ES2383239T3 - Compuestos de ácidos policíclicos útiles como antagonistas de CRTH2 y como agentes antialérgicos - Google Patents

Compuestos de ácidos policíclicos útiles como antagonistas de CRTH2 y como agentes antialérgicos Download PDF

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ES2383239T3
ES2383239T3 ES07859872T ES07859872T ES2383239T3 ES 2383239 T3 ES2383239 T3 ES 2383239T3 ES 07859872 T ES07859872 T ES 07859872T ES 07859872 T ES07859872 T ES 07859872T ES 2383239 T3 ES2383239 T3 ES 2383239T3
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esi
phenoxy
preparation
nmr
propyl
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Tadashi Terasaka
Tatsuya; HAYASHIDA Hisashi ZENKOH
Hiroshi; SATO Junji MATSUDA
Yoshimasa;NAGATA Hiroshi IMAMURA
Norio; TENDA Yoshiyuki SEKI
Mamoru; TAKEDA Masahiro TASAKI
Seiichiro; YASUDA Minoru TABUCHI
Kazunori Tsubaki
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Astellas Pharma Inc
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Astellas Pharma Inc
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/63—One oxygen atom
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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CN105353095B (zh) * 2015-11-16 2017-10-20 华南农业大学 一种西地那非及其结构类似物的免疫检测方法
WO2017104728A1 (ja) * 2015-12-16 2017-06-22 国立大学法人東京大学 食物アレルギー治療薬
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