FI113174B - Menetelmä ja välituote 5-amino-8-metyyli-7-pyrrolidinyylikinoliini-3-karboksyylihappojohdannaisten valmistamiseksi - Google Patents

Menetelmä ja välituote 5-amino-8-metyyli-7-pyrrolidinyylikinoliini-3-karboksyylihappojohdannaisten valmistamiseksi Download PDF

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Publication number
FI113174B
FI113174B FI942976A FI942976A FI113174B FI 113174 B FI113174 B FI 113174B FI 942976 A FI942976 A FI 942976A FI 942976 A FI942976 A FI 942976A FI 113174 B FI113174 B FI 113174B
Authority
FI
Finland
Prior art keywords
compound
methyl
amino
carboxylic acid
group
Prior art date
Application number
FI942976A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI942976A0 (fi
FI942976A (fi
Inventor
Yasuo Ito
Hideo Kato
Singo Yasuda
Noriyaki Kado
Toshihiko Yoshida
Yoichi Yamamoto
Original Assignee
Hokuriku Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hokuriku Pharmaceutical filed Critical Hokuriku Pharmaceutical
Publication of FI942976A0 publication Critical patent/FI942976A0/fi
Publication of FI942976A publication Critical patent/FI942976A/fi
Application granted granted Critical
Publication of FI113174B publication Critical patent/FI113174B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Epoxy Resins (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
FI942976A 1993-08-27 1994-06-21 Menetelmä ja välituote 5-amino-8-metyyli-7-pyrrolidinyylikinoliini-3-karboksyylihappojohdannaisten valmistamiseksi FI113174B (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
JP23431093 1993-08-27
JP23431093 1993-08-27
JP28627293 1993-10-22
JP28627293 1993-10-22
JP7631894 1994-03-24
JP7631894 1994-03-24

Publications (3)

Publication Number Publication Date
FI942976A0 FI942976A0 (fi) 1994-06-21
FI942976A FI942976A (fi) 1995-02-28
FI113174B true FI113174B (fi) 2004-03-15

Family

ID=27302121

Family Applications (1)

Application Number Title Priority Date Filing Date
FI942976A FI113174B (fi) 1993-08-27 1994-06-21 Menetelmä ja välituote 5-amino-8-metyyli-7-pyrrolidinyylikinoliini-3-karboksyylihappojohdannaisten valmistamiseksi

Country Status (23)

Country Link
US (1) US5547962A (de)
EP (1) EP0641793B1 (de)
JP (1) JP2673937B2 (de)
KR (1) KR100218807B1 (de)
CN (1) CN1048242C (de)
AT (1) ATE144508T1 (de)
AU (1) AU676729B2 (de)
CA (1) CA2126118C (de)
CZ (1) CZ286524B6 (de)
DE (1) DE69400791T2 (de)
DK (1) DK0641793T3 (de)
ES (1) ES2096413T3 (de)
FI (1) FI113174B (de)
GR (1) GR3021715T3 (de)
HU (1) HU221952B1 (de)
IL (1) IL110060A (de)
MY (1) MY111702A (de)
NO (1) NO305515B1 (de)
NZ (1) NZ260851A (de)
PL (1) PL175870B1 (de)
SG (1) SG52147A1 (de)
TW (1) TW252107B (de)
UA (1) UA39859C2 (de)

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US6121285A (en) 1995-11-22 2000-09-19 Daiichi Pharmaceutical Co., Ltd. Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
HUP0100051A3 (en) 1997-09-15 2002-08-28 Procter & Gamble Antimicrobial quinolones, their compositions and uses
US6387928B1 (en) 1997-09-15 2002-05-14 The Procter & Gamble Co. Antimicrobial quinolones, their compositions and uses
ES2203254T3 (es) * 1998-11-18 2004-04-01 Asahi Glass Company Ltd. Derivados de acido aminoacrilico y procedimiento de produccion correspondiente.
EP2275141A1 (de) 1999-03-17 2011-01-19 Daiichi Pharmaceutical Co., Ltd. Geschmacksmaskierte pharmazeutische Zusammensetzungen
MXPA02007667A (es) 2000-02-09 2003-04-14 Daiichi Seiyaku Co Agentes antibacterianos antiacidos-resistentes que contienen acidos piridoncarboxilicos como el ingrediente activo.
RU2002122758A (ru) * 2000-02-25 2004-01-10 Дайити Фармасьютикал Ко., Лтд. (JP) Способ получения хинолонкарбоновых кислот и их промежуточные соединения
US6825353B2 (en) 2000-02-25 2004-11-30 Daiichi Pharmaceutical Co., Ltd. Process for producing quinolonecarboxylic acids and intermediates thereof
KR20010044286A (ko) * 2001-02-01 2001-06-05 남근수 알킬-3-(2,6-디할로겐-5-플루오로)-옥소-3-피리딘프로피오네이트의 제조방법
EP1882685A4 (de) 2005-05-20 2010-10-27 Daiichi Sankyo Co Ltd Verfahren zur herstellung einer asymmetrischen, tetrasubstituierten kohlenstoffhaltigen verbindung
US7842818B2 (en) 2005-09-28 2010-11-30 Daiichi Sankyo Company, Limited Process for preparation of tetrasubstituted 5-azaspiro[2.4]- heptane derivatives and optically active intermediates thereof
KR101084521B1 (ko) * 2006-03-28 2011-11-18 워너 칠콧 컴퍼니 엘엘씨 퀴놀론 중간체를 제조하기 위한 커플링 방법
MX2008012328A (es) * 2006-03-28 2008-10-09 Procter & Gamble Sales de malato, y polimorfos de acido (3s,5s)-7-[3-amino-5-metil- piperidinil]-1-ciclopropil-1,4-dihidro-8-metoxi-4-oxo-3-quinolinc arboxilico.
CA2647457C (en) * 2006-03-28 2011-05-24 The Procter & Gamble Company A hydride reduction process for preparing quinolone intermediates
TWI362386B (en) * 2007-03-30 2012-04-21 Daiichi Sankyo Co Ltd A production method for the qunolon-carboxylic acid derivative
FR2928150A1 (fr) * 2008-02-29 2009-09-04 Vetoquinol Sa Sa Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens

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JPH0635457B2 (ja) * 1985-06-28 1994-05-11 杏林製薬株式会社 ピリドンカルボン酸誘導体およびその製造方法
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Also Published As

Publication number Publication date
HU221952B1 (hu) 2003-03-28
NZ260851A (en) 1996-03-26
UA39859C2 (uk) 2001-07-16
CZ286524B6 (cs) 2000-05-17
GR3021715T3 (en) 1997-02-28
US5547962A (en) 1996-08-20
NO942309D0 (no) 1994-06-17
DE69400791T2 (de) 1997-03-06
CA2126118C (en) 2001-02-06
IL110060A (en) 1999-10-28
CN1117491A (zh) 1996-02-28
MY111702A (en) 2000-11-30
DK0641793T3 (da) 1996-11-25
EP0641793A1 (de) 1995-03-08
CZ157494A3 (en) 1995-10-18
ATE144508T1 (de) 1996-11-15
HU9401954D0 (en) 1994-09-28
FI942976A0 (fi) 1994-06-21
ES2096413T3 (es) 1997-03-01
KR950005823A (ko) 1995-03-20
AU676729B2 (en) 1997-03-20
PL304063A1 (en) 1995-03-06
DE69400791D1 (de) 1996-11-28
NO942309L (no) 1995-02-28
SG52147A1 (en) 1998-09-28
CA2126118A1 (en) 1995-02-28
KR100218807B1 (ko) 1999-09-01
NO305515B1 (no) 1999-06-14
CN1048242C (zh) 2000-01-12
EP0641793B1 (de) 1996-10-23
TW252107B (de) 1995-07-21
FI942976A (fi) 1995-02-28
JPH07309864A (ja) 1995-11-28
IL110060A0 (en) 1994-10-07
JP2673937B2 (ja) 1997-11-05
PL175870B1 (pl) 1999-02-26
HUT67259A (en) 1995-03-28
AU6487094A (en) 1995-03-09

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