ES2280802T3 - Complejos de androstano antiinflamatorios o antialergicos. - Google Patents
Complejos de androstano antiinflamatorios o antialergicos. Download PDFInfo
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- ES2280802T3 ES2280802T3 ES03765110T ES03765110T ES2280802T3 ES 2280802 T3 ES2280802 T3 ES 2280802T3 ES 03765110 T ES03765110 T ES 03765110T ES 03765110 T ES03765110 T ES 03765110T ES 2280802 T3 ES2280802 T3 ES 2280802T3
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US200364 | 2002-07-22 | ||
| US10/200,364 US6858593B2 (en) | 2000-08-05 | 2002-07-22 | Anti-inflammatory androstane derivative compositions |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2280802T3 true ES2280802T3 (es) | 2007-09-16 |
Family
ID=30769534
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES03765110T Expired - Lifetime ES2280802T3 (es) | 2002-07-22 | 2003-07-21 | Complejos de androstano antiinflamatorios o antialergicos. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US6858593B2 (enExample) |
| EP (1) | EP1539796B1 (enExample) |
| JP (1) | JP2005537278A (enExample) |
| AT (1) | ATE353908T1 (enExample) |
| AU (1) | AU2003253354A1 (enExample) |
| DE (1) | DE60311831T2 (enExample) |
| DK (1) | DK1539796T3 (enExample) |
| ES (1) | ES2280802T3 (enExample) |
| PT (1) | PT1539796E (enExample) |
| SI (1) | SI1539796T1 (enExample) |
| WO (1) | WO2004009613A1 (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020133032A1 (en) * | 2000-02-25 | 2002-09-19 | Jufang Barkalow | Method for the preparation of fluticasone and related 17beta-carbothioic esters using a novel carbothioic acid synthesis and novel purification methods |
| US6777399B2 (en) * | 2000-08-05 | 2004-08-17 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative compositions |
| GB0019172D0 (en) | 2000-08-05 | 2000-09-27 | Glaxo Group Ltd | Novel compounds |
| AU7576001A (en) * | 2000-08-05 | 2002-02-18 | Glaxo Group Ltd | 6.alpha., 9.alpha.-difluoro-17.alpha.-`(2-furanylcarboxyl) oxy]-11.beta.-hydroxy-16.alpha.-methyl-3-oxo-androst-1,4,-diene-17-carbothioic acid s-fluoromethyl ester as an anti-inflammatory agent |
| US6759398B2 (en) * | 2000-08-05 | 2004-07-06 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative |
| US6858596B2 (en) | 2000-08-05 | 2005-02-22 | Smithkline Beecham Corporation | Formulation containing anti-inflammatory androstane derivative |
| UA77656C2 (en) | 2001-04-07 | 2007-01-15 | Glaxo Group Ltd | S-fluoromethyl ester of 6-alpha, 9-alpha-difluoro-17-alpha-[(2-furanylcarbonyl)oxy]-11-beta-hydroxy-16- alpha-methyl-3-oxoandrosta-1,4-dien-17-beta-carbothioacid as anti-inflammatory agent |
| WO2002088167A1 (en) * | 2001-04-30 | 2002-11-07 | Glaxo Group Limited | Anti-inflammatory 17.beta.-carbothioate ester derivatives of androstane with a cyclic ester group in position 17.alpha |
| ES2307751T3 (es) * | 2001-06-12 | 2008-12-01 | Glaxo Group Limited | Nuevos esteres heterociclicos centi-inflamatorios 17 alfa de derivados 17 beta de carbotioato de androstano. |
| GB0125259D0 (en) * | 2001-10-20 | 2001-12-12 | Glaxo Group Ltd | Novel compounds |
| US20050175545A1 (en) * | 2002-02-04 | 2005-08-11 | Keith Biggadike | Formulation for inhalation comprising a glucocorticoid and a beta 2-adrenoreceptor agonist |
| WO2003066655A1 (en) * | 2002-02-04 | 2003-08-14 | Glaxo Group Limited | Amorphous fluticasone 2-furoate, pharmaceutical compositions thereof and its conversion to the crystalline unsolvated form |
| GB0202635D0 (en) * | 2002-02-05 | 2002-03-20 | Glaxo Wellcome Mfg Pte Ltd | Formulation containing novel anti-inflammatory androstane derivative |
| GB2389530B (en) | 2002-06-14 | 2007-01-10 | Cipla Ltd | Pharmaceutical compositions |
| GB0507165D0 (en) * | 2005-04-08 | 2005-05-18 | Glaxo Group Ltd | Novel crystalline pharmaceutical product |
| GB0615108D0 (en) * | 2006-07-28 | 2006-09-06 | Glaxo Group Ltd | Novel formulations |
| US8148353B2 (en) * | 2008-08-07 | 2012-04-03 | Plus Chemicals Sa | Polymorphs of fluticasone furoate and process for preparation thereof |
| US20100240629A1 (en) * | 2009-03-19 | 2010-09-23 | Adrienne Kovacsne-Mezei | Polymorphs of fluticasone furoate and processes for preparation thereof |
| EP2593444B1 (en) | 2010-07-15 | 2015-04-08 | Battelle Memorial Institute | Biobased polyols for potential use as flame retardants in polyurethane and polyester applications |
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| AU2002321884A1 (en) | 2001-08-03 | 2003-02-24 | Smithkline Beecham Corporation | A method for preparing fluticasone derivatives |
| GB0124523D0 (en) | 2001-10-12 | 2001-12-05 | Glaxo Group Ltd | Pharmaceutical combination |
| GB0125259D0 (en) | 2001-10-20 | 2001-12-12 | Glaxo Group Ltd | Novel compounds |
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| GB0127160D0 (en) | 2001-11-12 | 2002-01-02 | Glaxo Group Ltd | Novel compounds |
-
2002
- 2002-07-22 US US10/200,364 patent/US6858593B2/en not_active Expired - Fee Related
-
2003
- 2003-07-21 JP JP2004522571A patent/JP2005537278A/ja active Pending
- 2003-07-21 AU AU2003253354A patent/AU2003253354A1/en not_active Abandoned
- 2003-07-21 PT PT03765110T patent/PT1539796E/pt unknown
- 2003-07-21 DE DE60311831T patent/DE60311831T2/de not_active Expired - Fee Related
- 2003-07-21 ES ES03765110T patent/ES2280802T3/es not_active Expired - Lifetime
- 2003-07-21 WO PCT/EP2003/008388 patent/WO2004009613A1/en not_active Ceased
- 2003-07-21 AT AT03765110T patent/ATE353908T1/de not_active IP Right Cessation
- 2003-07-21 DK DK03765110T patent/DK1539796T3/da active
- 2003-07-21 EP EP03765110A patent/EP1539796B1/en not_active Expired - Lifetime
- 2003-07-21 SI SI200330714T patent/SI1539796T1/sl unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2005537278A (ja) | 2005-12-08 |
| US20030109511A1 (en) | 2003-06-12 |
| DE60311831D1 (de) | 2007-03-29 |
| US6858593B2 (en) | 2005-02-22 |
| PT1539796E (pt) | 2007-04-30 |
| DE60311831T2 (de) | 2007-11-22 |
| WO2004009613A1 (en) | 2004-01-29 |
| ATE353908T1 (de) | 2007-03-15 |
| EP1539796A1 (en) | 2005-06-15 |
| EP1539796B1 (en) | 2007-02-14 |
| AU2003253354A1 (en) | 2004-02-09 |
| SI1539796T1 (sl) | 2007-06-30 |
| DK1539796T3 (da) | 2007-05-29 |
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