MX9200802A - Procedimientos mejorado e intermediario para ciertos agentes bis-aza-bi-ciclicos anxioliticos. - Google Patents

Procedimientos mejorado e intermediario para ciertos agentes bis-aza-bi-ciclicos anxioliticos.

Info

Publication number
MX9200802A
MX9200802A MX9200802A MX9200802A MX9200802A MX 9200802 A MX9200802 A MX 9200802A MX 9200802 A MX9200802 A MX 9200802A MX 9200802 A MX9200802 A MX 9200802A MX 9200802 A MX9200802 A MX 9200802A
Authority
MX
Mexico
Prior art keywords
aza
cyclical
improved
certain bis
phthalimido
Prior art date
Application number
MX9200802A
Other languages
English (en)
Inventor
Dennis Michael Godek
Charles William Murtiashaw
Frank John Urban
Brian Clement Vanderplas
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX9200802A publication Critical patent/MX9200802A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Reinforced Plastic Materials (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
MX9200802A 1991-02-27 1992-02-25 Procedimientos mejorado e intermediario para ciertos agentes bis-aza-bi-ciclicos anxioliticos. MX9200802A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/661,730 US5185449A (en) 1991-02-27 1991-02-27 Process and intermediate for certain bis-aza-bicyclic anxiolytic agents

Publications (1)

Publication Number Publication Date
MX9200802A true MX9200802A (es) 1992-08-01

Family

ID=24654869

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9200802A MX9200802A (es) 1991-02-27 1992-02-25 Procedimientos mejorado e intermediario para ciertos agentes bis-aza-bi-ciclicos anxioliticos.

Country Status (23)

Country Link
US (1) US5185449A (es)
EP (1) EP0586376B1 (es)
JP (1) JPH0784467B2 (es)
KR (1) KR100189044B1 (es)
AT (1) ATE153662T1 (es)
AU (1) AU647562B2 (es)
CA (1) CA2101433C (es)
DE (1) DE69126326T2 (es)
DK (1) DK0586376T3 (es)
ES (1) ES2101831T3 (es)
FI (1) FI107153B (es)
GR (1) GR3024125T3 (es)
HU (2) HU223138B1 (es)
IE (1) IE920600A1 (es)
IL (1) IL101022A (es)
MX (1) MX9200802A (es)
MY (1) MY110167A (es)
NO (1) NO302947B1 (es)
NZ (1) NZ241738A (es)
PT (1) PT100161B (es)
TW (1) TW268949B (es)
WO (1) WO1992015575A1 (es)
ZA (1) ZA921406B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2101252C (en) * 1991-02-27 1998-02-17 Frank J. Urban Process for preparing trans-piperidine-2,5- dicarboxylates
WO1996010570A1 (en) * 1994-09-30 1996-04-11 Pfizer Inc. NEUROLEPTIC 2,7-DISUBSTITUTED PERHYDRO-1H-PYRIDO[1,2-a]PYRAZINES
WO1996010571A1 (en) * 1994-09-30 1996-04-11 Pfizer Inc. 2,7-SUBSTITUTED OCTAHYDRO-1H-PYRIDO[1,2-a]PYRAZINE DERIVATIVES
US6670476B2 (en) 2000-11-29 2003-12-30 Pfizer Inc. Resolution of trans-7-(hydroxy-methyl)octa-hydro-2H-pyrido[1,2-a]pyrazine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3388128A (en) * 1965-09-03 1968-06-11 Allan R. Day Substituted 1, 4-diazabicyclo [4. 4. 9] decanes
WO1990008148A1 (en) * 1989-01-23 1990-07-26 Pfizer Inc. Bis-aza-bicyclic anxiolytic agents
CA2101252C (en) * 1991-02-27 1998-02-17 Frank J. Urban Process for preparing trans-piperidine-2,5- dicarboxylates

Also Published As

Publication number Publication date
HUT67440A (en) 1995-04-28
DE69126326T2 (de) 1997-09-04
AU9066691A (en) 1992-10-06
HU9302428D0 (en) 1993-11-29
IE920600A1 (en) 1992-09-09
CA2101433C (en) 1999-07-27
FI107153B (fi) 2001-06-15
AU647562B2 (en) 1994-03-24
NZ241738A (en) 1993-05-26
NO933048L (no) 1993-08-26
ZA921406B (en) 1993-08-26
FI933754A (fi) 1993-08-26
DK0586376T3 (da) 1997-10-27
DE69126326D1 (de) 1997-07-03
US5185449A (en) 1993-02-09
PT100161A (pt) 1993-05-31
ES2101831T3 (es) 1997-07-16
CA2101433A1 (en) 1992-08-28
NO302947B1 (no) 1998-05-11
JPH0784467B2 (ja) 1995-09-13
KR100189044B1 (ko) 1999-06-01
HU223138B1 (hu) 2004-03-29
WO1992015575A1 (en) 1992-09-17
IL101022A (en) 1996-06-18
JPH06501021A (ja) 1994-01-27
MY110167A (en) 1998-02-28
GR3024125T3 (en) 1997-10-31
NO933048D0 (no) 1993-08-26
PT100161B (pt) 1999-09-30
IL101022A0 (en) 1992-11-15
EP0586376A1 (en) 1994-03-16
FI933754A0 (fi) 1993-08-26
TW268949B (es) 1996-01-21
EP0586376B1 (en) 1997-05-28
ATE153662T1 (de) 1997-06-15

Similar Documents

Publication Publication Date Title
ES2101960T3 (es) Lactamas benzo-condensadas.
FR2687675B1 (fr) Nouveaux derives bicycliques de la pyridine, leur procede de preparation, les nouveaux intermediaires obtenus, leur application a titre de medicaments et les compositions pharmaceutiques les renfermant.
DK0776324T3 (da) Endothelin-antagonister
ATE417836T1 (de) Verfahren und intermediate zur herstellung von retroviralen proteasehemmern
NO1998008I1 (no) Naratriptan
EP0291799A3 (en) Dioxyalkylenearyl-dihydropyridines and their intermediary compounds, process for their preparation and their use
ATE54913T1 (de) Industrielle verbindungen anwendbar als zwischenprodukte in der herstellung von in stellung 2 substituierten 4-hydroxy 3quinolincarboxamid-derivaten und die herstellung von diesen zwischenprodukten.
MX9200802A (es) Procedimientos mejorado e intermediario para ciertos agentes bis-aza-bi-ciclicos anxioliticos.
FI832739A0 (fi) 5-alkyl-1,6-naftyridin-2(1h)-oner, mellanprodukter deras framstaellning och anvaendning som hjaertlaekemedel
FI896251A0 (fi) Menetelmä uusien terapeuttisesti käyttökelpoisten pyratsolopyridiinijohdannaisten valmistamiseksi
ATE150453T1 (de) Verfahren zur herstellung von trans-piperidin-2,5-dicarboxylaten
FI932691A (fi) Nya benzyl- och benzhydrylalkoholer
DE3864286D1 (de) Herstellungsverfahren von trifluormethylverbindungen.
ES2049652B1 (es) Procedimiento para la preparacion de un acido quinolin carboxilico.
IT1254201B (it) Procedimento per la preparazione di derivati del glicerolo otticamente attivi.
MX9703074A (es) Inhibidores de sintesis de apoliproteina-b.
ES2095831T3 (es) Acidos tetrahidro-4-fenilimino-3-tiofeno-aceticos.

Legal Events

Date Code Title Description
FG Grant or registration
MM Annulment or lapse due to non-payment of fees