ATE353908T1 - Entzündungshemmende bzw. antiallergische androstankomplexe - Google Patents

Entzündungshemmende bzw. antiallergische androstankomplexe

Info

Publication number
ATE353908T1
ATE353908T1 AT03765110T AT03765110T ATE353908T1 AT E353908 T1 ATE353908 T1 AT E353908T1 AT 03765110 T AT03765110 T AT 03765110T AT 03765110 T AT03765110 T AT 03765110T AT E353908 T1 ATE353908 T1 AT E353908T1
Authority
AT
Austria
Prior art keywords
androstane
antiallergic
complexes
inflammatory
crystalline
Prior art date
Application number
AT03765110T
Other languages
German (de)
English (en)
Inventor
Keith Biggadike
Olga Chetina
Steven John Coote
Andrew Simon Craig
Victor Witold Jacewicz
Michael John Millan
John Frederick Seager
Andrew Lewis Theophilus
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE353908T1 publication Critical patent/ATE353908T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT03765110T 2002-07-22 2003-07-21 Entzündungshemmende bzw. antiallergische androstankomplexe ATE353908T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10/200,364 US6858593B2 (en) 2000-08-05 2002-07-22 Anti-inflammatory androstane derivative compositions

Publications (1)

Publication Number Publication Date
ATE353908T1 true ATE353908T1 (de) 2007-03-15

Family

ID=30769534

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03765110T ATE353908T1 (de) 2002-07-22 2003-07-21 Entzündungshemmende bzw. antiallergische androstankomplexe

Country Status (11)

Country Link
US (1) US6858593B2 (enExample)
EP (1) EP1539796B1 (enExample)
JP (1) JP2005537278A (enExample)
AT (1) ATE353908T1 (enExample)
AU (1) AU2003253354A1 (enExample)
DE (1) DE60311831T2 (enExample)
DK (1) DK1539796T3 (enExample)
ES (1) ES2280802T3 (enExample)
PT (1) PT1539796E (enExample)
SI (1) SI1539796T1 (enExample)
WO (1) WO2004009613A1 (enExample)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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US6759398B2 (en) * 2000-08-05 2004-07-06 Smithkline Beecham Corporation Anti-inflammatory androstane derivative
US6858596B2 (en) 2000-08-05 2005-02-22 Smithkline Beecham Corporation Formulation containing anti-inflammatory androstane derivative
UA77656C2 (en) 2001-04-07 2007-01-15 Glaxo Group Ltd S-fluoromethyl ester of 6-alpha, 9-alpha-difluoro-17-alpha-[(2-furanylcarbonyl)oxy]-11-beta-hydroxy-16- alpha-methyl-3-oxoandrosta-1,4-dien-17-beta-carbothioacid as anti-inflammatory agent
WO2002088167A1 (en) * 2001-04-30 2002-11-07 Glaxo Group Limited Anti-inflammatory 17.beta.-carbothioate ester derivatives of androstane with a cyclic ester group in position 17.alpha
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US8148353B2 (en) * 2008-08-07 2012-04-03 Plus Chemicals Sa Polymorphs of fluticasone furoate and process for preparation thereof
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Also Published As

Publication number Publication date
JP2005537278A (ja) 2005-12-08
US20030109511A1 (en) 2003-06-12
DE60311831D1 (de) 2007-03-29
ES2280802T3 (es) 2007-09-16
US6858593B2 (en) 2005-02-22
PT1539796E (pt) 2007-04-30
DE60311831T2 (de) 2007-11-22
WO2004009613A1 (en) 2004-01-29
EP1539796A1 (en) 2005-06-15
EP1539796B1 (en) 2007-02-14
AU2003253354A1 (en) 2004-02-09
SI1539796T1 (sl) 2007-06-30
DK1539796T3 (da) 2007-05-29

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