FI114470B - Uusia allergisten sairauksien hoidossa käyttökelpoisia substituoituja piperidiinejä - Google Patents

Uusia allergisten sairauksien hoidossa käyttökelpoisia substituoituja piperidiinejä Download PDF

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Publication number
FI114470B
FI114470B FI970771A FI970771A FI114470B FI 114470 B FI114470 B FI 114470B FI 970771 A FI970771 A FI 970771A FI 970771 A FI970771 A FI 970771A FI 114470 B FI114470 B FI 114470B
Authority
FI
Finland
Prior art keywords
ethyl
carbonyl
pyrrolidine
benzoimidazole
piperidin
Prior art date
Application number
FI970771A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI970771A (fi
FI970771A0 (fi
Inventor
Timothy Paul Burkholder
Elizabeth Mary Kudlacz
Larry Don Bratton
George Daniel Maynard
John Michael Kane
Braulio Santiago
Original Assignee
Merrell Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Pharma Inc filed Critical Merrell Pharma Inc
Publication of FI970771A publication Critical patent/FI970771A/fi
Publication of FI970771A0 publication Critical patent/FI970771A0/fi
Application granted granted Critical
Publication of FI114470B publication Critical patent/FI114470B/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
FI970771A 1994-08-25 1997-02-24 Uusia allergisten sairauksien hoidossa käyttökelpoisia substituoituja piperidiinejä FI114470B (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US29596094A 1994-08-25 1994-08-25
US29596094 1994-08-25
US50191495A 1995-07-13 1995-07-13
US50191495 1995-07-13
PCT/US1995/010640 WO1996006094A1 (en) 1994-08-25 1995-08-17 Novel substituted piperidines useful for the treatment of allergic diseases
US9510640 1995-08-17

Publications (3)

Publication Number Publication Date
FI970771A FI970771A (fi) 1997-02-24
FI970771A0 FI970771A0 (fi) 1997-02-24
FI114470B true FI114470B (fi) 2004-10-29

Family

ID=26969426

Family Applications (1)

Application Number Title Priority Date Filing Date
FI970771A FI114470B (fi) 1994-08-25 1997-02-24 Uusia allergisten sairauksien hoidossa käyttökelpoisia substituoituja piperidiinejä

Country Status (20)

Country Link
US (1) US6329392B1 (hu)
EP (1) EP0777666B1 (hu)
JP (1) JPH10504580A (hu)
KR (1) KR100362620B1 (hu)
CN (1) CN1067385C (hu)
AT (1) ATE177095T1 (hu)
AU (1) AU693936B2 (hu)
CA (1) CA2198084C (hu)
DE (1) DE69508093T2 (hu)
DK (1) DK0777666T3 (hu)
ES (1) ES2132709T3 (hu)
FI (1) FI114470B (hu)
GR (1) GR3030253T3 (hu)
HU (1) HU221434B (hu)
IL (1) IL115040A (hu)
MX (1) MX9701305A (hu)
NO (1) NO313237B1 (hu)
NZ (1) NZ292683A (hu)
TW (1) TW430663B (hu)
WO (1) WO1996006094A1 (hu)

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Also Published As

Publication number Publication date
TW430663B (en) 2001-04-21
US6329392B1 (en) 2001-12-11
CA2198084A1 (en) 1996-02-29
IL115040A0 (en) 1995-12-08
AU693936B2 (en) 1998-07-09
EP0777666B1 (en) 1999-03-03
WO1996006094A1 (en) 1996-02-29
DE69508093D1 (de) 1999-04-08
CN1067385C (zh) 2001-06-20
JPH10504580A (ja) 1998-05-06
KR100362620B1 (ko) 2003-02-14
EP0777666A1 (en) 1997-06-11
NZ292683A (en) 1998-07-28
FI970771A (fi) 1997-02-24
MX9701305A (es) 1998-05-31
IL115040A (en) 2000-02-29
NO970831D0 (no) 1997-02-24
DK0777666T3 (da) 1999-09-27
GR3030253T3 (en) 1999-08-31
HUT76644A (en) 1997-10-28
ES2132709T3 (es) 1999-08-16
KR970705556A (ko) 1997-10-09
ATE177095T1 (de) 1999-03-15
AU3492895A (en) 1996-03-14
FI970771A0 (fi) 1997-02-24
DE69508093T2 (de) 1999-07-15
HU221434B (en) 2002-10-28
NO970831L (no) 1997-04-18
NO313237B1 (no) 2002-09-02
CA2198084C (en) 2000-03-28
CN1158612A (zh) 1997-09-03

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