DK0777666T3 - Substituerede piperidiner anvendelige ved behandling af allergiske sygdomme - Google Patents

Substituerede piperidiner anvendelige ved behandling af allergiske sygdomme

Info

Publication number
DK0777666T3
DK0777666T3 DK95931551T DK95931551T DK0777666T3 DK 0777666 T3 DK0777666 T3 DK 0777666T3 DK 95931551 T DK95931551 T DK 95931551T DK 95931551 T DK95931551 T DK 95931551T DK 0777666 T3 DK0777666 T3 DK 0777666T3
Authority
DK
Denmark
Prior art keywords
treatment
allergic diseases
useful
substituted piperidines
piperidines useful
Prior art date
Application number
DK95931551T
Other languages
English (en)
Inventor
John M Kane
Timothy P Burkholder
Elizabeth M Kudlacz
Larry D Bratton
George D Maynard
Braulio Santiago
Original Assignee
Merrell Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Pharma Inc filed Critical Merrell Pharma Inc
Application granted granted Critical
Publication of DK0777666T3 publication Critical patent/DK0777666T3/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
DK95931551T 1994-08-25 1995-08-17 Substituerede piperidiner anvendelige ved behandling af allergiske sygdomme DK0777666T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29596094A 1994-08-25 1994-08-25
US50191495A 1995-07-13 1995-07-13
PCT/US1995/010640 WO1996006094A1 (en) 1994-08-25 1995-08-17 Novel substituted piperidines useful for the treatment of allergic diseases

Publications (1)

Publication Number Publication Date
DK0777666T3 true DK0777666T3 (da) 1999-09-27

Family

ID=26969426

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95931551T DK0777666T3 (da) 1994-08-25 1995-08-17 Substituerede piperidiner anvendelige ved behandling af allergiske sygdomme

Country Status (20)

Country Link
US (1) US6329392B1 (da)
EP (1) EP0777666B1 (da)
JP (1) JPH10504580A (da)
KR (1) KR100362620B1 (da)
CN (1) CN1067385C (da)
AT (1) ATE177095T1 (da)
AU (1) AU693936B2 (da)
CA (1) CA2198084C (da)
DE (1) DE69508093T2 (da)
DK (1) DK0777666T3 (da)
ES (1) ES2132709T3 (da)
FI (1) FI114470B (da)
GR (1) GR3030253T3 (da)
HU (1) HU221434B (da)
IL (1) IL115040A (da)
MX (1) MX9701305A (da)
NO (1) NO313237B1 (da)
NZ (1) NZ292683A (da)
TW (1) TW430663B (da)
WO (1) WO1996006094A1 (da)

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Also Published As

Publication number Publication date
NO970831D0 (no) 1997-02-24
TW430663B (en) 2001-04-21
AU693936B2 (en) 1998-07-09
EP0777666B1 (en) 1999-03-03
CN1158612A (zh) 1997-09-03
US6329392B1 (en) 2001-12-11
IL115040A (en) 2000-02-29
CA2198084C (en) 2000-03-28
CA2198084A1 (en) 1996-02-29
HUT76644A (en) 1997-10-28
NZ292683A (en) 1998-07-28
DE69508093D1 (de) 1999-04-08
DE69508093T2 (de) 1999-07-15
FI114470B (fi) 2004-10-29
IL115040A0 (en) 1995-12-08
GR3030253T3 (en) 1999-08-31
NO313237B1 (no) 2002-09-02
FI970771A (fi) 1997-02-24
AU3492895A (en) 1996-03-14
KR970705556A (ko) 1997-10-09
FI970771A0 (fi) 1997-02-24
JPH10504580A (ja) 1998-05-06
WO1996006094A1 (en) 1996-02-29
CN1067385C (zh) 2001-06-20
MX9701305A (es) 1998-05-31
KR100362620B1 (ko) 2003-02-14
NO970831L (no) 1997-04-18
ATE177095T1 (de) 1999-03-15
ES2132709T3 (es) 1999-08-16
EP0777666A1 (en) 1997-06-11
HU221434B (en) 2002-10-28

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