FR2833596B1 - Procede de preparation de derives d'echinocandine - Google Patents

Procede de preparation de derives d'echinocandine

Info

Publication number
FR2833596B1
FR2833596B1 FR0116230A FR0116230A FR2833596B1 FR 2833596 B1 FR2833596 B1 FR 2833596B1 FR 0116230 A FR0116230 A FR 0116230A FR 0116230 A FR0116230 A FR 0116230A FR 2833596 B1 FR2833596 B1 FR 2833596B1
Authority
FR
France
Prior art keywords
preparation
echinocandin derivatives
echinocandin
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0116230A
Other languages
English (en)
French (fr)
Other versions
FR2833596A1 (fr
Inventor
Philippe Boffelli
Agnes Brouillard
Colette Colladant
Serge Droux
Michel Elter
Didier Ferroud
Guy Lemaitre
Joseph Paladino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Aventis Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR0116230A priority Critical patent/FR2833596B1/fr
Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA
Priority to CN02824928A priority patent/CN100584859C/zh
Priority to AT02805374T priority patent/ATE441662T1/de
Priority to NZ533864A priority patent/NZ533864A/xx
Priority to EA200400806A priority patent/EA007964B1/ru
Priority to AU2002364991A priority patent/AU2002364991B9/en
Priority to EP02805374A priority patent/EP1456229B1/fr
Priority to JP2003554717A priority patent/JP4510461B2/ja
Priority to PT02805374T priority patent/PT1456229E/pt
Priority to SI200230861T priority patent/SI1456229T1/sl
Priority to DE60233589T priority patent/DE60233589D1/de
Priority to PL02371763A priority patent/PL371763A1/xx
Priority to CA002469918A priority patent/CA2469918A1/fr
Priority to DK02805374T priority patent/DK1456229T3/da
Priority to BR0214937-0A priority patent/BR0214937A/pt
Priority to CNB2005101156130A priority patent/CN1326872C/zh
Priority to HU0402602A priority patent/HUP0402602A3/hu
Priority to ES02805374T priority patent/ES2333784T3/es
Priority to PCT/FR2002/004308 priority patent/WO2003054001A2/fr
Priority to KR10-2004-7009121A priority patent/KR20040066167A/ko
Priority to US11/591,898 priority patent/US20070105760A1/en
Priority to MXPA04005484A priority patent/MXPA04005484A/es
Priority to HK05104783.8A priority patent/HK1071900B/xx
Priority to TW091136168A priority patent/TWI322820B/zh
Priority to ARP020104846A priority patent/AR037827A1/es
Priority to IL16238502A priority patent/IL162385A0/xx
Publication of FR2833596A1 publication Critical patent/FR2833596A1/fr
Priority to ZA200404631A priority patent/ZA200404631B/en
Priority to CO04055277A priority patent/CO5590934A2/es
Priority to US10/867,070 priority patent/US7148322B2/en
Priority to NO20042640A priority patent/NO20042640L/no
Application granted granted Critical
Publication of FR2833596B1 publication Critical patent/FR2833596B1/fr
Priority to HK06107828.7A priority patent/HK1087720B/xx
Priority to CY20091101267T priority patent/CY1110694T1/el
Priority to US12/830,941 priority patent/US20100273977A1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
FR0116230A 2001-12-14 2001-12-14 Procede de preparation de derives d'echinocandine Expired - Fee Related FR2833596B1 (fr)

Priority Applications (33)

Application Number Priority Date Filing Date Title
FR0116230A FR2833596B1 (fr) 2001-12-14 2001-12-14 Procede de preparation de derives d'echinocandine
KR10-2004-7009121A KR20040066167A (ko) 2001-12-14 2002-12-12 에키노칸딘 유도체의 제조방법
NZ533864A NZ533864A (en) 2001-12-14 2002-12-12 Method for preparing echinocandin derivatives and their compositions
EA200400806A EA007964B1 (ru) 2001-12-14 2002-12-12 Способ получения эхинокандиновых соединений
AU2002364991A AU2002364991B9 (en) 2001-12-14 2002-12-12 Method for preparing echinocandin derivatives and their compositions
MXPA04005484A MXPA04005484A (es) 2001-12-14 2002-12-12 Procedimiento de preparacion de derivados de equinocandina.
JP2003554717A JP4510461B2 (ja) 2001-12-14 2002-12-12 エキノカンジン誘導体の製造方法
PT02805374T PT1456229E (pt) 2001-12-14 2002-12-12 Processo de preparação de derivados de equinocandina
SI200230861T SI1456229T1 (sl) 2001-12-14 2002-12-12 Postopek za pripravo ehinokandinskih derivatov
DE60233589T DE60233589D1 (de) 2001-12-14 2002-12-12 Verfahren zur herstellung von echinocandinderivaten
PL02371763A PL371763A1 (en) 2001-12-14 2002-12-12 Method for preparing echinocandin derivatives
CA002469918A CA2469918A1 (fr) 2001-12-14 2002-12-12 Procede de preparation de derives d'echinocandines et leurs compositions
DK02805374T DK1456229T3 (da) 2001-12-14 2002-12-12 Fremgangsmåe til fremstilling af echinocandin-derivater
BR0214937-0A BR0214937A (pt) 2001-12-14 2002-12-12 Processo de preparação de derivados de equinocandina
CNB2005101156130A CN1326872C (zh) 2001-12-14 2002-12-12 制备棘白菌素衍生物的方法
HU0402602A HUP0402602A3 (en) 2001-12-14 2002-12-12 Method for preparing echinocandin derivatives, their use, pharmaceutical compositions comprising thereof and their intermediates
CN02824928A CN100584859C (zh) 2001-12-14 2002-12-12 制备棘白菌素衍生物的方法
PCT/FR2002/004308 WO2003054001A2 (fr) 2001-12-14 2002-12-12 Procede de preparation de derives d'echinocandines et leurs compositions
US11/591,898 US20070105760A1 (en) 2001-12-14 2002-12-12 Process for the preparation of echinocandin derivatives
AT02805374T ATE441662T1 (de) 2001-12-14 2002-12-12 Verfahren zur herstellung von echinocandinderivaten
EP02805374A EP1456229B1 (fr) 2001-12-14 2002-12-12 Procede de preparation de derives d echinocandine
HK05104783.8A HK1071900B (en) 2001-12-14 2002-12-12 Method for preparing echinocandin derivatives
ES02805374T ES2333784T3 (es) 2001-12-14 2002-12-12 Procedimiento para la preparacion de derivados de equinocandina.
TW091136168A TWI322820B (en) 2001-12-14 2002-12-13 Process for the preparation of echinocandin derivatives
ARP020104846A AR037827A1 (es) 2001-12-14 2002-12-13 Procedimiento de preparacion de derivados de equinocandina
IL16238502A IL162385A0 (en) 2001-12-14 2002-12-24 Process for the preparation of echinocandin derivatives
ZA200404631A ZA200404631B (en) 2001-12-14 2004-06-10 Process for the preparation of echinocandin derivatives.
CO04055277A CO5590934A2 (es) 2001-12-14 2004-06-11 Procedimiento de preparacion de derivados de equinocandina
US10/867,070 US7148322B2 (en) 2001-12-14 2004-06-14 Process for the preparation of echinocandin derivatives
NO20042640A NO20042640L (no) 2001-12-14 2004-06-23 Fremgangsmate for fremstilling av ekinocandinderivater
HK06107828.7A HK1087720B (en) 2001-12-14 2006-07-13 Method for preparing echinocandin derivatives
CY20091101267T CY1110694T1 (el) 2001-12-14 2009-12-01 Μεθοδος παρασκευης παραγωγων της εχινοκανδινης
US12/830,941 US20100273977A1 (en) 2001-12-14 2010-07-06 Process for the preparation of echinocandin derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0116230A FR2833596B1 (fr) 2001-12-14 2001-12-14 Procede de preparation de derives d'echinocandine

Publications (2)

Publication Number Publication Date
FR2833596A1 FR2833596A1 (fr) 2003-06-20
FR2833596B1 true FR2833596B1 (fr) 2005-02-18

Family

ID=8870520

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0116230A Expired - Fee Related FR2833596B1 (fr) 2001-12-14 2001-12-14 Procede de preparation de derives d'echinocandine

Country Status (28)

Country Link
US (3) US20070105760A1 (enExample)
EP (1) EP1456229B1 (enExample)
JP (1) JP4510461B2 (enExample)
KR (1) KR20040066167A (enExample)
CN (2) CN100584859C (enExample)
AR (1) AR037827A1 (enExample)
AT (1) ATE441662T1 (enExample)
AU (1) AU2002364991B9 (enExample)
BR (1) BR0214937A (enExample)
CA (1) CA2469918A1 (enExample)
CO (1) CO5590934A2 (enExample)
CY (1) CY1110694T1 (enExample)
DE (1) DE60233589D1 (enExample)
DK (1) DK1456229T3 (enExample)
EA (1) EA007964B1 (enExample)
ES (1) ES2333784T3 (enExample)
FR (1) FR2833596B1 (enExample)
HU (1) HUP0402602A3 (enExample)
IL (1) IL162385A0 (enExample)
MX (1) MXPA04005484A (enExample)
NO (1) NO20042640L (enExample)
NZ (1) NZ533864A (enExample)
PL (1) PL371763A1 (enExample)
PT (1) PT1456229E (enExample)
SI (1) SI1456229T1 (enExample)
TW (1) TWI322820B (enExample)
WO (1) WO2003054001A2 (enExample)
ZA (1) ZA200404631B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2833596B1 (fr) * 2001-12-14 2005-02-18 Aventis Pharma Sa Procede de preparation de derives d'echinocandine
TW200826957A (en) * 2006-10-16 2008-07-01 Teva Gyogyszergyar Zartkoruen Mukodo Reszvenytarsasag Purification processes for echinocandin-type compounds
FR2921060B1 (fr) * 2007-09-14 2012-06-15 Novexel Nouveau procede de preparation d'une piperidine disubsituee et nouveaux intermediaires
FR2936798B1 (fr) * 2008-10-03 2012-09-28 Novexel Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens.
FR2936951B1 (fr) * 2008-10-10 2010-12-03 Novexel Nouvelles combinaisons de composes heterocycliques azotes antibacteriens avec d'autres composes antibacteriens et leur utilisation comme medicaments
FR2937034B1 (fr) * 2008-10-10 2012-11-23 Novexel Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens
CN101928670B (zh) 2009-09-24 2012-02-22 上海天伟生物制药有限公司 一种抗生素的高产菌株及其制备方法和用途
CN102627689B (zh) * 2012-03-30 2014-08-06 上海天伟生物制药有限公司 一种环肽类化合物的水合物及其制备方法和用途
CN102627688B (zh) * 2012-03-30 2014-12-31 上海天伟生物制药有限公司 一种高纯度环肽化合物及其制备方法和用途
CN102659930B (zh) * 2012-03-30 2014-04-23 上海天伟生物制药有限公司 一种高纯度环肽类物质的晶体及其制备方法和用途
WO2016056022A2 (en) * 2014-10-07 2016-04-14 Alaparthi Lakshmi Prasad Intermediates and processes to prepare anidulafungin
CN112646854B (zh) * 2020-12-11 2022-10-11 浙江工业大学 一种棘白菌素b合成培养基及应用
CN115785226A (zh) * 2021-09-09 2023-03-14 上海天伟生物制药有限公司 一种棘白菌素药物杂质及其制备、纯化方法和应用

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4293484A (en) * 1979-12-13 1981-10-06 Eli Lilly And Company Derivatives of A-30912H nucleus
US5207710A (en) * 1988-09-29 1993-05-04 Collagen Corporation Method for improving implant fixation
US5696270A (en) * 1989-05-23 1997-12-09 Abbott Laboratories Intermediate for making retroviral protease inhibiting compounds
US5386009A (en) * 1990-03-19 1995-01-31 Merck & Co. Inc. Lipopeptide derivatives
CZ288974B6 (cs) * 1992-03-19 2001-10-17 Eli Lilly And Company Acylový derivát echinocandinu, způsob jeho přípravy, farmaceutický prostředek s jeho obsahem a jeho pouľití
SG75092A1 (en) * 1993-08-09 2000-09-19 Biomeasure Inc Therapeutic peptide derivatives
JP3107691B2 (ja) * 1993-12-03 2000-11-13 株式会社東芝 半導体記憶装置及びその製造方法
EP0781141B1 (en) * 1994-09-16 2002-09-04 Merck & Co. Inc. Aza cyclohexapeptide compounds
US5646111A (en) * 1995-04-07 1997-07-08 Eli Lilly And Company Cyclic peptide antifungal Agents
US5652213A (en) * 1995-05-26 1997-07-29 Eli Lilly And Company Cyclic peptide antifungal agents
US5852213A (en) * 1996-07-10 1998-12-22 American Cyanamid Company Mercaptoketones and mercaptoalcohols and a process for their preparation
US6207710B1 (en) * 1996-11-22 2001-03-27 Elan Pharmaceuticals, Inc. Compounds for inhibiting β-amyloid peptide release and/or its synthesis
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
FR2794746B1 (fr) * 1999-06-09 2002-12-06 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
FR2794747B1 (fr) * 1999-06-09 2004-04-16 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
JP2003505468A (ja) * 1999-07-27 2003-02-12 アヴェンティス ファルマ ドイチェラント ゲーエムベーハー 新規なシクロヘキサペプチド化合物、それらの製造方法及びそれらの医薬品としての使用
FR2833596B1 (fr) * 2001-12-14 2005-02-18 Aventis Pharma Sa Procede de preparation de derives d'echinocandine

Also Published As

Publication number Publication date
IL162385A0 (en) 2005-11-20
DE60233589D1 (de) 2009-10-15
EP1456229A2 (fr) 2004-09-15
CO5590934A2 (es) 2005-12-30
HK1087720A1 (en) 2006-10-20
PT1456229E (pt) 2009-12-10
CN100584859C (zh) 2010-01-27
TW200301133A (en) 2003-07-01
NZ533864A (en) 2006-03-31
ZA200404631B (en) 2005-01-10
NO20042640L (no) 2004-06-23
EA200400806A1 (ru) 2004-12-30
EA007964B1 (ru) 2007-02-27
US20100273977A1 (en) 2010-10-28
AR037827A1 (es) 2004-12-09
CA2469918A1 (fr) 2003-07-03
WO2003054001A3 (fr) 2004-01-22
HUP0402602A3 (en) 2012-06-28
TWI322820B (en) 2010-04-01
US20070105760A1 (en) 2007-05-10
AU2002364991B2 (en) 2008-05-15
HK1071900A1 (zh) 2005-08-05
BR0214937A (pt) 2004-12-14
CN1604908A (zh) 2005-04-06
CN1326872C (zh) 2007-07-18
WO2003054001A2 (fr) 2003-07-03
EP1456229B1 (fr) 2009-09-02
CY1110694T1 (el) 2015-06-10
JP4510461B2 (ja) 2010-07-21
US20050032679A1 (en) 2005-02-10
US7148322B2 (en) 2006-12-12
AU2002364991A1 (en) 2003-07-09
AU2002364991B9 (en) 2008-10-09
SI1456229T1 (sl) 2010-02-26
CN1781938A (zh) 2006-06-07
HUP0402602A2 (hu) 2005-04-28
PL371763A1 (en) 2005-06-27
MXPA04005484A (es) 2004-12-06
JP2005523245A (ja) 2005-08-04
ES2333784T3 (es) 2010-03-01
ATE441662T1 (de) 2009-09-15
KR20040066167A (ko) 2004-07-23
FR2833596A1 (fr) 2003-06-20
DK1456229T3 (da) 2010-01-04

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Legal Events

Date Code Title Description
ST Notification of lapse

Effective date: 20120831