FI66002C - Foerfarande foer framstaellning av nya terapeutiskt anvaendbara substituerade 9,10-dihydro-4h-tieno(3,4-b)(1,5)bensodiazepin-10-oner samt deras syraadditionssalter - Google Patents
Foerfarande foer framstaellning av nya terapeutiskt anvaendbara substituerade 9,10-dihydro-4h-tieno(3,4-b)(1,5)bensodiazepin-10-oner samt deras syraadditionssalter Download PDFInfo
- Publication number
- FI66002C FI66002C FI814028A FI814028A FI66002C FI 66002 C FI66002 C FI 66002C FI 814028 A FI814028 A FI 814028A FI 814028 A FI814028 A FI 814028A FI 66002 C FI66002 C FI 66002C
- Authority
- FI
- Finland
- Prior art keywords
- group
- thieno
- dihydro
- benzodiazepin
- methyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Compositions Of Macromolecular Compounds (AREA)
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH358180 | 1980-05-07 | ||
CH358180 | 1980-05-07 | ||
CH65281 | 1981-02-02 | ||
CH65281 | 1981-02-02 | ||
PCT/EP1981/000042 WO1981003173A1 (en) | 1980-05-07 | 1981-05-06 | Thieno-tricyclic compounds,method for the preparation thereof,utilization of such compounds and drugs containing them |
EP8100042 | 1981-05-06 |
Publications (3)
Publication Number | Publication Date |
---|---|
FI814028L FI814028L (fi) | 1981-12-15 |
FI66002B FI66002B (fi) | 1984-04-30 |
FI66002C true FI66002C (fi) | 1984-08-10 |
Family
ID=25685262
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI814028A FI66002C (fi) | 1980-05-07 | 1981-12-15 | Foerfarande foer framstaellning av nya terapeutiskt anvaendbara substituerade 9,10-dihydro-4h-tieno(3,4-b)(1,5)bensodiazepin-10-oner samt deras syraadditionssalter |
Country Status (21)
Country | Link |
---|---|
EP (1) | EP0039519B1 (da) |
JP (1) | JPS6021994B2 (da) |
KR (1) | KR850000241B1 (da) |
AT (1) | ATE7299T1 (da) |
AU (1) | AU538031B2 (da) |
DD (1) | DD158902A5 (da) |
DE (1) | DE3163361D1 (da) |
DK (1) | DK157872C (da) |
ES (1) | ES8205802A1 (da) |
FI (1) | FI66002C (da) |
GR (1) | GR82676B (da) |
HK (1) | HK6890A (da) |
HU (1) | HU182712B (da) |
IE (1) | IE51200B1 (da) |
IL (1) | IL62792A (da) |
NO (1) | NO156753C (da) |
NZ (1) | NZ197017A (da) |
PL (1) | PL139428B1 (da) |
PT (1) | PT72982B (da) |
WO (1) | WO1981003173A1 (da) |
YU (1) | YU42398B (da) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3204153A1 (de) * | 1982-02-06 | 1983-08-11 | Dr. Karl Thomae Gmbh, 7950 Biberach | Substituierte thienobenzodiazepinone, verfahren zu ihrer herstellung und sie enthaltende arzneimittel |
DE3204169A1 (de) * | 1982-02-06 | 1983-08-11 | Dr. Karl Thomae Gmbh, 7950 Biberach | Substituierte thienobenzodiazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE3409237A1 (de) * | 1984-03-14 | 1985-09-19 | Dr. Karl Thomae Gmbh, 7950 Biberach | Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE3529372A1 (de) * | 1985-08-16 | 1987-02-19 | Dompe Farmaceutici Spa | Aminoacyl-derivat von 4,9-dihydro-10h-pyrido(3,2-b)-thieno(3,2-e) (1,4)-diazepinon und von 4,9-dihydro-10h-pyrido(3,2-b)thieno(3,4-e) (1,4)diazepinon, verfahren zu deren herstellung und diese verbindungen enthaltende pharmazeutische zusammensetzungen |
DE3643666A1 (de) * | 1986-12-20 | 1988-06-30 | Thomae Gmbh Dr K | Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE3726908A1 (de) * | 1987-08-13 | 1989-02-23 | Thomae Gmbh Dr K | Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
WO1989005644A2 (fr) * | 1987-12-22 | 1989-06-29 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Thienotricyclene |
DE3802334A1 (de) * | 1988-01-27 | 1989-08-10 | Thomae Gmbh Dr K | Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE3820345A1 (de) * | 1988-06-15 | 1989-12-21 | Thomae Gmbh Dr K | Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE3820346A1 (de) * | 1988-06-15 | 1989-12-21 | Thomae Gmbh Dr K | Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE4003322C1 (da) * | 1990-02-05 | 1991-06-20 | Byk Gulden Lomberg Chemische Fabrik Gmbh, 7750 Konstanz, De |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR1505795A (fr) * | 1965-12-17 | 1967-12-15 | Thomae Gmbh Dr K | Procédé pour fabriquer de nouvelles 11h-pyrido[2, 3-b][1, 5]benzodiazépine-5(6h)-ones substituées en position 11 |
DE1931487C3 (de) * | 1969-06-20 | 1975-12-18 | Dr. Karl Thomae Gmbh, 7950 Biberach | In 5-Stellung substituierte 5,10-Dihydro-11H-dibenzo eckige Klammer auf b,e eckige Klammer zu eckige Klammer auf 1,4 eckige Klammer zu diazepin-11 -one und Verfahren zu ihrer Herstellung |
DE1795183B1 (de) * | 1968-08-20 | 1972-07-20 | Thomae Gmbh Dr K | 5,11-Dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-on-derivate und Arzneimittel |
DE1795176C3 (de) * | 1968-08-20 | 1974-10-24 | Dr. Karl Thomae Gmbh, 7950 Biberach | hT-substituierte 5-Aminoacetyl-5,10-dihydro-l lH-dibenzo eckige Klammer auf b,e eckige Klammer zu eckige Klammer auf 1,4 eckige Klammer zu diazepin-11one und Verfahren zu ihrer Herstellung |
DE2424811C3 (de) * | 1974-05-22 | 1981-08-20 | Dr. Karl Thomae Gmbh, 7950 Biberach | Pyrido-benzodiazepinone, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel |
US4172831A (en) * | 1974-11-26 | 1979-10-30 | Lilly Industries Limited | Thieno-benzodiazepines |
US4115568A (en) * | 1974-11-26 | 1978-09-19 | Lilly Industries Limited | Thieno[3,2-b]-[1,5]benzodiazepines |
SU629879A3 (ru) * | 1974-11-26 | 1978-10-25 | Лилли Индастриз Лимитед, (Фирма) | Способ получени тиено(1,5) бензодиазепинов или их солей |
US3951981A (en) * | 1975-02-24 | 1976-04-20 | American Cyanamid Company | Substituted benzodiazepines and method of use |
US3953430A (en) * | 1975-02-24 | 1976-04-27 | American Cyanamid Company | Substituted benzodiazepin-10-ones and method of use |
US4144235A (en) * | 1978-03-13 | 1979-03-13 | American Cyanamid Company | Thieno[3,4-b][1,5]benzoxazepin-10-ones and thieno[3,4-b][1,5]benzothiazepin-10-ones |
US4168269A (en) * | 1978-04-12 | 1979-09-18 | American Cyanamid Company | Substituted thieno-benzodiazepines |
US4263207A (en) * | 1978-08-01 | 1981-04-21 | Merck & Co., Inc. | 10,11-Dihydrodibenzo[b,f][1,4]thiazepine carboxylic acids esters and amides thereof |
-
1981
- 1981-05-05 IL IL62792A patent/IL62792A/xx not_active IP Right Cessation
- 1981-05-06 AU AU70198/81A patent/AU538031B2/en not_active Ceased
- 1981-05-06 ES ES501929A patent/ES8205802A1/es not_active Expired
- 1981-05-06 PL PL1981231003A patent/PL139428B1/pl unknown
- 1981-05-06 EP EP81103437A patent/EP0039519B1/de not_active Expired
- 1981-05-06 HU HU811799A patent/HU182712B/hu not_active IP Right Cessation
- 1981-05-06 AT AT81103437T patent/ATE7299T1/de not_active IP Right Cessation
- 1981-05-06 WO PCT/EP1981/000042 patent/WO1981003173A1/de active IP Right Grant
- 1981-05-06 IE IE997/81A patent/IE51200B1/en not_active IP Right Cessation
- 1981-05-06 DD DD81229765A patent/DD158902A5/de unknown
- 1981-05-06 YU YU1161/81A patent/YU42398B/xx unknown
- 1981-05-06 KR KR1019810001564A patent/KR850000241B1/ko active
- 1981-05-06 NZ NZ197017A patent/NZ197017A/xx unknown
- 1981-05-06 DE DE8181103437T patent/DE3163361D1/de not_active Expired
- 1981-05-06 JP JP56501690A patent/JPS6021994B2/ja not_active Expired
- 1981-05-06 GR GR64851A patent/GR82676B/el unknown
- 1981-05-06 PT PT72982A patent/PT72982B/pt unknown
- 1981-12-15 FI FI814028A patent/FI66002C/fi not_active IP Right Cessation
-
1982
- 1982-01-05 DK DK001582A patent/DK157872C/da not_active IP Right Cessation
- 1982-01-06 NO NO82820025A patent/NO156753C/no unknown
-
1990
- 1990-01-25 HK HK68/90A patent/HK6890A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
DE3163361D1 (en) | 1984-06-07 |
PT72982A (en) | 1981-06-01 |
FI66002B (fi) | 1984-04-30 |
FI814028L (fi) | 1981-12-15 |
PL231003A1 (da) | 1981-12-23 |
DK157872B (da) | 1990-02-26 |
NO820025L (no) | 1982-01-06 |
IL62792A (en) | 1985-02-28 |
DK157872C (da) | 1990-07-30 |
GR82676B (da) | 1985-02-07 |
AU7019881A (en) | 1981-11-12 |
PT72982B (fr) | 1982-10-21 |
HK6890A (en) | 1990-02-02 |
IL62792A0 (en) | 1981-07-31 |
NO156753C (no) | 1987-11-18 |
IE810997L (en) | 1981-11-07 |
YU116181A (en) | 1984-02-29 |
HU182712B (en) | 1984-03-28 |
NZ197017A (en) | 1983-09-30 |
PL139428B1 (en) | 1987-01-31 |
ES501929A0 (es) | 1982-08-16 |
KR830006300A (ko) | 1983-09-20 |
DD158902A5 (de) | 1983-02-09 |
EP0039519A1 (de) | 1981-11-11 |
DK1582A (da) | 1982-01-05 |
EP0039519B1 (de) | 1984-05-02 |
KR850000241B1 (ko) | 1985-03-12 |
ATE7299T1 (de) | 1984-05-15 |
AU538031B2 (en) | 1984-07-26 |
WO1981003173A1 (en) | 1981-11-12 |
JPS6021994B2 (ja) | 1985-05-30 |
IE51200B1 (en) | 1986-10-29 |
YU42398B (en) | 1988-08-31 |
NO156753B (no) | 1987-08-10 |
JPS57500695A (da) | 1982-04-22 |
ES8205802A1 (es) | 1982-08-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM | Patent lapsed | ||
MM | Patent lapsed |
Owner name: BYK GULDEN LOMBERG CHEMISCHE FABRIK |