FI943808A - Triatsolopyrimidiinijohdannaisia angiotensiini II:n reseptoreiden vastavaikuttajina - Google Patents

Triatsolopyrimidiinijohdannaisia angiotensiini II:n reseptoreiden vastavaikuttajina Download PDF

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Publication number
FI943808A
FI943808A FI943808A FI943808A FI943808A FI 943808 A FI943808 A FI 943808A FI 943808 A FI943808 A FI 943808A FI 943808 A FI943808 A FI 943808A FI 943808 A FI943808 A FI 943808A
Authority
FI
Finland
Prior art keywords
angiotensin
receptor antagonists
triazolopyrimidine derivatives
derivatives
treatment
Prior art date
Application number
FI943808A
Other languages
English (en)
Swedish (sv)
Other versions
FI943808A0 (fi
Inventor
Nicole Bru-Magniez
Timur Guengor
Jean-Marie Teulon
Original Assignee
Union Pharma Scient Appl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9202109A external-priority patent/FR2687676B1/fr
Application filed by Union Pharma Scient Appl filed Critical Union Pharma Scient Appl
Publication of FI943808A0 publication Critical patent/FI943808A0/fi
Publication of FI943808A publication Critical patent/FI943808A/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Cardiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI943808A 1992-02-24 1994-08-19 Triatsolopyrimidiinijohdannaisia angiotensiini II:n reseptoreiden vastavaikuttajina FI943808A (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9202109A FR2687676B1 (fr) 1992-02-24 1992-02-24 Nouveaux derives de polyazaindenes antagonistes des recepteurs a l'angiotensine ii; leurs procedes de preparation, compositions pharmaceutiques les contenant.
FR9205417A FR2687677B1 (fr) 1992-02-24 1992-04-30 Nouveaux derives de polyazaindenes antagonistes des recepteurs a l'angiotensine ii ; leurs procedes de preparation, compositions pharmaceutiques les contenant.
PCT/FR1993/000161 WO1993017024A1 (fr) 1992-02-24 1993-02-18 Derives de triazolopyrimidines antagonistes des recepteurs a l'angiotensine ii

Publications (2)

Publication Number Publication Date
FI943808A0 FI943808A0 (fi) 1994-08-19
FI943808A true FI943808A (fi) 1994-10-24

Family

ID=26229283

Family Applications (2)

Application Number Title Priority Date Filing Date
FI943808A FI943808A (fi) 1992-02-24 1994-08-19 Triatsolopyrimidiinijohdannaisia angiotensiini II:n reseptoreiden vastavaikuttajina
FI943807A FI943807A (fi) 1992-02-24 1994-08-19 Pyratsolopyrimidiinijohdannaisia angiotensiini II:n reseptoreiden vastavaikuttajina

Family Applications After (1)

Application Number Title Priority Date Filing Date
FI943807A FI943807A (fi) 1992-02-24 1994-08-19 Pyratsolopyrimidiinijohdannaisia angiotensiini II:n reseptoreiden vastavaikuttajina

Country Status (19)

Country Link
EP (2) EP0628046B1 (fi)
JP (2) JP3372040B2 (fi)
KR (2) KR100272922B1 (fi)
AT (1) ATE179979T1 (fi)
AU (2) AU668139B2 (fi)
CA (2) CA2128871A1 (fi)
CZ (2) CZ282075B6 (fi)
DE (1) DE69324910T2 (fi)
EE (2) EE03045B1 (fi)
ES (1) ES2133390T3 (fi)
FI (2) FI943808A (fi)
FR (1) FR2687677B1 (fi)
HU (2) HUT70953A (fi)
MD (2) MD554G2 (fi)
NZ (2) NZ249509A (fi)
RU (1) RU2116308C1 (fi)
SK (2) SK99894A3 (fi)
TW (2) TW221438B (fi)
WO (2) WO1993017024A1 (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5389632A (en) * 1992-02-24 1995-02-14 Laboratoires Upsa Pyrazolopyrimidine derivatives which are angiotensin II receptor antagonists
IT1263804B (it) * 1993-01-22 1996-09-03 Luso Farmaco Inst Derivati pirimidinonici fusi con eterocicli azotati ad attivita' a ii antagonista
US5571813A (en) * 1993-06-10 1996-11-05 Beiersdorf-Lilly Gmbh Fused pyrimidine compounds and their use as pharmaceuticals
US20080188494A1 (en) * 2005-04-25 2008-08-07 Basf Aktiengesellschaft Use Of 5-Alkyl-6-Phenylalkyl-7-Aminoazolopyrimidines, Novel Azolopyrimidines, Processes For Their Preparation And Compositions Comprising Them
WO2008003753A1 (en) * 2006-07-07 2008-01-10 Biovitrum Ab (Publ) Pyrazolo [1,5-a] pyrimidine analogs for use as inhibitors of stearoyl-coa desaturase (scd) activity
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
RS53012B (en) * 2009-01-30 2014-04-30 Takeda Pharmaceutical Company Limited CONDENSED RING UNIT AND ITS USE
WO2012041817A1 (en) 2010-09-27 2012-04-05 Proximagen Ltd 7-hydroxy-pyrazolo[1,5-a] pyrimidine compounds and their use as ccr2 receptor antagonists

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL94390A (en) * 1989-05-30 1996-03-31 Merck & Co Inc The 6-membered trans-nitrogen-containing heterocycles are compressed with imidazo and pharmaceutical preparations containing them
CA2079344A1 (en) * 1990-03-30 1991-10-01 Eric E. Allen Substituted pyrimidines, pyrimidinones and pyridopyrimidines
FR2678618B1 (fr) * 1991-07-05 1993-11-05 Upsa Laboratoires Nouveaux derives de triazolo pyrimidine antagonistes des recepteurs a l'angiotensine ii; leurs procedes de preparation, compositions pharmaceutiques les contenant.

Also Published As

Publication number Publication date
AU668544B2 (en) 1996-05-09
AU3635893A (en) 1993-09-13
KR100272922B1 (ko) 2001-02-01
HU220392B (hu) 2002-01-28
ES2133390T3 (es) 1999-09-16
RU94040854A (ru) 1996-08-10
EE03046B1 (et) 1997-10-15
HU9402430D0 (en) 1994-10-28
CZ282075B6 (cs) 1997-05-14
RU2116308C1 (ru) 1998-07-27
MD553G2 (ro) 1996-12-31
MD553F1 (en) 1996-05-31
MD554G2 (ro) 1997-01-31
CZ204494A3 (en) 1994-12-15
DE69324910T2 (de) 1999-10-21
EP0628045A1 (fr) 1994-12-14
EE03045B1 (et) 1997-10-15
EP0628046B1 (fr) 1999-05-12
CA2128876A1 (en) 1993-09-02
HU9402429D0 (en) 1994-10-28
MD554F1 (en) 1996-05-31
WO1993017024A1 (fr) 1993-09-02
TW221438B (fi) 1994-03-01
TW222275B (fi) 1994-04-11
CA2128876C (en) 2004-02-03
JP3372040B2 (ja) 2003-01-27
CA2128871A1 (en) 1993-09-02
CZ204594A3 (en) 1994-12-15
ATE179979T1 (de) 1999-05-15
EP0628046A1 (fr) 1994-12-14
KR950700302A (ko) 1995-01-16
AU3635793A (en) 1993-09-13
FI943807A (fi) 1994-10-24
KR950700303A (ko) 1995-01-16
FR2687677B1 (fr) 1996-10-11
SK99894A3 (en) 1995-04-12
JPH07504178A (ja) 1995-05-11
FI943807A0 (fi) 1994-08-19
WO1993017023A1 (fr) 1993-09-02
SK99794A3 (en) 1995-04-12
SK280343B6 (sk) 1999-12-10
AU668139B2 (en) 1996-04-26
NZ249508A (en) 1996-07-26
JPH07504177A (ja) 1995-05-11
HUT70949A (en) 1995-11-28
DE69324910D1 (de) 1999-06-17
FR2687677A1 (fr) 1993-08-27
NZ249509A (en) 1996-06-25
HUT70953A (en) 1995-11-28
FI943808A0 (fi) 1994-08-19

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