FI72322C - Foerfarande foer framstaellning av terapeutiskt anvaendbara makrolider. - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbara makrolider. Download PDF

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Publication number
FI72322C
FI72322C FI830585A FI830585A FI72322C FI 72322 C FI72322 C FI 72322C FI 830585 A FI830585 A FI 830585A FI 830585 A FI830585 A FI 830585A FI 72322 C FI72322 C FI 72322C
Authority
FI
Finland
Prior art keywords
formula
preparation
hydrogen
group
macrolide
Prior art date
Application number
FI830585A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI830585A0 (fi
FI830585L (fi
FI72322B (fi
Inventor
Satoshi Omura
Akira Nakagawa
Original Assignee
Satoshi Omura
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Satoshi Omura filed Critical Satoshi Omura
Publication of FI830585A0 publication Critical patent/FI830585A0/fi
Publication of FI830585L publication Critical patent/FI830585L/fi
Application granted granted Critical
Publication of FI72322B publication Critical patent/FI72322B/fi
Publication of FI72322C publication Critical patent/FI72322C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI830585A 1982-02-25 1983-02-22 Foerfarande foer framstaellning av terapeutiskt anvaendbara makrolider. FI72322C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2948082 1982-02-25
JP57029480A JPS58146595A (ja) 1982-02-25 1982-02-25 マクロライド系抗生物質

Publications (4)

Publication Number Publication Date
FI830585A0 FI830585A0 (fi) 1983-02-22
FI830585L FI830585L (fi) 1983-08-26
FI72322B FI72322B (fi) 1987-01-30
FI72322C true FI72322C (fi) 1987-05-11

Family

ID=12277244

Family Applications (1)

Application Number Title Priority Date Filing Date
FI830585A FI72322C (fi) 1982-02-25 1983-02-22 Foerfarande foer framstaellning av terapeutiskt anvaendbara makrolider.

Country Status (24)

Country Link
US (1) US4440759A (enEXAMPLES)
EP (1) EP0087921B1 (enEXAMPLES)
JP (1) JPS58146595A (enEXAMPLES)
KR (1) KR850000962B1 (enEXAMPLES)
AT (1) ATE16008T1 (enEXAMPLES)
AU (1) AU555979B2 (enEXAMPLES)
CA (1) CA1202022A (enEXAMPLES)
CS (1) CS235309B2 (enEXAMPLES)
DD (1) DD210283A5 (enEXAMPLES)
DE (1) DE3360951D1 (enEXAMPLES)
DK (1) DK153795C (enEXAMPLES)
ES (2) ES8403926A1 (enEXAMPLES)
FI (1) FI72322C (enEXAMPLES)
GB (1) GB2115813B (enEXAMPLES)
GR (1) GR78112B (enEXAMPLES)
HU (1) HU194269B (enEXAMPLES)
IL (1) IL67973A0 (enEXAMPLES)
NZ (1) NZ203365A (enEXAMPLES)
PH (1) PH18435A (enEXAMPLES)
PL (1) PL138759B1 (enEXAMPLES)
PT (1) PT76272B (enEXAMPLES)
RO (1) RO85833B (enEXAMPLES)
SU (1) SU1360588A3 (enEXAMPLES)
ZA (1) ZA831206B (enEXAMPLES)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
AU561147B2 (en) * 1982-09-13 1987-04-30 Eli Lilly And Company 20-amino macrolide antibiotics
US4820695A (en) * 1982-09-13 1989-04-11 Eli Lilly And Company C-20-dihydro-deoxy-(cyclic amino)-derivatives of macrolide antibiotics
IL71032A0 (en) * 1983-02-28 1984-05-31 Lilly Co Eli C-20 and c-23-modified macrolide derivatives
US4629786A (en) * 1983-02-28 1986-12-16 Eli Lilly And Company C-20- and C-23 modified macrolide derivatives
ZA841277B (en) * 1983-02-28 1985-09-25 Lilly Co Eli C-20-and c-23-modified macrolide derivatives
US4801721A (en) * 1984-08-16 1989-01-31 Ryan James W Stereospecific synthesis of carboxyalkyl peptides
US4921947A (en) * 1986-03-31 1990-05-01 Eli Lilly And Company Process for preparing macrolide derivatives
FR2638458A1 (fr) * 1988-10-27 1990-05-04 Adir Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW309505B (enEXAMPLES) * 1993-03-31 1997-07-01 Toto Ltd
WO1996009312A1 (en) * 1994-09-22 1996-03-28 Pfizer Inc. Antibiotic macrolides
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
CN110590885A (zh) * 2019-09-30 2019-12-20 郑州大学 20-取代-5-o-碳霉胺糖基-泰乐内酯衍生物
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3178341A (en) * 1960-06-27 1965-04-13 Lilly Co Eli Antibiotics tylosin and desmycosin and derivatives thereof
GB1587685A (en) * 1977-03-09 1981-04-08 Microbial Chem Res Found Macrolactone derivatives and their production
JPS53132584A (en) * 1977-04-26 1978-11-18 Toyo Jozo Co Ltd 18-cyano-18-substituted amino-18-deoxy-macrolide anibiotic substance derivative
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
US4279896A (en) * 1980-06-23 1981-07-21 Schering Corporation Novel 20-imino macrolide antibacterial agents

Also Published As

Publication number Publication date
SU1360588A3 (ru) 1987-12-15
ES520037A0 (es) 1984-04-01
EP0087921B1 (en) 1985-10-09
KR850000962B1 (ko) 1985-07-02
PT76272A (en) 1983-03-01
FI830585A0 (fi) 1983-02-22
DK153795C (da) 1989-01-23
JPS58146595A (ja) 1983-09-01
IL67973A0 (en) 1983-06-15
HU194269B (en) 1988-01-28
ES8505207A1 (es) 1985-05-16
ZA831206B (en) 1983-11-30
FI830585L (fi) 1983-08-26
RO85833B (ro) 1984-11-30
KR840003646A (ko) 1984-09-15
DE3360951D1 (en) 1985-11-14
CA1202022A (en) 1986-03-18
PH18435A (en) 1985-07-08
ES526529A0 (es) 1985-05-16
AU555979B2 (en) 1986-10-16
RO85833A (ro) 1984-11-25
GB2115813B (en) 1985-09-11
NZ203365A (en) 1985-07-12
PT76272B (en) 1986-02-04
CS235309B2 (en) 1985-05-15
EP0087921A1 (en) 1983-09-07
GB2115813A (en) 1983-09-14
DK87783D0 (da) 1983-02-24
DK87783A (da) 1983-08-26
ATE16008T1 (de) 1985-10-15
DD210283A5 (de) 1984-06-06
GR78112B (enEXAMPLES) 1984-09-26
AU1180183A (en) 1983-09-01
JPH0142277B2 (enEXAMPLES) 1989-09-11
GB8305005D0 (en) 1983-03-30
DK153795B (da) 1988-09-05
US4440759A (en) 1984-04-03
PL138759B1 (en) 1986-10-31
FI72322B (fi) 1987-01-30
PL240735A1 (en) 1983-09-26
ES8403926A1 (es) 1984-04-01

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MM Patent lapsed

Owner name: OMURA, SATOSHI