PT100672A - Processo para a preparacao de intermediarios de sertralina e compostos assim obtidos - Google Patents

Processo para a preparacao de intermediarios de sertralina e compostos assim obtidos

Info

Publication number
PT100672A
PT100672A PT100672A PT10067292A PT100672A PT 100672 A PT100672 A PT 100672A PT 100672 A PT100672 A PT 100672A PT 10067292 A PT10067292 A PT 10067292A PT 100672 A PT100672 A PT 100672A
Authority
PT
Portugal
Prior art keywords
preparation
pct
sertraline
compounds
intermediaries
Prior art date
Application number
PT100672A
Other languages
English (en)
Other versions
PT100672B (pt
Inventor
Michael Trevelyan Williams
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT100672A publication Critical patent/PT100672A/pt
Publication of PT100672B publication Critical patent/PT100672B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/01Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/12Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
    • C07C233/14Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a ring other than a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00Systems containing two condensed rings
    • C07C2602/02Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT100672A 1991-07-11 1992-07-09 Processo para a preparacao de intermediarios de sertralina e compostos assim obtidos PT100672B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919114947A GB9114947D0 (en) 1991-07-11 1991-07-11 Process for preparing sertraline

Publications (2)

Publication Number Publication Date
PT100672A true PT100672A (pt) 1993-09-30
PT100672B PT100672B (pt) 1999-06-30

Family

ID=10698170

Family Applications (1)

Application Number Title Priority Date Filing Date
PT100672A PT100672B (pt) 1991-07-11 1992-07-09 Processo para a preparacao de intermediarios de sertralina e compostos assim obtidos

Country Status (14)

Country Link
US (1) US5463126A (pt)
EP (1) EP0594666B1 (pt)
JP (1) JP2566374B2 (pt)
AT (1) ATE127779T1 (pt)
CA (1) CA2109817C (pt)
DE (1) DE69204840T2 (pt)
DK (1) DK0594666T3 (pt)
ES (1) ES2078749T3 (pt)
FI (1) FI112210B (pt)
GB (1) GB9114947D0 (pt)
GR (1) GR3017766T3 (pt)
IE (1) IE67822B1 (pt)
PT (1) PT100672B (pt)
WO (1) WO1993001162A1 (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777000B1 (fr) * 1998-04-01 2002-09-27 Catalys Procede de preparation de la sertraline racemique
IL132500A0 (en) 1998-10-29 2001-03-19 Pfizer Prod Inc Stereoselective microbial reduction of a racemic tetralone
ES2255320T3 (es) * 1998-11-27 2006-06-16 Teva Pharmaceutical Industries Ltd. Forma v clorhidrato de sertralina.
US6500987B1 (en) 1998-11-27 2002-12-31 Teva Pharmaceutical Industries Ltd. Sertraline hydrochloride polymorphs
US6495721B1 (en) * 1999-08-09 2002-12-17 Teva Pharmaceutical Industries Ltd. Sertraline hydrochloride Form II and methods for the preparation thereof
TWI260315B (en) 1999-10-29 2006-08-21 Ciba Sc Holding Ag Polymorphic forms of sertraline hydrochloride
US20050119351A1 (en) * 1999-10-29 2005-06-02 Van Der Schaaf Paul A. Polymorphic forms of sertraline hydrochloride
US7442838B2 (en) * 1999-10-29 2008-10-28 Ciba Specialty Chemicals Corp. Polymorphic forms of sertraline hydrochloride
JP4057295B2 (ja) * 1999-12-21 2008-03-05 テバ ファーマシューティカル インダストリーズ リミティド 新規塩酸セルトラリン多形体、それらを調製するための方法、それらを含有する組成物およびそれらを用いる方法
IL151691A0 (en) * 2000-03-14 2003-04-10 Teva Pharma Novel process for preparing (+)-cis-sertraline
US6720003B2 (en) 2001-02-16 2004-04-13 Andrx Corporation Serotonin reuptake inhibitor formulations
CA2483569A1 (en) * 2002-04-29 2003-11-13 Tamar Nidam Process for preparation of polymorphic form ii of sertraline hydrochloride, pharmaceutical formulations and methods of administration thereof
US20060014838A1 (en) * 2004-07-14 2006-01-19 Sudhakar Valluri Process for converting trans-sertraline to cis-sertraline

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4269870A (en) * 1974-05-13 1981-05-26 Cooper Industries, Inc. Solder flux and method
US4071489A (en) * 1976-03-08 1978-01-31 Rohm And Haas Company Coating compositions from dicyclopentenyl acrylate and/or methacrylate
JPS5592293A (en) * 1978-12-28 1980-07-12 Sanwa Kagaku Kogyo Kk Solid flux for soldering
US4536518A (en) * 1979-11-01 1985-08-20 Pfizer Inc. Antidepressant derivatives of cis-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine
JPS5910497A (ja) * 1982-07-12 1984-01-19 Hitachi Ltd フラックス
JPH0773795B2 (ja) * 1985-07-02 1995-08-09 太陽インキ製造株式会社 はんだ付用水洗性フラツクス組成物
US4882339A (en) * 1987-07-10 1989-11-21 Ciba-Geigy Corporation 4-Amino-substituted 1,2-dihydroxynaphthalene derivatives useful in inhibiting 5-lipoxygenase activity in mammals
US5071875A (en) * 1989-09-25 1991-12-10 Northwestern University Substituted 2-amidotetralins as melatonin agonists and antagonists

Also Published As

Publication number Publication date
PT100672B (pt) 1999-06-30
ATE127779T1 (de) 1995-09-15
CA2109817C (en) 1999-08-31
GB9114947D0 (en) 1991-08-28
FI112210B (fi) 2003-11-14
FI940106A0 (fi) 1994-01-10
DE69204840T2 (de) 1996-02-22
IE67822B1 (en) 1996-05-01
GR3017766T3 (en) 1996-01-31
IE922248A1 (en) 1993-01-13
US5463126A (en) 1995-10-31
EP0594666A1 (en) 1994-05-04
DE69204840D1 (de) 1995-10-19
JPH06509080A (ja) 1994-10-13
EP0594666B1 (en) 1995-09-13
ES2078749T3 (es) 1995-12-16
WO1993001162A1 (en) 1993-01-21
DK0594666T3 (da) 1995-11-13
JP2566374B2 (ja) 1996-12-25
FI940106A (fi) 1994-01-10

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Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19930507

FG3A Patent granted, date of granting

Effective date: 19990316

MM4A Annulment/lapse due to non-payment of fees, searched and examined patent

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20070917