FI114799B - Uusi 7-substituoitu oksasteroidiyhdiste - Google Patents

Uusi 7-substituoitu oksasteroidiyhdiste Download PDF

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Publication number
FI114799B
FI114799B FI951505A FI951505A FI114799B FI 114799 B FI114799 B FI 114799B FI 951505 A FI951505 A FI 951505A FI 951505 A FI951505 A FI 951505A FI 114799 B FI114799 B FI 114799B
Authority
FI
Finland
Prior art keywords
group
compound
oxa
formula
homo
Prior art date
Application number
FI951505A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI951505A0 (fi
FI951505A (fi
Inventor
Naoyuki Koizumi
Shigehiro Takegawa
Shigeki Iwashita
Tomoko Kawachi
Fumiko Inoue
Seijiro Honma
Hiroo Takahashi
Mamoru Mieda
Kaoru Ueda
Kenyu Shibata
Original Assignee
Teikoku Hormone Mfg Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teikoku Hormone Mfg Co Ltd filed Critical Teikoku Hormone Mfg Co Ltd
Publication of FI951505A0 publication Critical patent/FI951505A0/fi
Publication of FI951505A publication Critical patent/FI951505A/fi
Application granted granted Critical
Publication of FI114799B publication Critical patent/FI114799B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J73/00Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J73/00Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J73/00Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/003Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by oxygen as hetero atom

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI951505A 1992-09-30 1995-03-29 Uusi 7-substituoitu oksasteroidiyhdiste FI114799B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP28361692 1992-09-30
JP28361692 1992-09-30
JP9301390 1993-09-29
PCT/JP1993/001390 WO1994007908A1 (en) 1992-09-30 1993-09-29 Novel 7-substituted oxa- or azasteroid compound

Publications (3)

Publication Number Publication Date
FI951505A0 FI951505A0 (fi) 1995-03-29
FI951505A FI951505A (fi) 1995-05-26
FI114799B true FI114799B (fi) 2004-12-31

Family

ID=17667815

Family Applications (1)

Application Number Title Priority Date Filing Date
FI951505A FI114799B (fi) 1992-09-30 1995-03-29 Uusi 7-substituoitu oksasteroidiyhdiste

Country Status (18)

Country Link
US (1) US5539127A (da)
EP (1) EP0663402B1 (da)
JP (1) JP3293629B2 (da)
KR (1) KR100231638B1 (da)
AT (1) ATE179179T1 (da)
AU (1) AU665455B2 (da)
CA (1) CA2145643A1 (da)
DE (1) DE69324595T2 (da)
DK (1) DK0663402T3 (da)
ES (1) ES2130284T3 (da)
FI (1) FI114799B (da)
GR (1) GR3030245T3 (da)
HU (1) HU221191B1 (da)
NO (1) NO306066B1 (da)
NZ (1) NZ256130A (da)
PL (1) PL176114B1 (da)
SG (1) SG48172A1 (da)
WO (1) WO1994007908A1 (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5245275A (en) * 1989-09-25 1993-09-14 General Electric Company Electronic watthour meter
DE19610645A1 (de) 1996-03-06 1997-09-11 Schering Ag Kombination von Dehydroepiandrosteron und Aromatasehemmern und Verwendung dieser Kombination zur Herstellung eines Arzeimittels zur Behandlung eines relativen und absoluten Androgenmangels beim Mann
JP5409393B2 (ja) * 2007-03-01 2014-02-05 ビーエーエスエフ ソシエタス・ヨーロピア エチレンアミンの製造方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4116978A (en) * 1977-07-20 1978-09-26 E. R. Squibb & Sons, Inc. D-homo oxasteroids
US4235893A (en) * 1978-05-08 1980-11-25 Brodie Angela M Ester derivatives of 4-hydroxy-4-androstene-3,17-dione and a method for inhibiting estrogen biosynthesis
DE3322285A1 (de) * 1983-06-18 1984-12-20 Schering AG, 1000 Berlin und 4709 Bergkamen 1-alkyl-androsta-1,4-dien-3,17-dione, verfahren zu deren herstellung und diese enthaltende pharmazeutische praeparate
GB8503940D0 (en) * 1985-02-15 1985-03-20 Erba Farmitalia 4-substituted androstendione derivatives
DE3622841C2 (de) * 1985-07-09 2001-01-25 Pharmacia & Upjohn Spa Substituierte Androsta-1,4-dien-3,17-dione und Verfahren zu deren Herstellung
GB8517360D0 (en) * 1985-07-09 1985-08-14 Erba Farmitalia Substituted androsta-1,4-diene-3,17-diones
US5227375A (en) * 1990-02-08 1993-07-13 Endorecherche, Inc. Aromatase inhibitors
US5219879A (en) * 1990-03-05 1993-06-15 Du Pont Merck Pharmaceutical Company Heterocyclic steroid compounds
KR0180008B1 (ko) * 1991-03-28 1999-04-01 야마구찌 다까시 신규 옥사-또는 아자스테로이드 유체
JPH05148294A (ja) * 1991-11-27 1993-06-15 Teikoku Hormone Mfg Co Ltd 3,5−ジエンステロイド誘導体

Also Published As

Publication number Publication date
FI951505A0 (fi) 1995-03-29
SG48172A1 (en) 1998-04-17
HU9500929D0 (en) 1995-05-29
PL176114B1 (pl) 1999-04-30
EP0663402A1 (en) 1995-07-19
NO951211L (no) 1995-05-30
NO306066B1 (no) 1999-09-13
DE69324595T2 (de) 1999-08-19
NO951211D0 (no) 1995-03-29
EP0663402A4 (en) 1996-06-12
HUT71519A (en) 1995-12-28
DE69324595D1 (de) 1999-05-27
PL308228A1 (en) 1995-07-24
KR100231638B1 (ko) 1999-12-01
EP0663402B1 (en) 1999-04-21
US5539127A (en) 1996-07-23
WO1994007908A1 (en) 1994-04-14
DK0663402T3 (da) 1999-10-25
FI951505A (fi) 1995-05-26
AU665455B2 (en) 1996-01-04
KR950703575A (ko) 1995-09-20
GR3030245T3 (en) 1999-08-31
CA2145643A1 (en) 1994-04-14
JP3293629B2 (ja) 2002-06-17
HU221191B1 (en) 2002-08-28
NZ256130A (en) 1996-05-28
ATE179179T1 (de) 1999-05-15
ES2130284T3 (es) 1999-07-01
AU4834293A (en) 1994-04-26

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