OA12169A - Nicotinamide benzofused-heterocyclyl derivatives useful as selective inhibitors of PDE4 isozymes. - Google Patents

Nicotinamide benzofused-heterocyclyl derivatives useful as selective inhibitors of PDE4 isozymes. Download PDF

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Publication number
OA12169A
OA12169A OA1200200229A OA1200200229A OA12169A OA 12169 A OA12169 A OA 12169A OA 1200200229 A OA1200200229 A OA 1200200229A OA 1200200229 A OA1200200229 A OA 1200200229A OA 12169 A OA12169 A OA 12169A
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OA
OAPI
Prior art keywords
formula
benzo
hydroxy
nicotinamide
methyl
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OA1200200229A
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English (en)
Inventor
Anthony Marfat
Robert James Chambers
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Pfizer Prod Inc
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Publication of OA12169A publication Critical patent/OA12169A/en

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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OA1200200229A 2000-01-31 2001-01-30 Nicotinamide benzofused-heterocyclyl derivatives useful as selective inhibitors of PDE4 isozymes. OA12169A (en)

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US17928400P 2000-01-31 2000-01-31

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OA12169A true OA12169A (en) 2006-05-08

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EP (1) EP1252158B1 (fr)
JP (1) JP3917863B2 (fr)
KR (1) KR20020072299A (fr)
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AP (1) AP2002002589A0 (fr)
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US7417038B1 (en) * 1998-10-15 2008-08-26 Imperial Innovations Limited Methods of treating cachexia
KR100782891B1 (ko) * 2000-01-28 2007-12-06 알자 코포레이션 과포화 용액으로 포획된 화합물을 포함하는 리포좀
WO2002022583A2 (fr) * 2000-09-18 2002-03-21 E. I. Du Pont De Nemours And Company Pyridinyl-amides et pyridinyl-imides utilisés comme fongicides
CA2436535A1 (fr) * 2001-01-31 2002-08-08 Prizer Products Inc. Derives de biaryl nicotinamide utiles comme inhibiteurs d'isozymes de pde4
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