FI864272A - Infusionsloesningar av 1-cyklopropyl-6-fluor-1,4-dihydro-4-oxo-7-(1-piperazinyl)-kinolin-3 -karboxylsyra. - Google Patents

Infusionsloesningar av 1-cyklopropyl-6-fluor-1,4-dihydro-4-oxo-7-(1-piperazinyl)-kinolin-3 -karboxylsyra. Download PDF

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Publication number
FI864272A
FI864272A FI864272A FI864272A FI864272A FI 864272 A FI864272 A FI 864272A FI 864272 A FI864272 A FI 864272A FI 864272 A FI864272 A FI 864272A FI 864272 A FI864272 A FI 864272A
Authority
FI
Finland
Prior art keywords
infusionsloesningar
carboxylsyra
quinolin
fluor
piperazinyl
Prior art date
Application number
FI864272A
Other languages
English (en)
Other versions
FI84555B (fi
FI84555C (fi
FI864272A0 (fi
Inventor
Robert Frank Lammens
Hans Friedrich Mahler
Peter Serno
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6284294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI864272(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of FI864272A0 publication Critical patent/FI864272A0/fi
Publication of FI864272A publication Critical patent/FI864272A/fi
Publication of FI84555B publication Critical patent/FI84555B/fi
Application granted granted Critical
Publication of FI84555C publication Critical patent/FI84555C/fi

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
FI864272A 1985-10-24 1986-10-22 Foerfarande foer framstaellning av infusionsloesningar som innehaoller 1-cyklopropyl-6-fluor-1,4-dihydro-4- oxo-7-(1-piperazinyl)-kinolin-3-karboxylsyra. FI84555C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3537761 1985-10-24
DE19853537761 DE3537761A1 (de) 1985-10-24 1985-10-24 Infusionsloesungen der 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7- (1-piperazinyl)-chinolin-3-carbonsaeure

Publications (4)

Publication Number Publication Date
FI864272A0 FI864272A0 (fi) 1986-10-22
FI864272A true FI864272A (fi) 1987-04-25
FI84555B FI84555B (fi) 1991-09-13
FI84555C FI84555C (fi) 1991-12-27

Family

ID=6284294

Family Applications (1)

Application Number Title Priority Date Filing Date
FI864272A FI84555C (fi) 1985-10-24 1986-10-22 Foerfarande foer framstaellning av infusionsloesningar som innehaoller 1-cyklopropyl-6-fluor-1,4-dihydro-4- oxo-7-(1-piperazinyl)-kinolin-3-karboxylsyra.

Country Status (27)

Country Link
US (1) US4957922A (fi)
EP (1) EP0219784B1 (fi)
JP (1) JPH0714879B2 (fi)
KR (1) KR940002664B1 (fi)
AR (1) AR244085A1 (fi)
AT (1) ATE59003T1 (fi)
AU (1) AU571796B2 (fi)
CA (1) CA1282006C (fi)
CY (1) CY1729A (fi)
DD (1) DD252125A5 (fi)
DE (2) DE3537761A1 (fi)
DK (1) DK175494B1 (fi)
ES (1) ES2021571B3 (fi)
FI (1) FI84555C (fi)
GR (1) GR3002544T3 (fi)
HK (1) HK115593A (fi)
HU (1) HUT42952A (fi)
IE (1) IE59385B1 (fi)
IL (1) IL80380A (fi)
NO (1) NO864022L (fi)
NZ (1) NZ218016A (fi)
PH (1) PH26419A (fi)
PL (1) PL152336B1 (fi)
PT (1) PT83588B (fi)
SU (1) SU1487801A3 (fi)
UA (1) UA8033A1 (fi)
ZA (1) ZA868057B (fi)

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JP2006151808A (ja) * 2002-12-24 2006-06-15 Dai Ichi Seiyaku Co Ltd 抗菌性水性製剤
US6861422B2 (en) * 2003-02-26 2005-03-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions
DE102004005186B3 (de) * 2004-02-02 2005-10-13 Krka Tovarna Zdravil, D.D. Verfahren zur Herstellung von gereinigtem Ciprofloxacin
WO2005123137A2 (en) * 2004-06-18 2005-12-29 Ranbaxy Laboratories Limited Lyophilized pharmaceutical composition comprising moxifloxacin hydrochloride
DE102004029784A1 (de) * 2004-06-21 2006-01-05 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue 2-Benzylaminodihydropteridinone, Verfahren zur deren Herstellung und deren Verwendung als Arzneimittel
DE102004033670A1 (de) * 2004-07-09 2006-02-02 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Pyridodihydropyrazinone, Verfahren zu Ihrer Herstellung und Ihre Verwendung als Arzneimittel
US20060035903A1 (en) * 2004-08-14 2006-02-16 Boehringer Ingelheim International Gmbh Storage stable perfusion solution for dihydropteridinones
US7728134B2 (en) * 2004-08-14 2010-06-01 Boehringer Ingelheim International Gmbh Hydrates and polymorphs of 4[[(7R)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-6-oxo-2-pteridinyl]amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide, process for their manufacture and their use as medicament
US20060058311A1 (en) 2004-08-14 2006-03-16 Boehringer Ingelheim International Gmbh Combinations for the treatment of diseases involving cell proliferation
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US20060074088A1 (en) * 2004-08-14 2006-04-06 Boehringer Ingelheim International Gmbh Dihydropteridinones for the treatment of cancer diseases
EP1632493A1 (de) * 2004-08-25 2006-03-08 Boehringer Ingelheim Pharma GmbH & Co.KG Dihydropteridinonderivative, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
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DE102004054873A1 (de) 2004-11-12 2006-05-18 Bayer Healthcare Ag Behandlung von Mastitis
DE102004058337A1 (de) * 2004-12-02 2006-06-14 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung von annelierten Piperazin-2-on Derivaten
EP1827498A2 (de) * 2004-12-09 2007-09-05 Bayer HealthCare AG Stabilisierung von glucocorticoidestern mit säuren
DE102005055385A1 (de) * 2004-12-09 2006-06-14 Bayer Healthcare Ag Arzneimittel zur hygienischen Applikation im Ohr
FR2896416B1 (fr) * 2006-01-24 2010-08-13 Vetoquinol Composition anti-infectieuse comprenant un compose de type pyrido (3,2,1-ij)-benzoxadiazine
US7439358B2 (en) * 2006-02-08 2008-10-21 Boehringer Ingelheim International Gmbh Specific salt, anhydrous and crystalline form of a dihydropteridione derivative
US20070197548A1 (en) * 2006-02-17 2007-08-23 Murthy Yerramilli V S Fluoroquinolone compositions
TW200900066A (en) * 2007-03-22 2009-01-01 Daiichi Sankyo Co Ltd Quinolone medical composition containing alcohols
BRPI0810192C1 (pt) * 2007-04-13 2021-05-25 Dong Wha Pharm Co Ltd aspartato do ácido 1-ciclopropil-6-fluoro-7-(8-metoxiimino-2,6-diaza-espiro [3,4] oct-6-il)-4-oxo-1,4-diidro- [1,8] naftiridina-3-carboxílico, método para preparação do mesmo e composição farmacêutica antimicrobiana compreendendo o mesmo.
JP5217276B2 (ja) * 2007-07-19 2013-06-19 ニプロ株式会社 注射用抗菌剤の製造方法
JP5261487B2 (ja) * 2007-08-03 2013-08-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ジヒドロプテリジノン誘導体の結晶形
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US9358233B2 (en) 2010-11-29 2016-06-07 Boehringer Ingelheim International Gmbh Method for treating acute myeloid leukemia
US9370535B2 (en) 2011-05-17 2016-06-21 Boehringer Ingelheim International Gmbh Method for treatment of advanced solid tumors
JP2016525532A (ja) 2013-07-26 2016-08-25 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 骨髄異形成症候群の処置
KR101646324B1 (ko) * 2014-03-04 2016-08-05 동화약품주식회사 1-시클로프로필-6-플루오로-7-(8-메톡시이미노-2,6-디아자-스피로[3,4]옥트-6-일)-4-옥소-1,4-디히드로-[1,8]나프티리딘-3-카르복실산 디-아스파르트산염의 수화물 및 이를 포함하는 항균활성 조성물
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Also Published As

Publication number Publication date
PH26419A (en) 1992-07-15
PT83588A (en) 1986-11-01
AU571796B2 (en) 1988-04-21
CA1282006C (en) 1991-03-26
HUT42952A (en) 1987-09-28
DK507886A (da) 1987-04-25
AR244085A1 (es) 1993-10-29
PT83588B (pt) 1989-05-31
DE3676158D1 (de) 1991-01-24
CY1729A (en) 1994-05-06
NZ218016A (en) 1989-02-24
DE3537761A1 (de) 1987-04-30
IL80380A0 (en) 1987-01-30
JPH0714879B2 (ja) 1995-02-22
JPS6299326A (ja) 1987-05-08
UA8033A1 (uk) 1995-12-26
KR940002664B1 (ko) 1994-03-28
ATE59003T1 (de) 1990-12-15
EP0219784A2 (de) 1987-04-29
HK115593A (en) 1993-11-05
ZA868057B (en) 1987-06-24
EP0219784B1 (de) 1990-12-12
EP0219784A3 (en) 1987-11-04
NO864022D0 (no) 1986-10-09
ES2021571B3 (es) 1991-11-16
NO864022L (no) 1987-04-27
GR3002544T3 (en) 1993-01-25
PL262006A1 (en) 1988-10-13
FI84555B (fi) 1991-09-13
FI84555C (fi) 1991-12-27
DK507886D0 (da) 1986-10-23
FI864272A0 (fi) 1986-10-22
KR870003786A (ko) 1987-05-04
SU1487801A3 (ru) 1989-06-15
IE862803L (en) 1987-04-24
DD252125A5 (de) 1987-12-09
IL80380A (en) 1990-11-29
PL152336B1 (en) 1990-12-31
DK175494B1 (da) 2004-11-08
IE59385B1 (en) 1994-02-23
AU6432786A (en) 1987-04-30
US4957922A (en) 1990-09-18

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Owner name: BAYER HEALTHCARE AG

MA Patent expired