AU2003253354A1 - Anti-inflammatory or anti-allergic androstane complexes - Google Patents

Anti-inflammatory or anti-allergic androstane complexes

Info

Publication number
AU2003253354A1
AU2003253354A1 AU2003253354A AU2003253354A AU2003253354A1 AU 2003253354 A1 AU2003253354 A1 AU 2003253354A1 AU 2003253354 A AU2003253354 A AU 2003253354A AU 2003253354 A AU2003253354 A AU 2003253354A AU 2003253354 A1 AU2003253354 A1 AU 2003253354A1
Authority
AU
Australia
Prior art keywords
androstane
allergic
complexes
inflammatory
crystalline
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003253354A
Other languages
English (en)
Inventor
Keith Biggadike
Olga Chetina
Steven John Coote
Andrew Simon Craig
Victor Witold Jacewicz
Michael John Millan
John Frederick Seager
Andrew Lewis Theophilus
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of AU2003253354A1 publication Critical patent/AU2003253354A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2003253354A 2002-07-22 2003-07-21 Anti-inflammatory or anti-allergic androstane complexes Abandoned AU2003253354A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10/200,364 US6858593B2 (en) 2000-08-05 2002-07-22 Anti-inflammatory androstane derivative compositions
US10/200,364 2002-07-22
PCT/EP2003/008388 WO2004009613A1 (en) 2002-07-22 2003-07-21 Anti-inflammatory or anti-allergic androstane complexes

Publications (1)

Publication Number Publication Date
AU2003253354A1 true AU2003253354A1 (en) 2004-02-09

Family

ID=30769534

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003253354A Abandoned AU2003253354A1 (en) 2002-07-22 2003-07-21 Anti-inflammatory or anti-allergic androstane complexes

Country Status (11)

Country Link
US (1) US6858593B2 (enExample)
EP (1) EP1539796B1 (enExample)
JP (1) JP2005537278A (enExample)
AT (1) ATE353908T1 (enExample)
AU (1) AU2003253354A1 (enExample)
DE (1) DE60311831T2 (enExample)
DK (1) DK1539796T3 (enExample)
ES (1) ES2280802T3 (enExample)
PT (1) PT1539796E (enExample)
SI (1) SI1539796T1 (enExample)
WO (1) WO2004009613A1 (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020133032A1 (en) * 2000-02-25 2002-09-19 Jufang Barkalow Method for the preparation of fluticasone and related 17beta-carbothioic esters using a novel carbothioic acid synthesis and novel purification methods
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US6777399B2 (en) * 2000-08-05 2004-08-17 Smithkline Beecham Corporation Anti-inflammatory androstane derivative compositions
US6858596B2 (en) * 2000-08-05 2005-02-22 Smithkline Beecham Corporation Formulation containing anti-inflammatory androstane derivative
US6759398B2 (en) * 2000-08-05 2004-07-06 Smithkline Beecham Corporation Anti-inflammatory androstane derivative
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US7291608B2 (en) * 2001-04-30 2007-11-06 Glaxo Group Limited Anti-inflammatory 17.β.-carbothioate ester derivatives of androstane with a cyclic ester group in position 17.α
ES2307751T3 (es) * 2001-06-12 2008-12-01 Glaxo Group Limited Nuevos esteres heterociclicos centi-inflamatorios 17 alfa de derivados 17 beta de carbotioato de androstano.
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GB0507165D0 (en) * 2005-04-08 2005-05-18 Glaxo Group Ltd Novel crystalline pharmaceutical product
GB0615108D0 (en) * 2006-07-28 2006-09-06 Glaxo Group Ltd Novel formulations
US8148353B2 (en) * 2008-08-07 2012-04-03 Plus Chemicals Sa Polymorphs of fluticasone furoate and process for preparation thereof
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Also Published As

Publication number Publication date
DE60311831D1 (de) 2007-03-29
JP2005537278A (ja) 2005-12-08
US6858593B2 (en) 2005-02-22
PT1539796E (pt) 2007-04-30
EP1539796B1 (en) 2007-02-14
EP1539796A1 (en) 2005-06-15
US20030109511A1 (en) 2003-06-12
SI1539796T1 (sl) 2007-06-30
ES2280802T3 (es) 2007-09-16
DE60311831T2 (de) 2007-11-22
ATE353908T1 (de) 2007-03-15
DK1539796T3 (da) 2007-05-29
WO2004009613A1 (en) 2004-01-29

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Legal Events

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MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase