FI113263B - Menetelmä 6-fluori-2-halogeenikinoliinin valmistamiseksi - Google Patents

Menetelmä 6-fluori-2-halogeenikinoliinin valmistamiseksi Download PDF

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Publication number
FI113263B
FI113263B FI954750A FI954750A FI113263B FI 113263 B FI113263 B FI 113263B FI 954750 A FI954750 A FI 954750A FI 954750 A FI954750 A FI 954750A FI 113263 B FI113263 B FI 113263B
Authority
FI
Finland
Prior art keywords
radical
alkyl
hal
general formula
difluoro
Prior art date
Application number
FI954750A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI954750A (fi
FI954750A0 (fi
Inventor
Herve Garcia
Roland Jacquot
Patrick Leon
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of FI954750A publication Critical patent/FI954750A/fi
Publication of FI954750A0 publication Critical patent/FI954750A0/fi
Application granted granted Critical
Publication of FI113263B publication Critical patent/FI113263B/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D251/00Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/12Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D251/26Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
    • C07D251/40Nitrogen atoms
    • C07D251/54Three nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI954750A 1993-04-08 1995-10-05 Menetelmä 6-fluori-2-halogeenikinoliinin valmistamiseksi FI113263B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR9304163 1993-04-08
FR9304163A FR2703681B1 (fr) 1993-04-08 1993-04-08 Procede de preparation de fluoro-6-halogeno-2 quinoleine
PCT/FR1994/000391 WO1994024113A1 (fr) 1993-04-08 1994-04-07 Procede de preparation de fluoro-6 halogeno-2 quinoleine
FR9400391 1994-04-07

Publications (3)

Publication Number Publication Date
FI954750A FI954750A (fi) 1995-10-05
FI954750A0 FI954750A0 (fi) 1995-10-05
FI113263B true FI113263B (fi) 2004-03-31

Family

ID=9445879

Family Applications (1)

Application Number Title Priority Date Filing Date
FI954750A FI113263B (fi) 1993-04-08 1995-10-05 Menetelmä 6-fluori-2-halogeenikinoliinin valmistamiseksi

Country Status (21)

Country Link
US (1) US5624933A (ko)
EP (1) EP0693060B1 (ko)
JP (1) JP3666753B2 (ko)
KR (1) KR100330141B1 (ko)
AT (1) ATE164155T1 (ko)
AU (1) AU680493B2 (ko)
CA (1) CA2158746C (ko)
CZ (1) CZ283705B6 (ko)
DE (1) DE69409101T2 (ko)
DK (1) DK0693060T3 (ko)
ES (1) ES2114189T3 (ko)
FI (1) FI113263B (ko)
FR (1) FR2703681B1 (ko)
GR (1) GR3026401T3 (ko)
HU (1) HU221861B1 (ko)
IL (1) IL109255A (ko)
NO (1) NO305752B1 (ko)
NZ (1) NZ265072A (ko)
SK (1) SK281139B6 (ko)
TW (1) TW261612B (ko)
WO (1) WO1994024113A1 (ko)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7510170B2 (en) 2006-11-09 2009-03-31 Guan Hong Enterprise Co., Ltd. Humidifying fan

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1458205A (en) * 1973-04-13 1976-12-08 Pfizer Fused pyrimidin-4- 3h-ones as antiallergy agents
US4190659A (en) * 1973-08-27 1980-02-26 Sandoz, Inc. Pharmaceutical preparation and use of 4-hydroxy-2-quinolinone-3-carboxylic acid esters
US4710507A (en) * 1983-12-22 1987-12-01 Pfizer Inc. Quinolone inotropic agents
DK111387A (da) * 1986-03-05 1987-09-06 Otsuka Pharma Co Ltd Carbostyrilderivater og salte deraf, laegemiddel indeholdende saadanne derivater samt fremgangsmaade til fremstilling af derivaterne
DE3713672A1 (de) * 1987-04-24 1988-11-17 Bayer Ag Verfahren zur herstellung von parenteral verabreichbaren chinoloncarbonsaeuren
AU623474B2 (en) * 1989-01-16 1992-05-14 Laboratoire Roger Bellon New benzo(1,8)naphthyridine derivatives, their preparation and compositions containing them
NZ232092A (en) * 1989-01-16 1992-05-26 Bellon Labor Sa Roger 8-halo-7-fluoro-4-oxo-1,4-dihydro-benzo(b)(1,8) naphthyridine-3-carboxylic acid esters and preparation thereof
NZ232090A (en) * 1989-01-16 1990-12-21 Bellon Labor Sa Roger Halogen-containing 1-substituted-4-oxo-1,4-dihydro-benzo(b)(1,8)naphthyridine-3-carboxylic acid derivatives, preparation and pharmaceutical compositions thereof
US4948894A (en) * 1989-02-21 1990-08-14 American Cyanamid Company 8-fluoro and 7, 8, 10-trifluoro-9-(substituted)-6-oxo-6H-benzo-(C)quinolizine-5-carboxylic acids
RO108347B1 (ro) * 1989-10-30 1994-04-28 Bellon Labor Sa Roger DERIVATI DE BENZO-(b)-NAFTIRIDIN-1,8 SI PROCEDEU DE PREPARARE A ACESTORA
FR2682384B1 (fr) * 1991-10-10 1995-04-07 Bellon Laboratoires Procede de preparation de benzo (b) naphtyridines.
FR2682378B1 (fr) * 1991-10-10 1995-04-07 Bellon Laboratoires Nouveaux derives de l'acide fluoroquinoleine carboxylique-3 et leur preparation.

Also Published As

Publication number Publication date
CZ283705B6 (cs) 1998-06-17
ES2114189T3 (es) 1998-05-16
JPH08508747A (ja) 1996-09-17
IL109255A (en) 2000-01-31
EP0693060A1 (fr) 1996-01-24
FI954750A (fi) 1995-10-05
FR2703681A1 (fr) 1994-10-14
GR3026401T3 (en) 1998-06-30
WO1994024113A1 (fr) 1994-10-27
HU221861B1 (hu) 2003-02-28
SK125695A3 (en) 1996-06-05
TW261612B (ko) 1995-11-01
NO305752B1 (no) 1999-07-19
US5624933A (en) 1997-04-29
FR2703681B1 (fr) 1995-05-12
FI954750A0 (fi) 1995-10-05
IL109255A0 (en) 1994-07-31
NO953914L (no) 1995-10-02
NZ265072A (en) 1997-08-22
DK0693060T3 (da) 1998-10-19
SK281139B6 (sk) 2000-12-11
ATE164155T1 (de) 1998-04-15
AU6540894A (en) 1994-11-08
HU9502934D0 (en) 1995-12-28
JP3666753B2 (ja) 2005-06-29
KR960701854A (ko) 1996-03-28
CA2158746C (fr) 2006-08-29
NO953914D0 (no) 1995-10-02
CA2158746A1 (fr) 1994-10-27
CZ260095A3 (en) 1996-01-17
EP0693060B1 (fr) 1998-03-18
DE69409101D1 (de) 1998-04-23
HUT73560A (en) 1996-08-28
KR100330141B1 (ko) 2002-09-27
DE69409101T2 (de) 1998-07-23
AU680493B2 (en) 1997-07-31

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MA Patent expired