GB1598294A - Process for the preparation of kanamycin derivatives - Google Patents
Process for the preparation of kanamycin derivatives Download PDFInfo
- Publication number
- GB1598294A GB1598294A GB16571/78A GB1657178A GB1598294A GB 1598294 A GB1598294 A GB 1598294A GB 16571/78 A GB16571/78 A GB 16571/78A GB 1657178 A GB1657178 A GB 1657178A GB 1598294 A GB1598294 A GB 1598294A
- Authority
- GB
- United Kingdom
- Prior art keywords
- kanamycin
- acid
- amino
- polysilylated
- silyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Saccharide Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US79180677A | 1977-04-28 | 1977-04-28 | |
| US88858578A | 1978-03-20 | 1978-03-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1598294A true GB1598294A (en) | 1981-09-16 |
Family
ID=27121201
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB16571/78A Expired GB1598294A (en) | 1977-04-28 | 1978-04-26 | Process for the preparation of kanamycin derivatives |
Country Status (27)
| Country | Link |
|---|---|
| JP (1) | JPS53149951A (da) |
| AR (1) | AR218910A1 (da) |
| AT (1) | AT357675B (da) |
| CA (2) | CA1100953A (da) |
| CH (1) | CH639104A5 (da) |
| CS (1) | CS207607B2 (da) |
| CY (1) | CY1241A (da) |
| DE (2) | DE2818992A1 (da) |
| DK (2) | DK172543B1 (da) |
| EG (1) | EG13710A (da) |
| ES (1) | ES469303A1 (da) |
| FI (1) | FI781288A (da) |
| FR (2) | FR2388826A1 (da) |
| GB (1) | GB1598294A (da) |
| HK (1) | HK51484A (da) |
| IE (2) | IE46945B1 (da) |
| IT (2) | IT1156718B (da) |
| KE (1) | KE3398A (da) |
| LU (1) | LU79541A1 (da) |
| MY (1) | MY8500528A (da) |
| NL (1) | NL178790C (da) |
| NO (2) | NO149635C (da) |
| PL (1) | PL117307B1 (da) |
| PT (1) | PT67959B (da) |
| SE (2) | SE447259B (da) |
| SG (1) | SG22884G (da) |
| YU (2) | YU102578A (da) |
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003070693A1 (fr) * | 2002-02-19 | 2003-08-28 | Amato Pharmaceutical Products, Ltd. | Derive de l'acide lactique |
| US8383596B2 (en) | 2007-11-21 | 2013-02-26 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8492354B2 (en) | 2009-05-15 | 2013-07-23 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8524675B2 (en) | 2009-05-15 | 2013-09-03 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8524689B2 (en) | 2009-05-15 | 2013-09-03 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8653042B2 (en) | 2009-05-15 | 2014-02-18 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8658606B2 (en) | 2009-05-15 | 2014-02-25 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS55306A (en) * | 1978-04-28 | 1980-01-05 | Bristol Myers Co | Manufacture of 11nn*omegaaaminooalphaahydroxy alkanoyl**aminoglycoside antibiotic |
-
1978
- 1978-04-21 AR AR271852A patent/AR218910A1/es active
- 1978-04-25 CA CA301,962A patent/CA1100953A/en not_active Expired
- 1978-04-25 FI FI781288A patent/FI781288A/fi not_active Application Discontinuation
- 1978-04-25 NO NO781437A patent/NO149635C/no unknown
- 1978-04-25 CA CA301,968A patent/CA1105454A/en not_active Expired
- 1978-04-26 CY CY1241A patent/CY1241A/xx unknown
- 1978-04-26 DK DK197801830A patent/DK172543B1/da not_active IP Right Cessation
- 1978-04-26 NL NLAANVRAGE7804503,A patent/NL178790C/xx not_active IP Right Cessation
- 1978-04-26 GB GB16571/78A patent/GB1598294A/en not_active Expired
- 1978-04-26 DK DK182978A patent/DK165450C/da not_active IP Right Cessation
- 1978-04-27 FR FR7812589A patent/FR2388826A1/fr active Granted
- 1978-04-27 YU YU01025/78A patent/YU102578A/xx unknown
- 1978-04-27 YU YU1024/78A patent/YU41590B/xx unknown
- 1978-04-27 FR FR7812591A patent/FR2388827A1/fr active Granted
- 1978-04-27 IE IE841/78A patent/IE46945B1/en not_active IP Right Cessation
- 1978-04-27 IE IE842/78A patent/IE47271B1/en not_active IP Right Cessation
- 1978-04-27 CS CS782729A patent/CS207607B2/cs unknown
- 1978-04-27 PT PT67959A patent/PT67959B/pt unknown
- 1978-04-27 LU LU79541A patent/LU79541A1/xx unknown
- 1978-04-28 IT IT49136/78A patent/IT1156718B/it active
- 1978-04-28 JP JP5016078A patent/JPS53149951A/ja active Granted
- 1978-04-28 DE DE19782818992 patent/DE2818992A1/de active Granted
- 1978-04-28 PL PL1978206457A patent/PL117307B1/pl unknown
- 1978-04-28 DE DE19782818822 patent/DE2818822A1/de active Granted
- 1978-04-28 CH CH470278A patent/CH639104A5/de not_active IP Right Cessation
- 1978-04-28 IT IT49137/78A patent/IT1105500B/it active
- 1978-04-28 ES ES469303A patent/ES469303A1/es not_active Expired
- 1978-04-28 AT AT312778A patent/AT357675B/de not_active IP Right Cessation
- 1978-04-28 SE SE7804973A patent/SE447259B/sv not_active IP Right Cessation
- 1978-04-29 EG EG283/78A patent/EG13710A/xx active
-
1983
- 1983-04-05 NO NO83831197A patent/NO154697C/no unknown
- 1983-10-07 SE SE8305538A patent/SE461148B/sv not_active IP Right Cessation
-
1984
- 1984-03-12 SG SG228/84A patent/SG22884G/en unknown
- 1984-04-12 KE KE3398A patent/KE3398A/xx unknown
- 1984-06-22 HK HK514/84A patent/HK51484A/xx not_active IP Right Cessation
-
1985
- 1985-12-30 MY MY528/85A patent/MY8500528A/xx unknown
Cited By (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003070693A1 (fr) * | 2002-02-19 | 2003-08-28 | Amato Pharmaceutical Products, Ltd. | Derive de l'acide lactique |
| US8383596B2 (en) | 2007-11-21 | 2013-02-26 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8822424B2 (en) | 2007-11-21 | 2014-09-02 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US9266919B2 (en) | 2007-11-21 | 2016-02-23 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US9688711B2 (en) | 2007-11-21 | 2017-06-27 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US11117915B2 (en) | 2007-11-21 | 2021-09-14 | Cipla USA, Inc. | Antibacterial aminoglycoside analogs |
| US8492354B2 (en) | 2009-05-15 | 2013-07-23 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8524675B2 (en) | 2009-05-15 | 2013-09-03 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8524689B2 (en) | 2009-05-15 | 2013-09-03 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8653042B2 (en) | 2009-05-15 | 2014-02-18 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| US8658606B2 (en) | 2009-05-15 | 2014-02-25 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
| USRE47741E1 (en) | 2009-05-15 | 2019-11-26 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PE20 | Patent expired after termination of 20 years |
Effective date: 19980425 |