EE200200425A - Selektiivsete PDE4 isosüümide inhibiitoritena kasulikud nikotiinamiidi bensokondenseerunud heterotsüklüülderivaadid - Google Patents

Selektiivsete PDE4 isosüümide inhibiitoritena kasulikud nikotiinamiidi bensokondenseerunud heterotsüklüülderivaadid

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Publication number
EE200200425A
EE200200425A EEP200200425A EEP200200425A EE200200425A EE 200200425 A EE200200425 A EE 200200425A EE P200200425 A EEP200200425 A EE P200200425A EE P200200425 A EEP200200425 A EE P200200425A EE 200200425 A EE200200425 A EE 200200425A
Authority
EE
Estonia
Prior art keywords
nicotinamide
inhibitors
useful
selective pde4
pde4 isozymes
Prior art date
Application number
EEP200200425A
Other languages
English (en)
Estonian (et)
Inventor
Marfat Anthony
James Chamber Robert
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of EE200200425A publication Critical patent/EE200200425A/xx

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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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EEP200200425A 2000-01-31 2001-01-30 Selektiivsete PDE4 isosüümide inhibiitoritena kasulikud nikotiinamiidi bensokondenseerunud heterotsüklüülderivaadid EE200200425A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17928400P 2000-01-31 2000-01-31
PCT/IB2001/000124 WO2001057036A1 (fr) 2000-01-31 2001-01-30 Derives benzocondenses heterocycliques de nicotinamide utiles comme inhibiteurs selectifs d'isozymes pde4

Publications (1)

Publication Number Publication Date
EE200200425A true EE200200425A (et) 2003-10-15

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200200425A EE200200425A (et) 2000-01-31 2001-01-30 Selektiivsete PDE4 isosüümide inhibiitoritena kasulikud nikotiinamiidi bensokondenseerunud heterotsüklüülderivaadid

Country Status (40)

Country Link
US (1) US7354941B2 (fr)
EP (1) EP1252158B1 (fr)
JP (1) JP3917863B2 (fr)
KR (1) KR20020072299A (fr)
CN (1) CN1404481A (fr)
AP (1) AP2002002589A0 (fr)
AR (1) AR027337A1 (fr)
AT (1) ATE293624T1 (fr)
AU (1) AU2700201A (fr)
BG (1) BG106852A (fr)
BR (1) BR0107964A (fr)
CA (1) CA2398182C (fr)
CO (1) CO5261634A1 (fr)
CZ (1) CZ20022410A3 (fr)
DE (1) DE60110205T2 (fr)
EA (1) EA004885B1 (fr)
EE (1) EE200200425A (fr)
ES (1) ES2238415T3 (fr)
GE (1) GEP20043302B (fr)
GT (1) GT200100022A (fr)
HN (1) HN2001000019A (fr)
HU (1) HUP0204262A2 (fr)
IL (1) IL150641A0 (fr)
IS (1) IS6421A (fr)
MA (1) MA26870A1 (fr)
MX (1) MXPA02007419A (fr)
NO (1) NO20023613L (fr)
NZ (1) NZ519547A (fr)
OA (1) OA12169A (fr)
PA (1) PA8511201A1 (fr)
PE (1) PE20011058A1 (fr)
PL (1) PL357995A1 (fr)
PT (1) PT1252158E (fr)
SK (1) SK10142002A3 (fr)
SV (1) SV2002000299A (fr)
TN (1) TNSN01020A1 (fr)
TR (1) TR200201880T2 (fr)
UY (1) UY26569A1 (fr)
WO (1) WO2001057036A1 (fr)
ZA (1) ZA200206033B (fr)

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Publication number Priority date Publication date Assignee Title
DE69942009D1 (de) * 1998-10-15 2010-03-25 Imp Innovations Ltd Verbindungen für die behandlung von gewichtsverlust
DE60110057T2 (de) * 2000-01-28 2005-09-08 Alza Corp., Mountain View Liposomen enthaltend eine eingeschlossene verbindung in übersattigter lösung
MXPA03002338A (es) * 2000-09-18 2003-09-10 Du Pont Piridinilamidas y piridinilimidas para uso como fungicidas.
WO2002060898A1 (fr) 2001-01-31 2002-08-08 Pfizer Products Inc. Derives amide acide de thiazolyle, oxazolyle, pyrrolyle et imidazolyle utilises en tant qu'inhibiteurs des isozymes pde4
IL156460A0 (en) 2001-01-31 2004-01-04 Pfizer Prod Inc Ether derivatives useful as inhibitors of pde4 isozymes
EP1355884A1 (fr) * 2001-01-31 2003-10-29 Pfizer Products Inc. Derives de biaryl nicotinamide utiles comme inhibiteurs d'isozymes de pde4
US7250518B2 (en) 2001-01-31 2007-07-31 Pfizer Inc. Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes
GB0118373D0 (en) * 2001-07-27 2001-09-19 Glaxo Group Ltd Novel therapeutic method
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