FI107153B - Menetelmä ja välituote tietyille bis-atsa-bisyklisille tuskaisuutta poistaville aineille - Google Patents

Menetelmä ja välituote tietyille bis-atsa-bisyklisille tuskaisuutta poistaville aineille Download PDF

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Publication number
FI107153B
FI107153B FI933754A FI933754A FI107153B FI 107153 B FI107153 B FI 107153B FI 933754 A FI933754 A FI 933754A FI 933754 A FI933754 A FI 933754A FI 107153 B FI107153 B FI 107153B
Authority
FI
Finland
Prior art keywords
formula
compound
alkyl
process according
phthalimido
Prior art date
Application number
FI933754A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI933754A0 (fi
FI933754A (fi
Inventor
Frank John Urban
Charles William Murtiashaw
Dennis Michael Godek
Brian Clement Vanderplas
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI933754A0 publication Critical patent/FI933754A0/fi
Publication of FI933754A publication Critical patent/FI933754A/fi
Application granted granted Critical
Publication of FI107153B publication Critical patent/FI107153B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Reinforced Plastic Materials (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI933754A 1991-02-27 1993-08-26 Menetelmä ja välituote tietyille bis-atsa-bisyklisille tuskaisuutta poistaville aineille FI107153B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US07/661,730 US5185449A (en) 1991-02-27 1991-02-27 Process and intermediate for certain bis-aza-bicyclic anxiolytic agents
US66173091 1991-02-27
PCT/US1991/008400 WO1992015575A1 (fr) 1991-02-27 1991-11-19 Procede et produit intermediaire pour la preparation de certains agents anxiolytiques bis-aza-bicycliques
US9108400 1991-11-19

Publications (3)

Publication Number Publication Date
FI933754A0 FI933754A0 (fi) 1993-08-26
FI933754A FI933754A (fi) 1993-08-26
FI107153B true FI107153B (fi) 2001-06-15

Family

ID=24654869

Family Applications (1)

Application Number Title Priority Date Filing Date
FI933754A FI107153B (fi) 1991-02-27 1993-08-26 Menetelmä ja välituote tietyille bis-atsa-bisyklisille tuskaisuutta poistaville aineille

Country Status (23)

Country Link
US (1) US5185449A (fr)
EP (1) EP0586376B1 (fr)
JP (1) JPH0784467B2 (fr)
KR (1) KR100189044B1 (fr)
AT (1) ATE153662T1 (fr)
AU (1) AU647562B2 (fr)
CA (1) CA2101433C (fr)
DE (1) DE69126326T2 (fr)
DK (1) DK0586376T3 (fr)
ES (1) ES2101831T3 (fr)
FI (1) FI107153B (fr)
GR (1) GR3024125T3 (fr)
HU (2) HUT67440A (fr)
IE (1) IE920600A1 (fr)
IL (1) IL101022A (fr)
MX (1) MX9200802A (fr)
MY (1) MY110167A (fr)
NO (1) NO302947B1 (fr)
NZ (1) NZ241738A (fr)
PT (1) PT100161B (fr)
TW (1) TW268949B (fr)
WO (1) WO1992015575A1 (fr)
ZA (1) ZA921406B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69218414T2 (de) * 1991-02-27 1998-01-22 Pfizer Verfahren zur herstellung von trans-piperidin-2,5-dicarboxylaten
ES2166830T3 (es) * 1994-09-30 2002-05-01 Pfizer Derivados 2,7-sustituidos de octahidro-1h-pirido(1,2-a)pirazina.
WO1996010570A1 (fr) * 1994-09-30 1996-04-11 Pfizer Inc. PERHYDRO-1H-PYRIDO[1,2-a] PYRAZINES DISUBSTITUEES EN 2,7 A ACTION NEUROLEPTIQUE
US6670476B2 (en) 2000-11-29 2003-12-30 Pfizer Inc. Resolution of trans-7-(hydroxy-methyl)octa-hydro-2H-pyrido[1,2-a]pyrazine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3388128A (en) * 1965-09-03 1968-06-11 Allan R. Day Substituted 1, 4-diazabicyclo [4. 4. 9] decanes
WO1990008148A1 (fr) * 1989-01-23 1990-07-26 Pfizer Inc. Agents anxiolytiques bis-aza-bicycliques
DE69218414T2 (de) * 1991-02-27 1998-01-22 Pfizer Verfahren zur herstellung von trans-piperidin-2,5-dicarboxylaten

Also Published As

Publication number Publication date
EP0586376B1 (fr) 1997-05-28
ZA921406B (en) 1993-08-26
AU647562B2 (en) 1994-03-24
HU9302428D0 (en) 1993-11-29
PT100161B (pt) 1999-09-30
ES2101831T3 (es) 1997-07-16
DK0586376T3 (da) 1997-10-27
KR100189044B1 (ko) 1999-06-01
DE69126326D1 (de) 1997-07-03
HUT67440A (en) 1995-04-28
HU223138B1 (hu) 2004-03-29
JPH0784467B2 (ja) 1995-09-13
NO933048L (no) 1993-08-26
PT100161A (pt) 1993-05-31
IL101022A0 (en) 1992-11-15
AU9066691A (en) 1992-10-06
US5185449A (en) 1993-02-09
IE920600A1 (en) 1992-09-09
WO1992015575A1 (fr) 1992-09-17
CA2101433A1 (fr) 1992-08-28
FI933754A0 (fi) 1993-08-26
NO933048D0 (no) 1993-08-26
NO302947B1 (no) 1998-05-11
JPH06501021A (ja) 1994-01-27
CA2101433C (fr) 1999-07-27
MX9200802A (es) 1992-08-01
DE69126326T2 (de) 1997-09-04
NZ241738A (en) 1993-05-26
TW268949B (fr) 1996-01-21
IL101022A (en) 1996-06-18
FI933754A (fi) 1993-08-26
EP0586376A1 (fr) 1994-03-16
GR3024125T3 (en) 1997-10-31
ATE153662T1 (de) 1997-06-15
MY110167A (en) 1998-02-28

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MA Patent expired