EE03045B1 - Angiotensiin II retseptorite antagonistide pürasolopürimidiinide derivaadid, nende valmistamise meetod ja ravimvormid - Google Patents

Angiotensiin II retseptorite antagonistide pürasolopürimidiinide derivaadid, nende valmistamise meetod ja ravimvormid

Info

Publication number
EE03045B1
EE03045B1 EE9400440A EE9400440A EE03045B1 EE 03045 B1 EE03045 B1 EE 03045B1 EE 9400440 A EE9400440 A EE 9400440A EE 9400440 A EE9400440 A EE 9400440A EE 03045 B1 EE03045 B1 EE 03045B1
Authority
EE
Estonia
Prior art keywords
angiotensin
formulations
preparation
receptor antagonists
pyrazolopyrimidine derivatives
Prior art date
Application number
EE9400440A
Other languages
English (en)
Estonian (et)
Inventor
Bru-Magniez Nicole
G�ngor Timur
Teulon Jean-Marie
Original Assignee
Laboratoires Upsa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9202109A external-priority patent/FR2687676B1/fr
Application filed by Laboratoires Upsa filed Critical Laboratoires Upsa
Publication of EE03045B1 publication Critical patent/EE03045B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
EE9400440A 1992-02-24 1994-11-22 Angiotensiin II retseptorite antagonistide pürasolopürimidiinide derivaadid, nende valmistamise meetod ja ravimvormid EE03045B1 (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9202109A FR2687676B1 (fr) 1992-02-24 1992-02-24 Nouveaux derives de polyazaindenes antagonistes des recepteurs a l'angiotensine ii; leurs procedes de preparation, compositions pharmaceutiques les contenant.
FR9205417A FR2687677B1 (fr) 1992-02-24 1992-04-30 Nouveaux derives de polyazaindenes antagonistes des recepteurs a l'angiotensine ii ; leurs procedes de preparation, compositions pharmaceutiques les contenant.
PCT/FR1993/000160 WO1993017023A1 (fr) 1992-02-24 1993-02-18 Derives de pyrazolopyrimidines antagonistes des recepteurs a l'angiotensine ii

Publications (1)

Publication Number Publication Date
EE03045B1 true EE03045B1 (et) 1997-10-15

Family

ID=26229283

Family Applications (2)

Application Number Title Priority Date Filing Date
EE9400441A EE03046B1 (et) 1992-02-24 1994-11-22 Angiotensiin II retseptorite antagonistide triasolopürimidiinide derivaadid, nende valmistamise meetod ja ravimvormid
EE9400440A EE03045B1 (et) 1992-02-24 1994-11-22 Angiotensiin II retseptorite antagonistide pürasolopürimidiinide derivaadid, nende valmistamise meetod ja ravimvormid

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EE9400441A EE03046B1 (et) 1992-02-24 1994-11-22 Angiotensiin II retseptorite antagonistide triasolopürimidiinide derivaadid, nende valmistamise meetod ja ravimvormid

Country Status (19)

Country Link
EP (2) EP0628046B1 (xx)
JP (2) JP3372040B2 (xx)
KR (2) KR100272922B1 (xx)
AT (1) ATE179979T1 (xx)
AU (2) AU668139B2 (xx)
CA (2) CA2128876C (xx)
CZ (2) CZ204594A3 (xx)
DE (1) DE69324910T2 (xx)
EE (2) EE03046B1 (xx)
ES (1) ES2133390T3 (xx)
FI (2) FI943808A (xx)
FR (1) FR2687677B1 (xx)
HU (2) HU220392B (xx)
MD (2) MD553G2 (xx)
NZ (2) NZ249509A (xx)
RU (1) RU2116308C1 (xx)
SK (2) SK280343B6 (xx)
TW (2) TW222275B (xx)
WO (2) WO1993017023A1 (xx)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5389632A (en) * 1992-02-24 1995-02-14 Laboratoires Upsa Pyrazolopyrimidine derivatives which are angiotensin II receptor antagonists
IT1263804B (it) * 1993-01-22 1996-09-03 Luso Farmaco Inst Derivati pirimidinonici fusi con eterocicli azotati ad attivita' a ii antagonista
US5571813A (en) * 1993-06-10 1996-11-05 Beiersdorf-Lilly Gmbh Fused pyrimidine compounds and their use as pharmaceuticals
EP1876899A2 (de) * 2005-04-25 2008-01-16 Basf Aktiengesellschaft Verwendung von 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidinen, neue azolopyrimidine, verfahren zu ihrer herstellung und sie enthaltende mittel
WO2008003753A1 (en) * 2006-07-07 2008-01-10 Biovitrum Ab (Publ) Pyrazolo [1,5-a] pyrimidine analogs for use as inhibitors of stearoyl-coa desaturase (scd) activity
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
TW201444848A (zh) * 2009-01-30 2014-12-01 Takeda Pharmaceutical 稠環化合物及其用途
BR112013008695A2 (pt) 2010-09-27 2016-06-21 Proximagen Ltd compostos de 7-hidróxi-pirazol[1,5-a] pirimidina e seu uso como antagonistas do receptor ccr2

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL94390A (en) * 1989-05-30 1996-03-31 Merck & Co Inc The 6-membered trans-nitrogen-containing heterocycles are compressed with imidazo and pharmaceutical preparations containing them
CA2079344A1 (en) * 1990-03-30 1991-10-01 Eric E. Allen Substituted pyrimidines, pyrimidinones and pyridopyrimidines
FR2678618B1 (fr) * 1991-07-05 1993-11-05 Upsa Laboratoires Nouveaux derives de triazolo pyrimidine antagonistes des recepteurs a l'angiotensine ii; leurs procedes de preparation, compositions pharmaceutiques les contenant.

Also Published As

Publication number Publication date
EP0628046B1 (fr) 1999-05-12
CA2128871A1 (en) 1993-09-02
WO1993017024A1 (fr) 1993-09-02
HU9402429D0 (en) 1994-10-28
CA2128876A1 (en) 1993-09-02
WO1993017023A1 (fr) 1993-09-02
KR950700303A (ko) 1995-01-16
AU3635893A (en) 1993-09-13
CZ282075B6 (cs) 1997-05-14
MD553G2 (ro) 1996-12-31
DE69324910D1 (de) 1999-06-17
KR100272922B1 (ko) 2001-02-01
DE69324910T2 (de) 1999-10-21
NZ249508A (en) 1996-07-26
NZ249509A (en) 1996-06-25
RU2116308C1 (ru) 1998-07-27
FI943807A0 (fi) 1994-08-19
EP0628046A1 (fr) 1994-12-14
TW222275B (xx) 1994-04-11
SK99794A3 (en) 1995-04-12
EE03046B1 (et) 1997-10-15
CZ204594A3 (en) 1994-12-15
EP0628045A1 (fr) 1994-12-14
MD554F1 (en) 1996-05-31
AU668544B2 (en) 1996-05-09
FR2687677A1 (fr) 1993-08-27
ES2133390T3 (es) 1999-09-16
KR950700302A (ko) 1995-01-16
HU220392B (hu) 2002-01-28
HUT70949A (en) 1995-11-28
JPH07504177A (ja) 1995-05-11
TW221438B (xx) 1994-03-01
SK99894A3 (en) 1995-04-12
AU668139B2 (en) 1996-04-26
JP3372040B2 (ja) 2003-01-27
CZ204494A3 (en) 1994-12-15
CA2128876C (en) 2004-02-03
FI943808A0 (fi) 1994-08-19
HUT70953A (en) 1995-11-28
MD553F1 (en) 1996-05-31
FI943807A (fi) 1994-10-24
FI943808A (fi) 1994-10-24
MD554G2 (ro) 1997-01-31
AU3635793A (en) 1993-09-13
JPH07504178A (ja) 1995-05-11
SK280343B6 (sk) 1999-12-10
FR2687677B1 (fr) 1996-10-11
HU9402430D0 (en) 1994-10-28
ATE179979T1 (de) 1999-05-15
RU94040854A (ru) 1996-08-10

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Legal Events

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KB4A Valid patent at the end of a year

Effective date: 20021231

KB4A Valid patent at the end of a year

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KB4A Valid patent at the end of a year

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Effective date: 20101231