19, patents act 1949]
PE20 Patent expired after termination of 20 years

Effective date: 19980425