DK0573464T3 - Fremgangsmåde til fremstilling af trans-piperidin-2,5-dicarboxylater - Google Patents
Fremgangsmåde til fremstilling af trans-piperidin-2,5-dicarboxylaterInfo
- Publication number
- DK0573464T3 DK0573464T3 DK92904789.2T DK92904789T DK0573464T3 DK 0573464 T3 DK0573464 T3 DK 0573464T3 DK 92904789 T DK92904789 T DK 92904789T DK 0573464 T3 DK0573464 T3 DK 0573464T3
- Authority
- DK
- Denmark
- Prior art keywords
- preparation
- dicarboxylates
- piperidine
- trans
- pyrazines
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/582—Recycling of unreacted starting or intermediate materials
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66172691A | 1991-02-27 | 1991-02-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0573464T3 true DK0573464T3 (da) | 1997-09-01 |
Family
ID=24654845
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK92904789.2T DK0573464T3 (da) | 1991-02-27 | 1992-01-08 | Fremgangsmåde til fremstilling af trans-piperidin-2,5-dicarboxylater |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US5326874A (da) |
| EP (2) | EP0573464B1 (da) |
| JP (1) | JPH0725736B2 (da) |
| AT (1) | ATE150453T1 (da) |
| CA (2) | CA2101252C (da) |
| DE (1) | DE69218414T2 (da) |
| DK (1) | DK0573464T3 (da) |
| ES (1) | ES2099820T3 (da) |
| FI (2) | FI933755A (da) |
| GR (1) | GR3023381T3 (da) |
| IE (2) | IE970704A1 (da) |
| PT (1) | PT100159B (da) |
| WO (1) | WO1992015561A2 (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5185449A (en) * | 1991-02-27 | 1993-02-09 | Pfizer Inc. | Process and intermediate for certain bis-aza-bicyclic anxiolytic agents |
| WO1996010571A1 (en) * | 1994-09-30 | 1996-04-11 | Pfizer Inc. | 2,7-SUBSTITUTED OCTAHYDRO-1H-PYRIDO[1,2-a]PYRAZINE DERIVATIVES |
| USRE43932E1 (en) | 1997-07-18 | 2013-01-15 | Novartis Ag | Crystal modification of a N-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use |
| GB0001447D0 (en) | 2000-01-21 | 2000-03-08 | Novartis Ag | Organic compounds |
| PL362930A1 (en) | 2000-11-08 | 2004-11-02 | Syngenta Participations Ag | Pyrrolcarboxamides and pyrrolcarbothioamides and their agrochemical uses |
| AU2020347715A1 (en) | 2019-09-18 | 2022-04-07 | Baili-Bio (Chengdu) Pharmaceutical Co., Ltd. | Camptothecin derivative and conjugate thereof |
| CN116120460A (zh) | 2021-11-15 | 2023-05-16 | 成都百利多特生物药业有限责任公司 | 双特异性抗体-喜树碱类药物偶联物及其医药用途 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4018767A (en) * | 1975-05-22 | 1977-04-19 | Bristol-Myers Company | Anti-arrhythmic agents |
| US4401820A (en) * | 1981-01-23 | 1983-08-30 | Tanabe Seiyaku Co., Ltd. | Process for racemizing optically active α-amino acids or a salt thereof |
| US4505911A (en) * | 1983-10-13 | 1985-03-19 | Mead Johnson & Company | Isoindole diuretic derivatives, compositions and use |
| WO1990008148A1 (en) * | 1989-01-23 | 1990-07-26 | Pfizer Inc. | Bis-aza-bicyclic anxiolytic agents |
| US5157034A (en) * | 1991-02-27 | 1992-10-20 | Pfizer Inc. | Neuroleptic perhydro-1H-pyrido[1,2-a]pyrazines |
| US5185449A (en) * | 1991-02-27 | 1993-02-09 | Pfizer Inc. | Process and intermediate for certain bis-aza-bicyclic anxiolytic agents |
-
1992
- 1992-01-08 CA CA002101252A patent/CA2101252C/en not_active Expired - Fee Related
- 1992-01-08 WO PCT/US1992/000029 patent/WO1992015561A2/en active IP Right Grant
- 1992-01-08 EP EP92904789A patent/EP0573464B1/en not_active Expired - Lifetime
- 1992-01-08 ES ES92904789T patent/ES2099820T3/es not_active Expired - Lifetime
- 1992-01-08 DE DE69218414T patent/DE69218414T2/de not_active Expired - Fee Related
- 1992-01-08 AT AT92904789T patent/ATE150453T1/de not_active IP Right Cessation
- 1992-01-08 CA CA002195622A patent/CA2195622C/en not_active Expired - Fee Related
- 1992-01-08 EP EP96201187A patent/EP0737683A1/en not_active Withdrawn
- 1992-01-08 US US08/104,153 patent/US5326874A/en not_active Expired - Lifetime
- 1992-01-08 JP JP4505284A patent/JPH0725736B2/ja not_active Expired - Lifetime
- 1992-01-08 DK DK92904789.2T patent/DK0573464T3/da active
- 1992-02-25 PT PT100159A patent/PT100159B/pt not_active IP Right Cessation
- 1992-02-26 IE IE19970704A patent/IE970704A1/en unknown
- 1992-02-26 IE IE059992A patent/IE920599A1/en not_active Application Discontinuation
-
1993
- 1993-08-26 FI FI933755A patent/FI933755A/fi unknown
-
1994
- 1994-03-24 US US08/217,532 patent/US5489688A/en not_active Expired - Fee Related
-
1996
- 1996-07-05 FI FI962768A patent/FI962768A0/fi unknown
-
1997
- 1997-05-09 GR GR970401034T patent/GR3023381T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI962768A (fi) | 1996-07-05 |
| JPH06500121A (ja) | 1994-01-06 |
| JPH0725736B2 (ja) | 1995-03-22 |
| CA2195622A1 (en) | 1992-08-28 |
| ATE150453T1 (de) | 1997-04-15 |
| CA2101252C (en) | 1998-02-17 |
| US5326874A (en) | 1994-07-05 |
| GR3023381T3 (en) | 1997-08-29 |
| EP0573464B1 (en) | 1997-03-19 |
| DE69218414T2 (de) | 1998-01-22 |
| FI962768A0 (fi) | 1996-07-05 |
| CA2195622C (en) | 1999-08-17 |
| FI933755A0 (fi) | 1993-08-26 |
| US5489688A (en) | 1996-02-06 |
| IE970704A1 (en) | 2000-02-23 |
| IE920599A1 (en) | 1992-09-09 |
| EP0737683A1 (en) | 1996-10-16 |
| CA2101252A1 (en) | 1992-08-28 |
| EP0573464A1 (en) | 1993-12-15 |
| ES2099820T3 (es) | 1997-06-01 |
| FI933755A (fi) | 1993-08-26 |
| PT100159B (pt) | 1999-07-30 |
| WO1992015561A2 (en) | 1992-09-17 |
| WO1992015561A3 (en) | 1993-01-07 |
| DE69218414D1 (de) | 1997-04-24 |
| PT100159A (pt) | 1993-05-31 |
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