FI943222A - Uusia adenosiinijohdannaisia, menetelmä niiden valmistamiseksi sekä niitä sisältäviä lääkeyhdisteitä - Google Patents

Uusia adenosiinijohdannaisia, menetelmä niiden valmistamiseksi sekä niitä sisältäviä lääkeyhdisteitä Download PDF

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Publication number
FI943222A
FI943222A FI943222A FI943222A FI943222A FI 943222 A FI943222 A FI 943222A FI 943222 A FI943222 A FI 943222A FI 943222 A FI943222 A FI 943222A FI 943222 A FI943222 A FI 943222A
Authority
FI
Finland
Prior art keywords
manufacture
processes
those containing
pharmaceutical compounds
containing pharmaceutical
Prior art date
Application number
FI943222A
Other languages
English (en)
Swedish (sv)
Other versions
FI106205B (fi
FI943222A0 (fi
Inventor
Nicole Bru-Magniez
Timur Guengor
Jean-Marie Teulon
Original Assignee
Union Pharma Scient Appl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Union Pharma Scient Appl filed Critical Union Pharma Scient Appl
Publication of FI943222A0 publication Critical patent/FI943222A0/fi
Publication of FI943222A publication Critical patent/FI943222A/fi
Application granted granted Critical
Publication of FI106205B publication Critical patent/FI106205B/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Pain & Pain Management (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI943222A 1992-01-08 1994-07-06 Menetelmä terapeuttisesti aktiivisten adenosiinijohdannaisten valmistamiseksi FI106205B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR9200138 1992-01-08
FR9200138A FR2685918B1 (fr) 1992-01-08 1992-01-08 Nouveaux derives de l'adenosine, leurs procedes de preparation, compositions pharmaceutiques les contenant.
PCT/FR1992/001241 WO1993014102A1 (fr) 1992-01-08 1992-12-29 Nouveaux derives de l'adenosine, leurs procedes de preparation, compositions pharmaceutiques les contenant
FR9201241 1992-12-29

Publications (3)

Publication Number Publication Date
FI943222A0 FI943222A0 (fi) 1994-07-06
FI943222A true FI943222A (fi) 1994-08-18
FI106205B FI106205B (fi) 2000-12-15

Family

ID=9425478

Family Applications (1)

Application Number Title Priority Date Filing Date
FI943222A FI106205B (fi) 1992-01-08 1994-07-06 Menetelmä terapeuttisesti aktiivisten adenosiinijohdannaisten valmistamiseksi

Country Status (25)

Country Link
US (2) US5229505A (fi)
EP (1) EP0623138B1 (fi)
JP (1) JP3224542B2 (fi)
KR (1) KR100232672B1 (fi)
AT (1) ATE153342T1 (fi)
AU (1) AU661894B2 (fi)
CA (1) CA2127472C (fi)
CZ (1) CZ289047B6 (fi)
DE (1) DE69219901T2 (fi)
DK (1) DK0623138T3 (fi)
EE (1) EE03087B1 (fi)
ES (1) ES2105285T3 (fi)
FI (1) FI106205B (fi)
FR (1) FR2685918B1 (fi)
GE (1) GEP19981357B (fi)
GR (1) GR3024386T3 (fi)
HU (1) HU221304B1 (fi)
LV (1) LV11899B (fi)
MD (1) MD502G2 (fi)
NZ (1) NZ246904A (fi)
RU (1) RU2129560C1 (fi)
SK (1) SK282205B6 (fi)
TW (1) TW254945B (fi)
UA (1) UA44221C2 (fi)
WO (1) WO1993014102A1 (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2685918B1 (fr) * 1992-01-08 1995-06-23 Union Pharma Scient Appl Nouveaux derives de l'adenosine, leurs procedes de preparation, compositions pharmaceutiques les contenant.
FR2714907B1 (fr) * 1994-01-07 1996-03-29 Union Pharma Scient Appl Nouveaux dérivés de l'Adénosine, leurs procédés de préparation, compositions pharmaceutiques les contenant.
WO1995018817A1 (fr) * 1994-01-07 1995-07-13 Laboratoires Upsa Nouveaux derives de l'adenosine, leurs procedes de preparation, compositions pharmaceutiques les contenant
TW528755B (en) 1996-12-24 2003-04-21 Glaxo Group Ltd 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives
FR2772271B1 (fr) * 1997-12-11 2000-09-01 Union Pharma Scient Appl Nouvelle association pharmaceutique a activite analgesique
YU44900A (sh) 1998-01-31 2003-01-31 Glaxo Group Limited Derivati 2-(purin-9-il)tetrahidrofuran-3,4-diola
YU81100A (sh) 1998-06-23 2003-10-31 Glaxo Group Limited Derivati 2-(purin-9-il)tetrahidrofuran-3,4 diola
JP2002173427A (ja) * 1998-09-01 2002-06-21 Yamasa Shoyu Co Ltd 眼疾患治療用医薬組成物
DE19924818A1 (de) * 1999-05-29 2000-11-30 Bayer Ag Substituierte Phenylcyclohexancarbonsäureamide
WO2001035928A1 (en) * 1999-11-17 2001-05-25 Microchips, Inc. Microfabricated devices for the delivery of molecules into a carrier fluid
AU2001278708A1 (en) * 2000-09-08 2002-03-22 Toa Eiyo Ltd. Adenosine derivatives and use thereof
EP1352910A1 (en) * 2002-04-10 2003-10-15 Grünenthal GmbH New analogs of nitrobenzylthioinosine
AR049384A1 (es) 2004-05-24 2006-07-26 Glaxo Group Ltd Derivados de purina
GB0514809D0 (en) 2005-07-19 2005-08-24 Glaxo Group Ltd Compounds

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE788958A (fr) * 1971-09-18 1973-03-19 Schering Ag Derives d'adenosine et leur procede de preparation
US4167565A (en) * 1976-11-08 1979-09-11 Abbott Laboratories Adenosine-5'-carboxamides and method of use
US5310731A (en) * 1984-06-28 1994-05-10 Whitby Research, Inc. N-6 substituted-5'-(N-substitutedcarboxamido)adenosines as cardiac vasodilators and antihypertensive agents
US4755594A (en) * 1986-01-31 1988-07-05 Warner-Lambert Company N6 -substituted adenosines
JPH0696534B2 (ja) * 1986-04-25 1994-11-30 ヘキストジヤパン株式会社 抗痴呆剤
AU8276187A (en) * 1986-10-31 1988-05-25 Warner-Lambert Company Selected n6-substituted adenosines having selective a2 binding activity
AU8274187A (en) * 1986-10-31 1988-05-25 Warner-Lambert Company Heteroaromatic derivatives of adenosine
IL84414A0 (en) * 1986-11-14 1988-04-29 Ciba Geigy Ag N9-cyclopentyl-substituted adenine derivatives
SU1661367A1 (ru) * 1988-11-01 1991-07-07 Всесоюзный научно-исследовательский институт по креплению скважин и буровым растворам Способ гидрофобизации тампонажных материалов
AU654507B2 (en) * 1990-09-25 1994-11-10 Rhone-Poulenc Rorer International (Holdings) Inc. Compounds having antihypertensive and anti-ischemic properties
FR2685918B1 (fr) * 1992-01-08 1995-06-23 Union Pharma Scient Appl Nouveaux derives de l'adenosine, leurs procedes de preparation, compositions pharmaceutiques les contenant.

Also Published As

Publication number Publication date
LV11899B (lv) 1998-03-20
HU221304B1 (en) 2002-09-28
SK282205B6 (sk) 2001-12-03
FI106205B (fi) 2000-12-15
ES2105285T3 (es) 1997-10-16
JPH07502738A (ja) 1995-03-23
US5480983A (en) 1996-01-02
AU661894B2 (en) 1995-08-10
EP0623138A1 (fr) 1994-11-09
DK0623138T3 (da) 1997-12-15
HU9402040D0 (en) 1994-09-28
RU94039545A (ru) 1997-04-27
GEP19981357B (en) 1998-08-25
KR100232672B1 (ko) 1999-12-01
MD502G2 (ro) 1996-11-30
JP3224542B2 (ja) 2001-10-29
HUT68095A (en) 1995-05-29
MD502F1 (en) 1996-03-29
CZ289047B6 (cs) 2001-10-17
EP0623138B1 (fr) 1997-05-21
SK81894A3 (en) 1995-04-12
DE69219901T2 (de) 1997-11-13
CZ164394A3 (en) 1995-02-15
CA2127472A1 (en) 1993-07-22
FR2685918B1 (fr) 1995-06-23
NZ246904A (en) 1995-04-27
EE03087B1 (et) 1998-04-15
AU3455093A (en) 1993-08-03
US5229505A (en) 1993-07-20
ATE153342T1 (de) 1997-06-15
CA2127472C (en) 2003-11-18
GR3024386T3 (en) 1997-11-28
FR2685918A1 (fr) 1993-07-09
DE69219901D1 (de) 1997-06-26
RU2129560C1 (ru) 1999-04-27
UA44221C2 (uk) 2002-02-15
WO1993014102A1 (fr) 1993-07-22
FI943222A0 (fi) 1994-07-06
TW254945B (fi) 1995-08-21
LV11899A (lv) 1997-12-20

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