HN2001000019A - Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4. - Google Patents
Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4.Info
- Publication number
- HN2001000019A HN2001000019A HN2001000019A HN2001000019A HN2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A
- Authority
- HN
- Honduras
- Prior art keywords
- pde4
- isozimas
- benzocondensada
- heterociclico
- nicotinamide
- Prior art date
Links
- 101100296720 Dictyostelium discoideum Pde4 gene Proteins 0.000 title abstract 2
- 101100082610 Plasmodium falciparum (isolate 3D7) PDEdelta gene Proteins 0.000 title abstract 2
- 229940124639 Selective inhibitor Drugs 0.000 title abstract 2
- DFPAKSUCGFBDDF-UHFFFAOYSA-N Nicotinamide Chemical class NC(=O)C1=CC=CN=C1 DFPAKSUCGFBDDF-UHFFFAOYSA-N 0.000 title 1
- 208000006673 asthma Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 230000000241 respiratory effect Effects 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract
LA PRESENTE INVENCION SE REFIERE TAMBIEN AL USO DE INHIBIDORES SELECTIVOS DE LAS PDE4 PARA UN MEJOR TRATAMIENTO TERAPEUTICO DE UNA SERIE DE ENFERMEDADES Y CONDICIONES INFLAMATORIAS, RESPIRATORIAS Y ALERGICAS, PERO ESPECIALMENTE PARA EL TRATAMIENTO DEL ASMA
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US17928400P | 2000-01-31 | 2000-01-31 |
Publications (1)
Publication Number | Publication Date |
---|---|
HN2001000019A true HN2001000019A (es) | 2001-09-06 |
Family
ID=22655931
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HN2001000019A HN2001000019A (es) | 2000-01-31 | 2001-06-30 | Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4. |
Country Status (40)
Country | Link |
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US (1) | US7354941B2 (es) |
EP (1) | EP1252158B1 (es) |
JP (1) | JP3917863B2 (es) |
KR (1) | KR20020072299A (es) |
CN (1) | CN1404481A (es) |
AP (1) | AP2002002589A0 (es) |
AR (1) | AR027337A1 (es) |
AT (1) | ATE293624T1 (es) |
AU (1) | AU2700201A (es) |
BG (1) | BG106852A (es) |
BR (1) | BR0107964A (es) |
CA (1) | CA2398182C (es) |
CO (1) | CO5261634A1 (es) |
CZ (1) | CZ20022410A3 (es) |
DE (1) | DE60110205T2 (es) |
EA (1) | EA004885B1 (es) |
EE (1) | EE200200425A (es) |
ES (1) | ES2238415T3 (es) |
GE (1) | GEP20043302B (es) |
GT (1) | GT200100022A (es) |
HN (1) | HN2001000019A (es) |
HU (1) | HUP0204262A2 (es) |
IL (1) | IL150641A0 (es) |
IS (1) | IS6421A (es) |
MA (1) | MA26870A1 (es) |
MX (1) | MXPA02007419A (es) |
NO (1) | NO20023613L (es) |
NZ (1) | NZ519547A (es) |
OA (1) | OA12169A (es) |
PA (1) | PA8511201A1 (es) |
PE (1) | PE20011058A1 (es) |
PL (1) | PL357995A1 (es) |
PT (1) | PT1252158E (es) |
SK (1) | SK10142002A3 (es) |
SV (1) | SV2002000299A (es) |
TN (1) | TNSN01020A1 (es) |
TR (1) | TR200201880T2 (es) |
UY (1) | UY26569A1 (es) |
WO (1) | WO2001057036A1 (es) |
ZA (1) | ZA200206033B (es) |
Families Citing this family (43)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK1121111T3 (da) * | 1998-10-15 | 2010-05-31 | Imp Innovations Ltd | Forbindelser til behandling af vægttab |
MXPA02007320A (es) * | 2000-01-28 | 2004-07-30 | Alza Corp | Liposomas conteniendo un compuesto atrapado en solucion supersaturada. |
AU2002211233A1 (en) | 2000-09-18 | 2002-03-26 | E.I. Du Pont De Nemours And Company | Pyridinyl amides and imides for use as fungicides |
WO2002060896A1 (en) | 2001-01-31 | 2002-08-08 | Pfizer Products Inc. | Ether derivatives useful as inhibitors of pde4 isozymes |
US7250518B2 (en) | 2001-01-31 | 2007-07-31 | Pfizer Inc. | Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes |
CA2436535A1 (en) | 2001-01-31 | 2002-08-08 | Prizer Products Inc. | Nicotinamide biaryl derivatives useful as inhibitors of pde4 isozymes |
PL365443A1 (en) | 2001-01-31 | 2005-01-10 | Pfizer Products Inc. | Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes |
GB0118373D0 (en) * | 2001-07-27 | 2001-09-19 | Glaxo Group Ltd | Novel therapeutic method |
US20050014762A1 (en) * | 2001-09-19 | 2005-01-20 | Rolf Beume | Combination |
BR0212606A (pt) * | 2001-09-19 | 2004-08-17 | Altana Pharma Ag | Combinação |
IS7221A (is) * | 2001-11-15 | 2004-04-15 | Memory Pharmaceuticals Corporation | Hringlaga adenosínmónófosfat fosfódíesterasa 4D7 ísóform og aðferðir til notkunar þeirra |
CA2475712C (en) | 2002-02-11 | 2009-11-24 | Simon Bailey | Nicotinamide derivatives useful as pde4 inhibitors |
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