FI902845A0 - Menetelmä 4-amino-1-hydroksibutylideeni-1,1-bisfosfonihapon tai sen suolojen valmistamiseksi - Google Patents

Menetelmä 4-amino-1-hydroksibutylideeni-1,1-bisfosfonihapon tai sen suolojen valmistamiseksi

Info

Publication number
FI902845A0
FI902845A0 FI902845A FI902845A FI902845A0 FI 902845 A0 FI902845 A0 FI 902845A0 FI 902845 A FI902845 A FI 902845A FI 902845 A FI902845 A FI 902845A FI 902845 A0 FI902845 A0 FI 902845A0
Authority
FI
Finland
Prior art keywords
salts
amino
hydroxybutylidene
preparation
bisphosphonic acid
Prior art date
Application number
FI902845A
Other languages
English (en)
Swedish (sv)
Other versions
FI93219C (fi
FI93219B (fi
Inventor
Gerard R Kieczykowski
Ronald B Jobson
David G Melillo
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23431886&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI902845(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of FI902845A0 publication Critical patent/FI902845A0/fi
Application granted granted Critical
Publication of FI93219B publication Critical patent/FI93219B/fi
Publication of FI93219C publication Critical patent/FI93219C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se)
    • C07F9/3804—Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se) not used, see subgroups
    • C07F9/3839—Polyphosphonic acids
    • C07F9/3873—Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Seasonings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
FI902845A 1989-06-09 1990-06-07 Menetelmä 4-amino-1-hydroksibutylideeni-1,1-bisfosfonihapon tai sen suolojen valmistamiseksi FI93219C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US36382089 1989-06-09
US07/363,820 US4922007A (en) 1989-06-09 1989-06-09 Process for preparing 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid or salts thereof

Publications (3)

Publication Number Publication Date
FI902845A0 true FI902845A0 (fi) 1990-06-07
FI93219B FI93219B (fi) 1994-11-30
FI93219C FI93219C (fi) 1995-03-10

Family

ID=23431886

Family Applications (1)

Application Number Title Priority Date Filing Date
FI902845A FI93219C (fi) 1989-06-09 1990-06-07 Menetelmä 4-amino-1-hydroksibutylideeni-1,1-bisfosfonihapon tai sen suolojen valmistamiseksi

Country Status (23)

Country Link
US (1) US4922007A (fi)
EP (1) EP0402152B1 (fi)
JP (2) JPH0662651B2 (fi)
KR (1) KR0137455B1 (fi)
AT (1) ATE129713T1 (fi)
AU (1) AU625704C (fi)
CA (1) CA2018477C (fi)
CH (1) CH0402152H1 (fi)
CY (1) CY1894A (fi)
DE (1) DE69023280T2 (fi)
DK (1) DK0402152T3 (fi)
ES (1) ES2080116T3 (fi)
FI (1) FI93219C (fi)
GR (1) GR3018379T3 (fi)
HK (1) HK69596A (fi)
HU (1) HU211908A9 (fi)
IE (1) IE69564B1 (fi)
IL (1) IL94612A (fi)
LV (1) LV11472B (fi)
NO (2) NO177997C (fi)
NZ (1) NZ233972A (fi)
PT (1) PT94306B (fi)
ZA (1) ZA904446B (fi)

Families Citing this family (118)

* Cited by examiner, † Cited by third party
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JPH0748391A (ja) 1995-02-21
NO902559D0 (no) 1990-06-08
AU625704B2 (en) 1992-07-16
CY1894A (en) 1990-06-08
HU211908A9 (en) 1996-01-29
NZ233972A (en) 1992-05-26
IL94612A (en) 1995-03-30
KR910000768A (ko) 1991-01-30
PT94306B (pt) 1997-05-28
NO902559L (no) 1990-12-10
LV11472A (lv) 1996-08-20
CH0402152H1 (fr) 2006-02-28
FI93219C (fi) 1995-03-10
CA2018477A1 (en) 1990-12-09
KR0137455B1 (ko) 1998-05-01
PT94306A (pt) 1991-02-08
IL94612A0 (en) 1991-04-15
EP0402152A3 (en) 1991-07-03
DK0402152T3 (da) 1995-12-04
DE69023280T2 (de) 1996-06-20
NO941726D0 (no) 1994-05-09
CA2018477C (en) 1995-08-01
IE902073L (en) 1990-12-09
IE69564B1 (en) 1996-10-02
AU625704C (en) 2001-07-26
NO178228B (no) 1995-11-06
JPH03101684A (ja) 1991-04-26
ZA904446B (en) 1992-06-24
NO178228C (no) 1996-02-14
ATE129713T1 (de) 1995-11-15
US4922007A (en) 1990-05-01
NO177997B (no) 1995-09-25
EP0402152B1 (en) 1995-11-02
ES2080116T3 (es) 1996-02-01
HK69596A (en) 1996-04-26
DE69023280D1 (de) 1995-12-07
EP0402152A2 (en) 1990-12-12
JPH0662651B2 (ja) 1994-08-17
GR3018379T3 (en) 1996-03-31
NO177997C (no) 1996-01-03
NO941726L (no) 1990-12-10
FI93219B (fi) 1994-11-30
AU5701990A (en) 1990-12-13
LV11472B (en) 1996-12-20

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