ES2286263T3 - Sistemas de suministro secuencial de farmacos. - Google Patents
Sistemas de suministro secuencial de farmacos. Download PDFInfo
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- ES2286263T3 ES2286263T3 ES02749899T ES02749899T ES2286263T3 ES 2286263 T3 ES2286263 T3 ES 2286263T3 ES 02749899 T ES02749899 T ES 02749899T ES 02749899 T ES02749899 T ES 02749899T ES 2286263 T3 ES2286263 T3 ES 2286263T3
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- XNGIFLGASWRNHJ-UHFFFAOYSA-L phthalate(2-) Chemical compound [O-]C(=O)C1=CC=CC=C1C([O-])=O XNGIFLGASWRNHJ-UHFFFAOYSA-L 0.000 description 1
- 239000000419 plant extract Substances 0.000 description 1
- 229950005134 polycarbophil Drugs 0.000 description 1
- 229940113116 polyethylene glycol 1000 Drugs 0.000 description 1
- 229940057838 polyethylene glycol 4000 Drugs 0.000 description 1
- 229920001282 polysaccharide Polymers 0.000 description 1
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- 229940100467 polyvinyl acetate phthalate Drugs 0.000 description 1
- 229920002451 polyvinyl alcohol Polymers 0.000 description 1
- 229920000523 polyvinylpolypyrrolidone Polymers 0.000 description 1
- 235000013809 polyvinylpolypyrrolidone Nutrition 0.000 description 1
- 239000001267 polyvinylpyrrolidone Substances 0.000 description 1
- 239000011736 potassium bicarbonate Substances 0.000 description 1
- 235000015497 potassium bicarbonate Nutrition 0.000 description 1
- 229910000028 potassium bicarbonate Inorganic materials 0.000 description 1
- 229910000027 potassium carbonate Inorganic materials 0.000 description 1
- 235000011181 potassium carbonates Nutrition 0.000 description 1
- TYJJADVDDVDEDZ-UHFFFAOYSA-M potassium hydrogencarbonate Chemical compound [K+].OC([O-])=O TYJJADVDDVDEDZ-UHFFFAOYSA-M 0.000 description 1
- 229920001592 potato starch Polymers 0.000 description 1
- 229940069328 povidone Drugs 0.000 description 1
- 239000002244 precipitate Substances 0.000 description 1
- 230000002028 premature Effects 0.000 description 1
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- 239000000047 product Substances 0.000 description 1
- 230000002035 prolonged effect Effects 0.000 description 1
- 235000010232 propyl p-hydroxybenzoate Nutrition 0.000 description 1
- 239000004405 propyl p-hydroxybenzoate Substances 0.000 description 1
- 229960003415 propylparaben Drugs 0.000 description 1
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- 230000009467 reduction Effects 0.000 description 1
- 230000001105 regulatory effect Effects 0.000 description 1
- 230000002441 reversible effect Effects 0.000 description 1
- 239000010670 sage oil Substances 0.000 description 1
- ZLGIYFNHBLSMPS-ATJNOEHPSA-N shellac Chemical compound OCCCCCC(O)C(O)CCCCCCCC(O)=O.C1C23[C@H](C(O)=O)CCC2[C@](C)(CO)[C@@H]1C(C(O)=O)=C[C@@H]3O ZLGIYFNHBLSMPS-ATJNOEHPSA-N 0.000 description 1
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- 235000019812 sodium carboxymethyl cellulose Nutrition 0.000 description 1
- 229920001027 sodium carboxymethylcellulose Polymers 0.000 description 1
- BYKRNSHANADUFY-UHFFFAOYSA-M sodium octanoate Chemical compound [Na+].CCCCCCCC([O-])=O BYKRNSHANADUFY-UHFFFAOYSA-M 0.000 description 1
- 238000007711 solidification Methods 0.000 description 1
- 230000008023 solidification Effects 0.000 description 1
- 239000011877 solvent mixture Substances 0.000 description 1
- 239000000600 sorbitol Substances 0.000 description 1
- 238000001179 sorption measurement Methods 0.000 description 1
- 238000005563 spheronization Methods 0.000 description 1
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- 239000000454 talc Substances 0.000 description 1
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- 230000001225 therapeutic effect Effects 0.000 description 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/48—Ergoline derivatives, e.g. lysergic acid, ergotamine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
- A61K9/025—Suppositories; Bougies; Bases therefor; Ovules characterised by shape or structure, e.g. hollow layered, coated
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Urology & Nephrology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
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| US901983 | 2001-07-10 | ||
| US09/901,983 US20030068356A1 (en) | 2001-07-10 | 2001-07-10 | Sequential drug delivery systems |
Publications (1)
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| ES2286263T3 true ES2286263T3 (es) | 2007-12-01 |
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| ES07006505.7T Expired - Lifetime ES2604780T3 (es) | 2001-07-10 | 2002-07-10 | Sistemas de liberación secuencial de fármacos |
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| EP (2) | EP1818029B1 (enExample) |
| JP (1) | JP4617081B2 (enExample) |
| AT (1) | ATE363261T1 (enExample) |
| AU (2) | AU2002320385B2 (enExample) |
| CA (1) | CA2451106C (enExample) |
| DE (1) | DE60220408T2 (enExample) |
| DK (1) | DK1406568T3 (enExample) |
| ES (2) | ES2286263T3 (enExample) |
| WO (1) | WO2003005944A1 (enExample) |
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| US20080213363A1 (en) * | 2003-01-23 | 2008-09-04 | Singh Nikhilesh N | Methods and compositions for delivering 5-HT3 antagonists across the oral mucosa |
| EP1449525A1 (en) * | 2003-02-20 | 2004-08-25 | Cross Chem Llc | chewing gum in the form of multi-layer tablets |
| KR100767271B1 (ko) * | 2003-07-11 | 2007-10-17 | 에프. 호프만-라 로슈 아게 | 사퀴나비르 메실레이트 경구 투여 형태 |
| UA81335C2 (uk) * | 2003-07-11 | 2007-12-25 | Ф.Хоффманн-Ля Рош Аг | Оральна дозована форма саквінавіру мезилату |
| CN1819821B (zh) | 2003-08-08 | 2010-10-13 | 拜奥维尔实验室国际股份有限公司 | 盐酸安非他酮的改良释放片剂 |
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| KR101184138B1 (ko) * | 2003-12-31 | 2012-09-19 | 시마 랩스 인크. | 일반적인 선형 발포성 경구 펜타닐 투약 제형 및 투여 방법 |
| WO2005065317A2 (en) * | 2003-12-31 | 2005-07-21 | Cima Labs Inc. | Effervescent oral fentanyl dosage form |
| NZ548215A (en) * | 2003-12-31 | 2009-08-28 | Cima Labs Inc | Effervescent oral opiate dosage form |
| US20070036853A1 (en) * | 2003-12-31 | 2007-02-15 | Cima Labs Inc. | Generally linear effervescent oral fentanyl dosage form and methods of administering |
-
2001
- 2001-07-10 US US09/901,983 patent/US20030068356A1/en not_active Abandoned
-
2002
- 2002-07-10 WO PCT/US2002/021796 patent/WO2003005944A1/en not_active Ceased
- 2002-07-10 AT AT02749899T patent/ATE363261T1/de active
- 2002-07-10 EP EP07006505.7A patent/EP1818029B1/en not_active Expired - Lifetime
- 2002-07-10 CA CA002451106A patent/CA2451106C/en not_active Expired - Fee Related
- 2002-07-10 ES ES02749899T patent/ES2286263T3/es not_active Expired - Lifetime
- 2002-07-10 ES ES07006505.7T patent/ES2604780T3/es not_active Expired - Lifetime
- 2002-07-10 DK DK02749899T patent/DK1406568T3/da active
- 2002-07-10 JP JP2003511754A patent/JP4617081B2/ja not_active Expired - Fee Related
- 2002-07-10 EP EP02749899A patent/EP1406568B1/en not_active Expired - Lifetime
- 2002-07-10 AU AU2002320385A patent/AU2002320385B2/en not_active Ceased
- 2002-07-10 DE DE60220408T patent/DE60220408T2/de not_active Expired - Lifetime
-
2003
- 2003-07-18 US US10/623,069 patent/US20030232080A1/en not_active Abandoned
-
2004
- 2004-09-08 US US10/936,185 patent/US7670617B2/en not_active Expired - Fee Related
-
2008
- 2008-08-01 AU AU2008203464A patent/AU2008203464B2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| ATE363261T1 (de) | 2007-06-15 |
| US20050031677A1 (en) | 2005-02-10 |
| HK1106126A1 (en) | 2008-03-07 |
| EP1406568A4 (en) | 2004-12-15 |
| EP1818029B1 (en) | 2016-09-07 |
| EP1818029A3 (en) | 2008-06-11 |
| US20030232080A1 (en) | 2003-12-18 |
| DE60220408T2 (de) | 2008-01-31 |
| AU2008203464A1 (en) | 2008-08-21 |
| EP1406568A1 (en) | 2004-04-14 |
| DK1406568T3 (da) | 2007-10-01 |
| AU2008203464B2 (en) | 2010-07-01 |
| JP4617081B2 (ja) | 2011-01-19 |
| CA2451106A1 (en) | 2003-01-23 |
| EP1818029A2 (en) | 2007-08-15 |
| WO2003005944A1 (en) | 2003-01-23 |
| ES2604780T3 (es) | 2017-03-09 |
| EP1406568B1 (en) | 2007-05-30 |
| US20030068356A1 (en) | 2003-04-10 |
| JP2004534839A (ja) | 2004-11-18 |
| US7670617B2 (en) | 2010-03-02 |
| DE60220408D1 (de) | 2007-07-12 |
| CA2451106C (en) | 2009-12-22 |
| AU2002320385B2 (en) | 2008-05-01 |
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