ES2078749T3 - Procedimiento para preparar sertralina. - Google Patents

Procedimiento para preparar sertralina.

Info

Publication number
ES2078749T3
ES2078749T3 ES92914143T ES92914143T ES2078749T3 ES 2078749 T3 ES2078749 T3 ES 2078749T3 ES 92914143 T ES92914143 T ES 92914143T ES 92914143 T ES92914143 T ES 92914143T ES 2078749 T3 ES2078749 T3 ES 2078749T3
Authority
ES
Spain
Prior art keywords
procedure
preparing sertraline
sertraline
formula
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES92914143T
Other languages
English (en)
Inventor
Michael Trevelyan Williams
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Application granted granted Critical
Publication of ES2078749T3 publication Critical patent/ES2078749T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/12—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
    • C07C233/14—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)

Abstract

LA INVENCION SE REFIERE A LA FORMA DE CIS-ESTEROISOMERICA SUSTANCIAL Y GEOMETRICAMENTE PURA DE UN COMPUESTO DE FORMULA (I) Y LA FORMA CIS-ESTEROISOMERICA SUSTANCIAL, GEOMETRICA Y OPTICAMENTE PURA DE UN COMPUESTO DE FORMULA (II) R1 ES H O ALQUILO C1-C4, JUNTO CON LOS PROCESOS PARA SU PREPARACION. LOS COMPUESTOS SON INTERMEDIOS PARA LA PREPARACION DE AGENTE ANTIDEPRESORES COMO SERTRALINA.
ES92914143T 1991-07-11 1992-07-03 Procedimiento para preparar sertralina. Expired - Lifetime ES2078749T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919114947A GB9114947D0 (en) 1991-07-11 1991-07-11 Process for preparing sertraline

Publications (1)

Publication Number Publication Date
ES2078749T3 true ES2078749T3 (es) 1995-12-16

Family

ID=10698170

Family Applications (1)

Application Number Title Priority Date Filing Date
ES92914143T Expired - Lifetime ES2078749T3 (es) 1991-07-11 1992-07-03 Procedimiento para preparar sertralina.

Country Status (14)

Country Link
US (1) US5463126A (es)
EP (1) EP0594666B1 (es)
JP (1) JP2566374B2 (es)
AT (1) ATE127779T1 (es)
CA (1) CA2109817C (es)
DE (1) DE69204840T2 (es)
DK (1) DK0594666T3 (es)
ES (1) ES2078749T3 (es)
FI (1) FI112210B (es)
GB (1) GB9114947D0 (es)
GR (1) GR3017766T3 (es)
IE (1) IE67822B1 (es)
PT (1) PT100672B (es)
WO (1) WO1993001162A1 (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777000B1 (fr) * 1998-04-01 2002-09-27 Catalys Procede de preparation de la sertraline racemique
IL132500A0 (en) 1998-10-29 2001-03-19 Pfizer Prod Inc Stereoselective microbial reduction of a racemic tetralone
WO2000032551A1 (en) * 1998-11-27 2000-06-08 Teva Pharmaceutical Industries Ltd. Sertraline hydrochloride polymorphs
US6500987B1 (en) * 1998-11-27 2002-12-31 Teva Pharmaceutical Industries Ltd. Sertraline hydrochloride polymorphs
RU2161851C1 (ru) * 1999-05-24 2001-01-10 Научно-производственное внедренческое предприятие "Феррогидродинамика" Электрическая машина
US6495721B1 (en) 1999-08-09 2002-12-17 Teva Pharmaceutical Industries Ltd. Sertraline hydrochloride Form II and methods for the preparation thereof
US20050119351A1 (en) * 1999-10-29 2005-06-02 Van Der Schaaf Paul A. Polymorphic forms of sertraline hydrochloride
TWI260315B (en) * 1999-10-29 2006-08-21 Ciba Sc Holding Ag Polymorphic forms of sertraline hydrochloride
US7442838B2 (en) * 1999-10-29 2008-10-28 Ciba Specialty Chemicals Corp. Polymorphic forms of sertraline hydrochloride
PT1248605E (pt) * 1999-12-21 2007-03-30 Teva Pharma Novos polimorfos de cloridrato de sertralina, processos para a sua preparação, composições que os contêm e métodos para a sua utilização
KR20070002101A (ko) * 2000-03-14 2007-01-04 테바 파마슈티컬 인더스트리즈 리미티드 (+)-시스-세르트랄린의 신규한 제조 방법
US6720003B2 (en) 2001-02-16 2004-04-13 Andrx Corporation Serotonin reuptake inhibitor formulations
WO2003093217A1 (en) * 2002-04-29 2003-11-13 Teva Pharmaceutical Industries Ltd. Process for preparation of polymorphic form ii of sertraline hydrochloride, pharmaceutical formulations and methods of administration thereof
US20060014838A1 (en) * 2004-07-14 2006-01-19 Sudhakar Valluri Process for converting trans-sertraline to cis-sertraline
KR20250034266A (ko) * 2023-09-01 2025-03-11 환인제약 주식회사 설트랄린 또는 이의 염을 포함하는 약학적 조성물

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4269870A (en) * 1974-05-13 1981-05-26 Cooper Industries, Inc. Solder flux and method
US4071489A (en) * 1976-03-08 1978-01-31 Rohm And Haas Company Coating compositions from dicyclopentenyl acrylate and/or methacrylate
JPS5592293A (en) * 1978-12-28 1980-07-12 Sanwa Kagaku Kogyo Kk Solid flux for soldering
US4536518A (en) * 1979-11-01 1985-08-20 Pfizer Inc. Antidepressant derivatives of cis-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine
JPS5910497A (ja) * 1982-07-12 1984-01-19 Hitachi Ltd フラックス
JPH0773795B2 (ja) * 1985-07-02 1995-08-09 太陽インキ製造株式会社 はんだ付用水洗性フラツクス組成物
US4882339A (en) * 1987-07-10 1989-11-21 Ciba-Geigy Corporation 4-Amino-substituted 1,2-dihydroxynaphthalene derivatives useful in inhibiting 5-lipoxygenase activity in mammals
US5071875A (en) * 1989-09-25 1991-12-10 Northwestern University Substituted 2-amidotetralins as melatonin agonists and antagonists

Also Published As

Publication number Publication date
DE69204840T2 (de) 1996-02-22
ATE127779T1 (de) 1995-09-15
PT100672B (pt) 1999-06-30
WO1993001162A1 (en) 1993-01-21
GR3017766T3 (en) 1996-01-31
IE67822B1 (en) 1996-05-01
FI940106A0 (fi) 1994-01-10
FI112210B (fi) 2003-11-14
PT100672A (pt) 1993-09-30
FI940106L (fi) 1994-01-10
JPH06509080A (ja) 1994-10-13
GB9114947D0 (en) 1991-08-28
US5463126A (en) 1995-10-31
DK0594666T3 (da) 1995-11-13
JP2566374B2 (ja) 1996-12-25
CA2109817C (en) 1999-08-31
EP0594666A1 (en) 1994-05-04
EP0594666B1 (en) 1995-09-13
IE922248A1 (en) 1993-01-13
DE69204840D1 (de) 1995-10-19

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