FI60555C - Foerfarande foer framstaellning av terapeutiskt anvaendbara aromatiska karboxylamidderivat - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbara aromatiska karboxylamidderivat Download PDF

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Publication number
FI60555C
FI60555C FI145/74A FI14574A FI60555C FI 60555 C FI60555 C FI 60555C FI 145/74 A FI145/74 A FI 145/74A FI 14574 A FI14574 A FI 14574A FI 60555 C FI60555 C FI 60555C
Authority
FI
Finland
Prior art keywords
formula
acid
cooh
aromatic
compound
Prior art date
Application number
FI145/74A
Other languages
English (en)
Finnish (fi)
Other versions
FI60555B (fi
Inventor
Kozaburo Harita
Yukiyoshi Ajisawa
Kinji Iizuka
Yukihiko Kinoshita
Tetsuhide Kamijo
Michihiro Kobayashi
Original Assignee
Kissei Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kissei Pharmaceutical filed Critical Kissei Pharmaceutical
Publication of FI60555B publication Critical patent/FI60555B/fi
Application granted granted Critical
Publication of FI60555C publication Critical patent/FI60555C/fi

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/12—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI145/74A 1973-01-18 1974-01-18 Foerfarande foer framstaellning av terapeutiskt anvaendbara aromatiska karboxylamidderivat FI60555C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP735973 1973-01-18
JP735973A JPS5640710B2 (ru) 1973-01-18 1973-01-18

Publications (2)

Publication Number Publication Date
FI60555B FI60555B (fi) 1981-10-30
FI60555C true FI60555C (fi) 1982-02-10

Family

ID=11663750

Family Applications (1)

Application Number Title Priority Date Filing Date
FI145/74A FI60555C (fi) 1973-01-18 1974-01-18 Foerfarande foer framstaellning av terapeutiskt anvaendbara aromatiska karboxylamidderivat

Country Status (18)

Country Link
US (2) US3940422A (ru)
JP (1) JPS5640710B2 (ru)
AT (1) AT333726B (ru)
BE (1) BE809935A (ru)
BG (1) BG24538A3 (ru)
CH (2) CH613442A5 (ru)
DE (1) DE2402398C3 (ru)
DK (1) DK139676C (ru)
ES (1) ES422395A1 (ru)
FI (1) FI60555C (ru)
FR (1) FR2214476B1 (ru)
GB (1) GB1446141A (ru)
HU (1) HU168055B (ru)
IT (1) IT1054151B (ru)
NL (1) NL179370C (ru)
NO (1) NO142441C (ru)
SE (1) SE411117B (ru)
SU (1) SU520041A3 (ru)

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JPH078851B2 (ja) * 1985-07-29 1995-02-01 鐘淵化学工業株式会社 ３−フエニルチオメチルスチレン誘導体
JPH0733357B2 (ja) * 1986-09-30 1995-04-12 日本レダリ−株式会社 ケイ皮酸誘導体
JPH0692353B2 (ja) * 1987-05-26 1994-11-16 マルコ製薬株式会社 新規なアミノ安息香酸アミド誘導体およびその製造法
JP2632732B2 (ja) * 1989-11-06 1997-07-23 株式会社興人 Ｎ―（３’，４’―ジメトキシシンナモイル）アントラニル酸の製造方法
US6515009B1 (en) * 1991-09-27 2003-02-04 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
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US6306421B1 (en) 1992-09-25 2001-10-23 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US6251920B1 (en) 1993-05-13 2001-06-26 Neorx Corporation Prevention and treatment of cardiovascular pathologies
US5770609A (en) * 1993-01-28 1998-06-23 Neorx Corporation Prevention and treatment of cardiovascular pathologies
US6491938B2 (en) 1993-05-13 2002-12-10 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US6663881B2 (en) 1993-01-28 2003-12-16 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US5981568A (en) 1993-01-28 1999-11-09 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US5595722A (en) * 1993-01-28 1997-01-21 Neorx Corporation Method for identifying an agent which increases TGF-beta levels
DE69435137D1 (de) * 1993-05-13 2008-10-16 Poniard Pharmaceuticals Inc Prävention und behandlung von pathologien, die mit einer abnormalen proliferationglatter muskelzellen verbunden sind
US6197789B1 (en) 1995-06-07 2001-03-06 Neorx Corporation Prevention and treatment of cardiovascular pathologies with tamoxifen analogues
US20030083733A1 (en) * 1997-10-10 2003-05-01 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US20020091433A1 (en) * 1995-04-19 2002-07-11 Ni Ding Drug release coated stent
US5837313A (en) * 1995-04-19 1998-11-17 Schneider (Usa) Inc Drug release stent coating process
US6099562A (en) * 1996-06-13 2000-08-08 Schneider (Usa) Inc. Drug coating with topcoat
US6017919A (en) * 1996-02-06 2000-01-25 Japan Tobacco Inc. Compounds and pharmaceutical use thereof
US6019104A (en) * 1996-12-30 2000-02-01 Kissei Pharmaceutical Co., Ltd. Method for the treatment or prevention of restenosis associated with coronary intervention
DE19935219A1 (de) 1999-07-27 2001-02-01 Boehringer Ingelheim Pharma Carbonsäureamide, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Herstellung
DE10065042A1 (de) 2000-12-23 2002-06-27 Boehringer Ingelheim Pharma Carbonsäureamide, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Herstellung
DE10065043A1 (de) * 2000-12-23 2002-07-04 Boehringer Ingelheim Pharma Carbonsäureamide, diese Verbindungen enthaltene Arzneimittel, deren Verwendung und Herstellung
US6613083B2 (en) * 2001-05-02 2003-09-02 Eckhard Alt Stent device and method
EP1318141A1 (en) * 2001-12-04 2003-06-11 Dsm Nv Process for treating an aqueous medium containing phosphate, cyclohexanone and cyclohexanone oxime
MXPA04005414A (es) * 2001-12-04 2004-10-11 Dsm Ip Assets Bv Procedimiento para el tratamiento de un medio acuoso que contiene ciclohexanona oxima y ciclohexanona.
CA2468544A1 (en) * 2001-12-10 2003-06-19 Amgen Inc. Vanilloid receptor ligands
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DE10254872A1 (de) 2002-11-25 2004-06-03 Symrise Gmbh & Co. Kg Anthranilsäureamide und deren Derivate als kosmetische und pharmazeutische Wirkstoffe
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CN102574843B (zh) 2009-10-22 2015-06-17 法博太科制药有限公司 抗纤维化剂的稠环类似物
DE102009046115A1 (de) * 2009-10-28 2011-09-08 Bayer Schering Pharma Aktiengesellschaft Substituierte 3-Phenylpropansäuren und ihre Verwendung
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US10188754B2 (en) 2013-05-16 2019-01-29 The Johns Hopkins University Compositions and methods for chemical exchange saturation transfer (CEST) based magnetic resonance imaging (MRI)
CN104693063A (zh) * 2015-03-18 2015-06-10 中国药科大学制药有限公司 一种曲尼司特的合成方法
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Also Published As

Publication number Publication date
NO142441C (no) 1980-08-20
AU6461374A (en) 1975-07-17
FR2214476B1 (ru) 1977-08-12
IT1054151B (it) 1981-11-10
FR2214476A1 (ru) 1974-08-19
NL179370B (nl) 1986-04-01
FI60555B (fi) 1981-10-30
DK139676C (da) 1979-09-10
DK139676B (da) 1979-03-26
ATA44374A (de) 1976-04-15
GB1446141A (en) 1976-08-18
US3940422A (en) 1976-02-24
DE2402398C3 (de) 1981-07-23
CH613442A5 (ru) 1979-09-28
SE411117B (sv) 1979-12-03
ES422395A1 (es) 1976-08-01
DE2402398B2 (de) 1980-10-09
DE2402398A1 (de) 1974-08-08
BE809935A (fr) 1974-05-16
JPS5640710B2 (ru) 1981-09-22
NO142441B (no) 1980-05-12
NO740137L (no) 1974-07-19
BG24538A3 (en) 1978-03-10
USRE32944E (en) 1989-06-06
NL179370C (nl) 1986-09-01
SU520041A3 (ru) 1976-06-30
HU168055B (ru) 1976-02-28
AT333726B (de) 1976-12-10
JPS4993335A (ru) 1974-09-05
NL7400754A (ru) 1974-07-22
CH615152A5 (en) 1980-01-15

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